My Bibliography

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Woong Sub Byun, Zhe Zhuang, Anna P. Hnatiuk, Cyrus Jin, Zixuan Jiang, Kheewoong Baek, Evelyn Chao, Katherine A. Donovan, Eric S. Fischer, Mark Mercola, Nathanael S. Gray. Discovery of BRD9 Molecular Glue Degraders That Spare Cardiomyocytes. Journal of the American Chemical Society. 2025 October. doi: 10.1021/jacs.5c09857.

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Katrina Warner, Moritz Hunkeler, Kheewoong Baek, Anna Schmoker, Shourya S. Roy Burman, Daan Overwijn, Cyrus Jin, Katherine A. Donovan, Eric S. Fischer. Structural ubiquitin contributes to K48 linkage specificity of the HECT ligase Tom1. Cell Reports. 2025 May. doi: 10.1016/j.celrep.2025.115688.

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Joseph D. Hurley, Irina Shlosman, Megha Lakshminarayan, Ziyuan Zhao, Hong Yue, Radosław P. Nowak, Eric S. Fischer, Andrew C. Kruse. Decoding Protein–Peptide Interactions Using a Large, Target-Agnostic Yeast Surface Display Library. ACS Chemical Biology. 2025 September. doi: 10.1021/acschembio.5c00265.

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Binita Shah, Moritz Hunkeler, Ariana Bratt, Hong Yue, Isabella Jaen Maisonet, Eric S. Fischer, Sara J. Buhrlage. Structural basis of VCP-VCPIP1-p47 ternary complex in Golgi maintenance. Nature Communications. 2025 August. doi: 10.1038/s41467-025-63161-3.

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Tian Qiu, Zhe Zhuang, Woong Sub Byun, Zuzanna Kozicka, Kheewoong Baek, Jianing Zhong, Abby M. Thornhill, Julia K. Ryan, Katherine A. Donovan, Eric S. Fischer, Benjamin L. Ebert, Nathanael S. Gray. Development of FBXO22 Degraders and the Recruitment Ligand 2-Pyridinecarboxyaldehyde (2-PCA). Journal of the American Chemical Society. 2025 December. doi: 10.1021/jacs.5c14141.

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Słabicki M, Park J, Nowak RP, Roy Burman SS, Pellman J, Zou C, Razumkov H, Carreiro J, Rastogi S, Goldstein A, Nagiec MM, Donovan KA, Che J, Hunkeler M, Geng Q, Hsu CL, Lakshminarayan M, Shu C, Zon RL, Kozicka Z, Park PMC, Tsai JM, Yoon H, Jones LH, Sperling AS, Gray NS, Fischer ES, Ebert BL. Expanding the druggable zinc-finger proteome defines properties of drug-induced degradation. Mol Cell. 2025 Aug 21;85(16):3184-3201.e14. doi: 10.1016/j.molcel.2025.07.019. PubMed PMID: 40845806; PubMed Central PMCID: PMC12458990.

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Qiu T, Zhuang Z, Byun WS, Kozicka Z, Baek K, Zhong J, Thornhill AM, Ryan JK, Donovan KA, Fischer ES, Ebert BL, Gray NS. Development of Degraders and 2-pyridinecarboxyaldehyde (2-PCA) as a recruitment Ligand for FBXO22. bioRxiv. 2025 Aug 20;. doi: 10.1101/2025.08.19.671158. PubMed PMID: 40894587; PubMed Central PMCID: PMC12393450.

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Zhuang Z, Byun WS, Kozicka Z, Donovan KA, Dwyer BG, Thornhill AM, Jones HM, Jiang Z, Zhu X, Fischer ES, Thomä NH, Gray NS. Rational Design of CDK12/13 and BRD4 Molecular Glue Degraders. Angew Chem Int Ed Engl. 2025 Sep 15;64(38):e202508427. doi: 10.1002/anie.202508427. Epub 2025 Aug 7. PubMed PMID: 40626960; PubMed Central PMCID: PMC12831537.

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Kamaraj R, Mejdrová I, Krutakova M, Smutny T, Škach K, Dohnalova K, Smutna L, Nellore DSS, Dusek J, Chalupsky K, Hricová J, Kronenberger T, Stahl A, Templin M, Braeuning A, Nencka R, Pavek P. Discovery of PXR Antagonist MI891 and PXR Degrader MI1013 and Their Roles in Hepatic Gene Regulation. J Med Chem. 2025 Jul 24;68(14):14271-14299. doi: 10.1021/acs.jmedchem.4c03134. Epub 2025 Jul 12. PubMed PMID: 40650588; PubMed Central PMCID: PMC12305494.

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Zhai S, Honin I, Schäker-Hübner L, Hanl M, Jacobi L, Dressler F, Pieńkowska DE, König P, Gerhartz J, Voget R, Bendas G, Gütschow M, Meissner F, Burckhardt BB, Nowak RP, Steinebach C, Hansen FK. Development and Characterization of the First Selective Class IIb Histone Deacetylase Degraders. J Med Chem. 2025 Jul 10;68(13):13793-13821. doi: 10.1021/acs.jmedchem.5c00674. Epub 2025 Jun 18. PubMed PMID: 40532131; PubMed Central PMCID: PMC12245577.

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Coomar S, Gasser JA, Słabicki M, Donovan KA, Fischer ES, Ebert BL, Gillingham D, Thomä NH. Niclosamide: CRL4(AMBRA1) mediated degradation of cyclin D1 following mitochondrial membrane depolarization. RSC Med Chem. 2025 Jul 16;16(7):3049-3057. doi: 10.1039/d5md00054h. eCollection 2025 Jul 16. PubMed PMID: 40337304; PubMed Central PMCID: PMC12054360.

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Gui F, Jiang B, Jiang J, He Z, Tsujino T, Takai T, Arai S, Pana C, Köllermann J, Bradshaw GA, Eisert R, Kalocsay M, Fassl A, Balk SP, Kibel AS, Jia L. Acute BRCAness induction and AR pathway blockage through CDK12/7/9 degradation enhances PARP inhibitor sensitivity in prostate cancer. Sci Adv. 2025 Apr 25;11(17):eadu0847. doi: 10.1126/sciadv.adu0847. Epub 2025 Apr 23. PubMed PMID: 40267193; PubMed Central PMCID: PMC12017310.

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Monsen PJ, Bommi PV, Grigorescu AA, Lauing KL, Mao Y, Berardi P, Zhai L, Ojo O, Penco-Campillo M, Koch T, Egozi M, Jha S, Dunne SF, Jiang H, Song G, Zhang F, Kregel S, Vaziri-Gohar A, Fanning SW, Sanchez-Gomez P, Allen JM, Yamini B, Lukas RV, Wainwright DA, Schiltz GE. Rational Design and Optimization of a Potent IDO1 Proteolysis Targeting Chimera (PROTAC). J Med Chem. 2025 Feb 27;68(4):4961-4987. doi: 10.1021/acs.jmedchem.5c00026. Epub 2025 Feb 13. PubMed PMID: 39946350; PubMed Central PMCID: PMC11874035.

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Geng Q, Jiang Z, Byun WS, Donovan KA, Zhuang Z, Jiang F, Jones HM, Razumkov H, Tang MT, Sarott RC, Fischer ES, Corsello SM, Hinshaw SM, Gray NS. Development of Potent and Selective CK1α Molecular Glue Degraders. J Med Chem. 2025 Feb 13;68(3):3180-3196. doi: 10.1021/acs.jmedchem.4c02415. Epub 2025 Jan 28. PubMed PMID: 39873536; PubMed Central PMCID: PMC12861308.

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Feller F, Honin I, Miranda M, Weber H, Henze S, Hanl M, Hansen FK. Development of the First-in-Class FEM1B-Recruiting Histone Deacetylase Degraders. J Med Chem. 2025 Jan 23;68(2):1824-1843. doi: 10.1021/acs.jmedchem.4c02569. Epub 2025 Jan 13. PubMed PMID: 39804678; PubMed Central PMCID: PMC11780399.

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Yingpeng Liu, Radosław P. Nowak, Jianwei Che, Katherine A. Donovan, Fidel Huerta, Hu Liu, Rebecca J. Metivier, Eric S. Fischer, Lyn H. Jones. Development of sulfonyl fluoride chemical probes to advance the discovery of cereblon modulators. RSC Medicinal Chemistry. 2024. doi: 10.1039/D3MD00652B.

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Han-Yuan Liu, Zhengnian Li, Theresia Reindl, Zhixiang He, Xueer Qiu, Ryan P. Golden, Katherine A. Donovan, Adam Bailey, Eric S. Fischer, Tinghu Zhang, Nathanael S. Gray, Priscilla L. Yang. Broad-spectrum activity against mosquito-borne flaviviruses achieved by a targeted protein degradation mechanism. Nature Communications. 2024 June. doi: 10.1038/s41467-024-49161-9.

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Jonathan M. Tsai, Radosław P. Nowak, Benjamin L. Ebert, Eric S. Fischer. Targeted protein degradation: from mechanisms to clinic. Nature Reviews Molecular Cell Biology. 2024 September. doi: 10.1038/s41580-024-00729-9.

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Hai-Tsang Huang, Ryan J. Lumpkin, Ryan W. Tsai, Shuyao Su, Xu Zhao, Yuan Xiong, James Chen, Nada Mageed, Katherine A. Donovan, Eric S. Fischer, William R. Sellers. Ubiquitin-specific proximity labeling for the identification of E3 ligase substrates. Nature Chemical Biology. 2024 September. doi: 10.1038/s41589-024-01590-9.

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Binita Shah, Moritz Hunkeler, Ariana Bratt, Hong Yue, Isabella Jaen Maisonet, Eric S. Fischer, Sara J. Buhrlage. Ternary complex formation of VCP, VCPIP1 and p47 facilitates Golgi reassembly. 2024 October. DOI: 10.1101/2024.10.01.616120.

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Razumkov H, Jiang Z, Baek K, You I, Geng Q, Donovan KA, Tang MT, Metivier RJ, Mageed N, Seo P, Li Z, Byun WS, Hinshaw SM, Sarott RC, Fischer ES, Gray NS. Discovery of CRBN-Dependent WEE1 Molecular Glue Degraders from a Multicomponent Combinatorial Library. J Am Chem Soc. 2024 Nov 20;146(46):31433-31443. doi: 10.1021/jacs.4c06127. Epub 2024 Nov 5. PubMed PMID: 39499896; PubMed Central PMCID: PMC11800961.

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Baek K, Metivier RJ, Roy Burman SS, Bushman JW, Yoon H, Lumpkin RJ, Abeja DM, Lakshminarayan M, Yue H, Ojeda S, Verano AL, Gray NS, Donovan KA, Fischer ES. Unveiling the hidden interactome of CRBN molecular glues with chemoproteomics. bioRxiv. 2024 Oct 4;. doi: 10.1101/2024.09.11.612438. PubMed PMID: 39314457; PubMed Central PMCID: PMC11419069.

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Zhuang Z, Byun WS, Kozicka Z, Dwyer BG, Donovan KA, Jiang Z, Jones HM, Abeja DM, Nix MN, Zhong J, Słabicki M, Fischer ES, Ebert BL, Gray NS. Discovery of electrophilic degraders that exploit S(N)Ar chemistry. bioRxiv. 2024 Sep 27;. doi: 10.1101/2024.09.25.615094. PubMed PMID: 39386645; PubMed Central PMCID: PMC11463635.

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Hassan MM, Li YD, Ma MW, Teng M, Byun WS, Puvar K, Lumpkin R, Sandoval B, Rutter JC, Jin CY, Wang MY, Xu S, Schmoker AM, Cheong H, Groendyke BJ, Qi J, Fischer ES, Ebert BL, Gray NS. Exploration of the tunability of BRD4 degradation by DCAF16 trans-labelling covalent glues. Eur J Med Chem. 2024 Dec 5;279:116904. doi: 10.1016/j.ejmech.2024.116904. Epub 2024 Sep 24. PubMed PMID: 39341093; PubMed Central PMCID: PMC11960843.

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Li YD, Ma MW, Hassan MM, Hunkeler M, Teng M, Puvar K, Rutter JC, Lumpkin RJ, Sandoval B, Jin CY, Schmoker AM, Ficarro SB, Cheong H, Metivier RJ, Wang MY, Xu S, Byun WS, Groendyke BJ, You I, Sigua LH, Tavares I, Zou C, Tsai JM, Park PMC, Yoon H, Majewski FC, Sperling HT, Marto JA, Qi J, Nowak RP, Donovan KA, Słabicki M, Gray NS, Fischer ES, Ebert BL. Template-assisted covalent modification underlies activity of covalent molecular glues. Nat Chem Biol. 2024 Dec;20(12):1640-1649. doi: 10.1038/s41589-024-01668-4. Epub 2024 Jul 29. PubMed PMID: 39075252; PubMed Central PMCID: PMC11582070.

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Ji W, Du G, Jiang J, Lu W, Mills CE, Yuan L, Jiang F, He Z, Bradshaw GA, Chung M, Jiang Z, Byun WS, Hinshaw SM, Zhang T, Gray NS. Discovery of bivalent small molecule degraders of cyclin-dependent kinase 7 (CDK7). Eur J Med Chem. 2024 Oct 5;276:116613. doi: 10.1016/j.ejmech.2024.116613. Epub 2024 Jun 27. PubMed PMID: 39004018; PubMed Central PMCID: PMC11316633.

