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hMMP14 assay from US Patent US10550100: "5-[3-[piperzin-1-yl]-3-oxo-propyl]-imidazolidine-2,4-dione derivatives as ADAMTS 4 and 5 inhibitors for treating E.G. osteoarthritis"
Assay data:40 Activity ≤ 1 µM, 40 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
hMMP13 assay from US Patent US10550100: "5-[3-[piperzin-1-yl]-3-oxo-propyl]-imidazolidine-2,4-dione derivatives as ADAMTS 4 and 5 inhibitors for treating E.G. osteoarthritis"
Assay data:81 Activity ≤ 1 µM, 81 Tested
hTACE assay from US Patent US10550100: "5-[3-[piperzin-1-yl]-3-oxo-propyl]-imidazolidine-2,4-dione derivatives as ADAMTS 4 and 5 inhibitors for treating E.G. osteoarthritis"
Assay data:36 Active, 90 Activity ≤ 1 µM, 90 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
hADAMTS-6 Assay from US Patent US10550100: "5-[3-[piperzin-1-yl]-3-oxo-propyl]-imidazolidine-2,4-dione derivatives as ADAMTS 4 and 5 inhibitors for treating E.G. osteoarthritis"
Assay data:82 Active, 114 Activity ≤ 1 µM, 114 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Depositor
hADAMTS-5 assay from US Patent US10550100: "5-[3-[piperzin-1-yl]-3-oxo-propyl]-imidazolidine-2,4-dione derivatives as ADAMTS 4 and 5 inhibitors for treating E.G. osteoarthritis"
Assay data:38 Active, 108 Activity ≤ 1 µM, 108 Tested
Rat ADAMTS-5 assay from US Patent US10550100: "5-[3-[piperzin-1-yl]-3-oxo-propyl]-imidazolidine-2,4-dione derivatives as ADAMTS 4 and 5 inhibitors for treating E.G. osteoarthritis"
Assay data:14 Active, 17 Activity ≤ 1 µM, 17 Tested
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