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Agonist activity at human human NOD1 expressed in HEK-Blue NOD1 reporter cells at 2 uM by colorimetry based SEAP assay
Assay data:27 Tested
SummaryPubMed CitationRelated BioAssays by Target
Agonist activity at NOD1 in HEK-Blue hNOD1 cells assessed as increase in NFkappaB activation at 10 uM incubated for 18 hrs by SEAP-based spectrophotometry analysis
Assay data:2 Tested
Agonist activity at NOD1 in HEK-Blue hNOD2 cells assessed as increase in NFkappaB transactivation-mediated SEAP activity measured after 18 hrs by spectrophotometric method
Assay data:39 Tested
Inhibition of human NOD1 in human THP-1 cells assessed as inhibition of lauroyl-gamma-D-Glu-mDAP stimulated RIP2 phoshorylation measured after 90 mins by western blot method
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of human NOD1 in human THP-1 cells assessed as inhibition of lauroyl-gamma-D-Glu-mDAP stimulated reduction in IkappaBalpha expression measured after 90 mins by western blot method
Inhibition of human NOD1 in human THP-1 cells assessed as inhibition of lauroyl-gamma-D-Glu-mDAP stimulated p38 phosphorylation measured after 90 mins by western blot method
Inhibition of human NOD1 in human THP-1 cells assessed as inhibition of lauroyl-gamma-D-Glu-mDAP stimulated JNK phoshorylation measured after 90 mins by western blot method
Inhibition of human NOD1 in human THP-1 cells assessed as inhibition of lauroyl-gamma-D-Glu-mDAP stimulated ERK phosphorylation measured after 90 mins by western blot method
Inhibition of human NOD1 in human THP-1 cells assessed as inhibition of lauroyl-gamma-D-Glu-mDAP stimulated IL-6 m-RNA expression measured after 150 mins by Real time quantitative reverse transcriptase PCR method
Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed by stimulated with lauroyl-gamma-D-Glu-mDAP for 20 hrs by spectrophotometer method
Assay data:18 Active, 1 Activity ≤ 1 µM, 45 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as reduction in secreted alkaline phosphatase reporter activity at 10 uM preincubated for 3 hrs followed by stimulated with lauroyl-gamma-D-Glu-mDAP for 20 hrs by spectrophotometer method
Assay data:45 Tested
Antagonist activity at NOD1 in human THP-1 cells assessed as reduction in C12-iE-DAP-induced IL-8 secretion at 20 uM preincubated for 1 hr followed by C12-iE-DAP stimulation and measured after 20 hrs by ELISA
Assay data:4 Active, 4 Tested
Antagonist activity at human NOD1 expressed in HEK293 cells assessed as reduction in C12-iE-DAP-induced NF-kappaB activation preincubated for 1 hr followed by C12-iE-DAP stimulation and measured after 18 hrs by SEAP reporter gene based spectrophotometric analysis
Assay data:6 Active, 1 Activity ≤ 1 µM, 19 Tested
Antagonist activity at human NOD1 expressed in HEK293 cells assessed as reduction in C12-iE-DAP-induced NF-kappaB activation at 10 uM preincubated for 1 hr followed by C12-iE-DAP stimulation and measured after 18 hrs by SEAP reporter gene based spectrophotometric analysis
Assay data:9 Active, 15 Tested
Agonist activity at human NOD1 expressed in HEK293 cells assessed as increase in NF-kappaB activation up to 10 uM incubated for 24 hrs by quanti-blue SEAP reporter gene assay
Assay data:1 Tested
Antagonist activity at recombinant human NOD1 expressed in HEK293 cells assessed as inhibition of C12-iE-DAP-induced IL8 release measured after 24 hrs by HTRF assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested
Antagonist activity at NOD1 in human THP-1 cells assessed as inhibition of C12-iE-DAP-induced IL8 mRNA expression preincubated for 1 hr followed by C12-iE-DAP addition and measured after 90 mins by qRT-PCR analysis
Antagonist activity at NOD1 in human THP-1 cells assessed as inhibition of C12-iE-DAP-induced TNFalpha mRNA expression preincubated for 1 hr followed by C12-iE-DAP addition and measured after 90 mins by qRT-PCR analysis
Antagonist activity at NOD1 in human THP-1 cells assessed as inhibition of C12-iE-DAP-induced IL6 mRNA expression preincubated for 1 hr followed by C12-iE-DAP addition and measured after 90 mins by qRT-PCR analysis
Antagonist activity at NOD1 in human THP-1 cells assessed as inhibition of C12-iE-DAP-induced IkappaBalpha degradation at 1 to 10 uM preincubated for 1 hr followed by C12-iE-DAP addition and measured after 30 mins by Western blot analysis
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