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Radko-Juettner S, Yue H, Myers JA, Carter RD, Robertson AN, Mittal P, Zhu Z, Hansen BS, Donovan KA, Hunkeler M, Rosikiewicz W, Wu Z, McReynolds MG, Roy Burman SS, Schmoker AM, Mageed N, Brown SA, Mobley RJ, Partridge JF, Stewart EA, Pruett-Miller SM, Nabet B, Peng J, Gray NS, Fischer ES, Roberts CWM. Author Correction: Targeting DCAF5 suppresses SMARCB1-mutant cancer by stabilizing SWI/SNF. Nature. 2024 May;629(8012):E12. doi: 10.1038/s41586-024-07402-3. PubMed PMID: 38684813.

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Radko-Juettner S, Yue H, Myers JA, Carter RD, Robertson AN, Mittal P, Zhu Z, Hansen BS, Donovan KA, Hunkeler M, Rosikiewicz W, Wu Z, McReynolds MG, Roy Burman SS, Schmoker AM, Mageed N, Brown SA, Mobley RJ, Partridge JF, Stewart EA, Pruett-Miller SM, Nabet B, Peng J, Gray NS, Fischer ES, Roberts CWM. Targeting DCAF5 suppresses SMARCB1-mutant cancer by stabilizing SWI/SNF. Nature. 2024 Apr;628(8007):442-449. doi: 10.1038/s41586-024-07250-1. Epub 2024 Mar 27. PubMed PMID: 38538798; PubMed Central PMCID: PMC11184678.

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Mercer JAM, DeCarlo SJ, Roy Burman SS, Sreekanth V, Nelson AT, Hunkeler M, Chen PJ, Donovan KA, Kokkonda P, Tiwari PK, Shoba VM, Deb A, Choudhary A, Fischer ES, Liu DR. Continuous evolution of compact protein degradation tags regulated by selective molecular glues. Science. 2024 Mar 15;383(6688):eadk4422. doi: 10.1126/science.adk4422. Epub 2024 Mar 15. PubMed PMID: 38484051; PubMed Central PMCID: PMC11203266.

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Erickson EC, You I, Perry G, Dugourd A, Donovan KA, Crafter C, Johannes JW, Williamson S, Moss JI, Ros S, Ziegler RE, Barry ST, Fischer ES, Gray NS, Madsen RR, Toker A. Multiomic profiling of breast cancer cells uncovers stress MAPK-associated sensitivity to AKT degradation. Sci Signal. 2024 Feb 27;17(825):eadf2670. doi: 10.1126/scisignal.adf2670. Epub 2024 Feb 27. PubMed PMID: 38412255; PubMed Central PMCID: PMC10949348.

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Wang L, Shi S, Unterreiner A, Kapetanovic R, Ghosh S, Sanchez J, Aslani S, Xiong Y, Hsu CL, Donovan KA, Farady CJ, Fischer ES, Bornancin F, Matthias P. HDAC6/aggresome processing pathway importance for inflammasome formation is context-dependent. J Biol Chem. 2024 Feb;300(2):105638. doi: 10.1016/j.jbc.2024.105638. Epub 2024 Jan 8. PubMed PMID: 38199570; PubMed Central PMCID: PMC10850954.

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Moritz Hunkeler, Cyrus Y. Jin, Eric S. Fischer. Structures of BIRC6-client complexes provide a mechanism of SMAC-mediated release of caspases. Science. 2023 March. doi: 10.1126/science.ade5750.

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Alexander Hanzl, Eleonora Barone, Sophie Bauer, Hong Yue, Radosław P. Nowak, Elisa Hahn, Eugenia V. Pankevich, Anna Koren, Stefan Kubicek, Eric S. Fischer, Georg E. Winter. E3-Specific Degrader Discovery by Dynamic Tracing of Substrate Receptor Abundance. Journal of the American Chemical Society. 2023 January. doi: 10.1021/jacs.2c10784.

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Longlong Wang, Adeline Unterreiner, Ronan Kapetanovic, Selma Aslani, Yuan Xiong, Katherine A. Donovan, Christopher J. Farady, Eric S. Fischer, Frédéric Bornancin, Patrick Matthias. HDAC6/aggresome processing pathway importance for inflammasome formation is context dependent. 2023 August. DOI: 10.1101/2023.08.15.553363.

