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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
1924 1
1925 1
1937 2
1938 1
1940 1
1941 1
1943 1
1945 65
1946 202
1947 209
1948 174
1949 138
1950 191
1951 208
1952 234
1953 263
1954 284
1955 315
1956 322
1957 386
1958 480
1959 445
1960 268
1961 252
1962 352
1963 513
1964 605
1965 434
1966 558
1967 577
1968 673
1969 742
1970 721
1971 752
1972 779
1973 760
1974 819
1975 759
1976 738
1977 882
1978 857
1979 938
1980 941
1981 932
1982 922
1983 877
1984 918
1985 880
1986 874
1987 874
1988 848
1989 875
1990 954
1991 939
1992 930
1993 940
1994 1021
1995 1008
1996 1133
1997 1294
1998 1470
1999 1548
2000 1828
2001 1817
2002 2062
2003 2288
2004 2556
2005 2938
2006 3164
2007 3484
2008 3667
2009 3774
2010 4045
2011 4137
2012 4447
2013 4366
2014 4317
2015 4079
2016 3963
2017 3894
2018 3821
2019 3727
2020 4168
2021 3560
2022 2947
2023 2509
2024 1011

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Search Results

109,885 results

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Page 1
Thiazoles and Thiazolidinones as COX/LOX Inhibitors.
Liaras K, Fesatidou M, Geronikaki A. Liaras K, et al. Molecules. 2018 Mar 18;23(3):685. doi: 10.3390/molecules23030685. Molecules. 2018. PMID: 29562646 Free PMC article. Review.
In search for new drugs to avoid side effects, while maintaining high potency over inflammation, scientists turned their interest to the synthesis of dual COX/LOX inhibitors, which could provide numerous therapeutic advantages in terms of anti-inflammatory activity, improved gast …
In search for new drugs to avoid side effects, while maintaining high potency over inflammation, scientists turned their interest to the syn …
Thiazoles and thiazolidinones as antioxidants.
Geronikaki AA, Pitta EP, Liaras KS. Geronikaki AA, et al. Curr Med Chem. 2013;20(36):4460-80. doi: 10.2174/09298673113209990143. Curr Med Chem. 2013. PMID: 23834182 Review.
The aim of this review is to describe recent developments in the study of the antioxidant activity of thiazole and thiazolidinone derivatives, which are the core structure in a variety of pharmaceuticals with a broad spectrum of biological activity and their role in preven …
The aim of this review is to describe recent developments in the study of the antioxidant activity of thiazole and thiazolidinone der …
Synthetic and Medicinal Perspective of Fused-Thiazoles as Anticancer Agents.
Pawar S, Kumar K, Gupta MK, Rawal RK. Pawar S, et al. