Similar articles for PMID: 28389916

Year	Number of Results
1991	1
1992	1
1997	1
1999	2
2003	3
2004	2
2005	5
2006	2
2007	2
2008	6
2009	7
2010	7
2011	11
2012	10
2013	7
2014	10
2015	12
2016	13
2017	10
2018	14
2019	15
2020	13
2021	14
2022	8
2023	4
2024	0

1

A direct label-free MALDI-TOF mass spectrometry based assay for the characterization of inhibitors of protein lysine methyltransferases.

Guitot K, Drujon T, Burlina F, Sagan S, Beaupierre S, Pamlard O, Dodd RH, Guillou C, Bolbach G, Sachon E, Guianvarc'h D. Guitot K, et al. Anal Bioanal Chem. 2017 Jun;409(15):3767-3777. doi: 10.1007/s00216-017-0319-5. Epub 2017 Apr 7. Anal Bioanal Chem. 2017. PMID: 28389916

2

Label-free measurement of histone lysine methyltransferases activity by matrix-assisted laser desorption/ionization time-of-flight mass spectrometry.

Guitot K, Scarabelli S, Drujon T, Bolbach G, Amoura M, Burlina F, Jeltsch A, Sagan S, Guianvarc'h D. Guitot K, et al. Anal Biochem. 2014 Jul 1;456:25-31. doi: 10.1016/j.ab.2014.04.006. Epub 2014 Apr 15. Anal Biochem. 2014. PMID: 24747023

3

Lysine Possesses the Optimal Chain Length for Histone Lysine Methyltransferase Catalysis.

Temimi AHKA, Reddy YV, White PB, Guo H, Qian P, Mecinović J. Temimi AHKA, et al. Sci Rep. 2017 Nov 23;7(1):16148. doi: 10.1038/s41598-017-16128-4. Sci Rep. 2017. PMID: 29170487 Free PMC article.

4

Structure-Activity Relationship Studies on (R)-PFI-2 Analogues as Inhibitors of Histone Lysine Methyltransferase SETD7.

Lenstra DC, Damen E, Leenders RGG, Blaauw RH, Rutjes FPJT, Wegert A, Mecinović J. Lenstra DC, et al. ChemMedChem. 2018 Jul 18;13(14):1405-1413. doi: 10.1002/cmdc.201800242. Epub 2018 Jun 25. ChemMedChem. 2018. PMID: 29869845

5

(R)-PFI-2 is a potent and selective inhibitor of SETD7 methyltransferase activity in cells.

Barsyte-Lovejoy D, Li F, Oudhoff MJ, Tatlock JH, Dong A, Zeng H, Wu H, Freeman SA, Schapira M, Senisterra GA, Kuznetsova E, Marcellus R, Allali-Hassani A, Kennedy S, Lambert JP, Couzens AL, Aman A, Gingras AC, Al-Awar R, Fish PV, Gerstenberger BS, Roberts L, Benn CL, Grimley RL, Braam MJ, Rossi FM, Sudol M, Brown PJ, Bunnage ME, Owen DR, Zaph C, Vedadi M, Arrowsmith CH. Barsyte-Lovejoy D, et al. Proc Natl Acad Sci U S A. 2014 Sep 2;111(35):12853-8. doi: 10.1073/pnas.1407358111. Epub 2014 Aug 18. Proc Natl Acad Sci U S A. 2014. PMID: 25136132 Free PMC article.

6

Development of homogeneous nonradioactive methyltransferase and demethylase assays targeting histone H3 lysine 4.

Gauthier N, Caron M, Pedro L, Arcand M, Blouin J, Labonté A, Normand C, Paquet V, Rodenbrock A, Roy M, Rouleau N, Beaudet L, Padrós J, Rodriguez-Suarez R. Gauthier N, et al. J Biomol Screen. 2012 Jan;17(1):49-58. doi: 10.1177/1087057111416659. Epub 2011 Sep 21. J Biomol Screen. 2012. PMID: 21940714

7

Design and synthesis of peptide-MCA substrates for a novel assay of histone methyltransferases and their inhibitors.

Chi H, Takemoto Y, Nsiama TK, Kato T, Nishino N, Ito A, Yoshida M. Chi H, et al. Bioorg Med Chem. 2014 Feb 15;22(4):1268-75. doi: 10.1016/j.bmc.2014.01.011. Epub 2014 Jan 21. Bioorg Med Chem. 2014. PMID: 24486204

8

Kinetic isotope effects reveal early transition state of protein lysine methyltransferase SET8.

Linscott JA, Kapilashrami K, Wang Z, Senevirathne C, Bothwell IR, Blum G, Luo M. Linscott JA, et al. Proc Natl Acad Sci U S A. 2016 Dec 27;113(52):E8369-E8378. doi: 10.1073/pnas.1609032114. Epub 2016 Dec 9. Proc Natl Acad Sci U S A. 2016. PMID: 27940912 Free PMC article.

9

High-throughput screening with nucleosome substrate identifies small-molecule inhibitors of the human histone lysine methyltransferase NSD2.

Coussens NP, Kales SC, Henderson MJ, Lee OW, Horiuchi KY, Wang Y, Chen Q, Kuznetsova E, Wu J, Chakka S, Cheff DM, Cheng KC, Shinn P, Brimacombe KR, Shen M, Simeonov A, Lal-Nag M, Ma H, Jadhav A, Hall MD. Coussens NP, et al. J Biol Chem. 2018 Aug 31;293(35):13750-13765. doi: 10.1074/jbc.RA118.004274. Epub 2018 Jun 26. J Biol Chem. 2018. PMID: 29945974 Free PMC article.

10

Extending matrix-assisted laser desorption/ionization triple quadrupole mass spectrometry enzyme screening assays to targets with small molecule substrates.

Rathore R, Corr JJ, Lebre DT, Seibel WL, Greis KD. Rathore R, et al. Rapid Commun Mass Spectrom. 2009 Oct 30;23(20):3293-300. doi: 10.1002/rcm.4248. Rapid Commun Mass Spectrom. 2009. PMID: 19757451

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