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Radosław P. Nowak, Leah Ragosta, Fidel Huerta, Hu Liu, Scott B. Ficarro, Justin T. Cruite, Rebecca J. Metivier, Katherine A. Donovan, Jarrod A. Marto, Eric S. Fischer, Breanna L. Zerfas, Lyn H. Jones. Development of a covalent cereblon-based PROTAC employing a fluorosulfate warhead. RSC Chemical Biology. 2023. doi: 10.1039/D3CB00103B.

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Justin T. Cruite, Radosław P. Nowak, Katherine A. Donovan, Scott B. Ficarro, Huang Huang, Hu Liu, Yingpeng Liu, Jarrod A. Marto, Rebecca J. Metivier, Eric S. Fischer, Lyn H. Jones. Covalent Stapling of the Cereblon Sensor Loop Histidine Using Sulfur-Heterocycle Exchange. ACS Medicinal Chemistry Letters. 2023 November. doi: 10.1021/acsmedchemlett.3c00371.

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Nguyen TM, Sreekanth V, Deb A, Kokkonda P, Tiwari PK, Donovan KA, Shoba V, Chaudhary SK, Mercer JAM, Lai S, Sadagopan A, Jan M, Fischer ES, Liu DR, Ebert BL, Choudhary A. Proteolysis-targeting chimeras with reduced off-targets. Nat Chem. 2024 Feb;16(2):218-228. doi: 10.1038/s41557-023-01379-8. Epub 2023 Dec 18. PubMed PMID: 38110475; PubMed Central PMCID: PMC10913580.

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Ji W, Byun WS, Lu W, Zhu X, Donovan KA, Dwyer BG, Che J, Yuan L, Abulaiti X, Corsello SM, Fischer ES, Zhang T, Gray NS. Proteomics-Based Discovery of First-in-Class Chemical Probes for Programmed Cell Death Protein 2 (PDCD2). Angew Chem Int Ed Engl. 2023 Oct 23;62(43):e202308292. doi: 10.1002/anie.202308292. Epub 2023 Sep 15. PubMed PMID: 37658265; PubMed Central PMCID: PMC10592021.

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Kozicka Z, Suchyta DJ, Focht V, Kempf G, Petzold G, Jentzsch M, Zou C, Di Genua C, Donovan KA, Coomar S, Cigler M, Mayor-Ruiz C, Schmid-Burgk JL, Häussinger D, Winter GE, Fischer ES, Słabicki M, Gillingham D, Ebert BL, Thomä NH. Design principles for cyclin K molecular glue degraders. Nat Chem Biol. 2024 Jan;20(1):93-102. doi: 10.1038/s41589-023-01409-z. Epub 2023 Sep 7. PubMed PMID: 37679459; PubMed Central PMCID: PMC10746543.

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Hatcher JM, Zwirek M, Sarhan AR, Vatsan PS, Tonelli F, Alessi DR, Davies P, Gray NS. Development of a highly potent and selective degrader of LRRK2. Bioorg Med Chem Lett. 2023 Oct 1;94:129449. doi: 10.1016/j.bmcl.2023.129449. Epub 2023 Aug 15. PubMed PMID: 37591317; PubMed Central PMCID: PMC11837620.

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Xiao Y, Hale S, Awasthee N, Meng C, Zhang X, Liu Y, Ding H, Huo Z, Lv D, Zhang W, He M, Zheng G, Liao D. HDAC3 and HDAC8 PROTAC dual degrader reveals roles of histone acetylation in gene regulation. Cell Chem Biol. 2023 Nov 16;30(11):1421-1435.e12. doi: 10.1016/j.chembiol.2023.07.010. Epub 2023 Aug 11. PubMed PMID: 37572669; PubMed Central PMCID: PMC10802846.

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Kim Y, Seo P, Jeon E, You I, Hwang K, Kim N, Tse J, Bae J, Choi HS, Hinshaw SM, Gray NS, Sim T. Targeted kinase degradation via the KLHDC2 ubiquitin E3 ligase. Cell Chem Biol. 2023 Nov 16;30(11):1414-1420.e5. doi: 10.1016/j.chembiol.2023.07.008. Epub 2023 Aug 10. PubMed PMID: 37567174; PubMed Central PMCID: PMC10839117.

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Koide E, Mohardt ML, Doctor ZM, Yang A, Hao M, Donovan KA, Kuismi CC, Nelson AJ, Abell K, Aguiar M, Che J, Stokes MP, Zhang T, Aguirre AJ, Fischer ES, Gray NS, Jiang B, Nabet B. Development and Characterization of Selective FAK Inhibitors and PROTACs with In Vivo Activity. Chembiochem. 2023 Oct 4;24(19):e202300141. doi: 10.1002/cbic.202300141. Epub 2023 Jul 24. PubMed PMID: 37088717; PubMed Central PMCID: PMC10590827.

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Monda JK, Ge X, Hunkeler M, Donovan KA, Ma MW, Jin CY, Leonard M, Fischer ES, Bennett EJ. HAPSTR1 localizes HUWE1 to the nucleus to limit stress signaling pathways. Cell Rep. 2023 May 30;42(5):112496. doi: 10.1016/j.celrep.2023.112496. Epub 2023 May 9. PubMed PMID: 37167062; PubMed Central PMCID: PMC10279472.

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Gao Y, Jiang B, Kim H, Berberich MJ, Che J, Donovan KA, Hatcher JM, Huerta F, Kwiatkowski NP, Liu Y, Liuni PP, Metivier RJ, Murali VK, Nowak RP, Zhang T, Fischer ES, Gray NS, Jones LH. Catalytic Degraders Effectively Address Kinase Site Mutations in EML4-ALK Oncogenic Fusions. J Med Chem. 2023 Apr 27;66(8):5524-5535. doi: 10.1021/acs.jmedchem.2c01864. Epub 2023 Apr 10. PubMed PMID: 37036171; PubMed Central PMCID: PMC11827123.

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Jiang B, Weinstock DM, Donovan KA, Sun HW, Wolfe A, Amaka S, Donaldson NL, Wu G, Jiang Y, Wilcox RA, Fischer ES, Gray NS, Wu W. ITK degradation to block T cell receptor signaling and overcome therapeutic resistance in T cell lymphomas. Cell Chem Biol. 2023 Apr 20;30(4):383-393.e6. doi: 10.1016/j.chembiol.2023.03.007. Epub 2023 Apr 3. PubMed PMID: 37015223; PubMed Central PMCID: PMC10151063.

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Teng M, Jiang J, Wang ES, Geng Q, Toenjes ST, Donovan KA, Mageed N, Yue H, Nowak RP, Wang J, Manz TD, Fischer ES, Cantley LC, Gray NS. Targeting the Dark Lipid Kinase PIP4K2C with a Potent and Selective Binder and Degrader. Angew Chem Int Ed Engl. 2023 Apr 24;62(18):e202302364. doi: 10.1002/anie.202302364. Epub 2023 Mar 27. PubMed PMID: 36898968; PubMed Central PMCID: PMC10150580.

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Perner F, Stein EM, Wenge DV, Singh S, Kim J, Apazidis A, Rahnamoun H, Anand D, Marinaccio C, Hatton C, Wen Y, Stone RM, Schaller D, Mowla S, Xiao W, Gamlen HA, Stonestrom AJ, Persaud S, Ener E, Cutler JA, Doench JG, McGeehan GM, Volkamer A, Chodera JD, Nowak RP, Fischer ES, Levine RL, Armstrong SA, Cai SF. MEN1 mutations mediate clinical resistance to menin inhibition. Nature. 2023 Mar;615(7954):913-919. doi: 10.1038/s41586-023-05755-9. Epub 2023 Mar 15. PubMed PMID: 36922589; PubMed Central PMCID: PMC10157896.

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Yue H, Nowak RP, Overwijn D, Payne NC, Fischinger S, Atyeo C, Lam EC, St Denis K, Brais LK, Konishi Y, Sklavenitis-Pistofidis R, Baden LR, Nilles EJ, Karlson EW, Yu XG, Li JZ, Woolley AE, Ghobrial IM, Meyerhardt JA, Balazs AB, Alter G, Mazitschek R, Fischer ES. Diagnostic TR-FRET assays for detection of antibodies in patient samples. Cell Rep Methods. 2023 Mar 27;3(3):100421. doi: 10.1016/j.crmeth.2023.100421. eCollection 2023 Mar 27. PubMed PMID: 37056371; PubMed Central PMCID: PMC10088089.

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Hunkeler M, Jin CY, Fischer ES. Structures of BIRC6-client complexes provide a mechanism of SMAC-mediated release of caspases. Science. 2023 Mar 17;379(6637):1105-1111. doi: 10.1126/science.ade5750. Epub 2023 Feb 9. PubMed PMID: 36758104.