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Antitrypanosomal activity against Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream by acid phosphatase method
Assay data:1 Active, 2 Tested
SummaryCompounds, ActivePubMed Citation
Inhibition of topoisomerase in Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as enzyme -DNA cleavable complex at 50 uM relative to DMSO
Assay data:2 Tested
SummaryPubMed Citation
Inhibition of topoisomerase in Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as enzyme-DNA cleavable complex at 50 uM (RvB = 2.2 +/- 0.05%)
Binding affinity to plasmid DNA assessed as DNA unwinding in presence of vaccinia virus topoisomerase 1B by electrophoresis
Antitrypanosomal activity against Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as decrease in topoisomerase 2mt level at 0-120 uM
Assay data:2 Active, 2 Tested
Antitrypanosomal activity against Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as decrease in topoisomerase 2mt level at 0-100 uM
Antitrypanosomal activity against Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as decrease in topoisomerase 1Amt level at 0-120 uM
Antitrypanosomal activity against Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as decrease in topoisomerase 1Amt level at 0-100 uM
Inhibition of mitochondrion topoisomerase 1A in Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as protection of linerarizd minicircle from exonuclase 3 at 63 uM
Inhibition of mitochondrion topoisomerase 1A in Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as protection of linerarizd minicircle from exonuclase 3 at 25.5 uM
Inhibition of mitochondrion topoisomerase 1A in Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as protection of linerarizd minicircle from lambda exonuclase at 63 uM
Inhibition of mitochondrion topoisomerase 1A in Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as protection of linerarizd minicircle from lambda exonuclase at 25.5 uM
Inhibition of mitochondrion topoisomerase 1A in Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as increase in protein-sensitive linear DNA forms at 60-100 uM
Inhibition of mitochondrion topoisomerase 1A in Trypanosoma brucei brucei MiTat 1.2 strain 427 bloodstream assessed as increase in protein-sensitive linear DNA forms at 0-40 uM
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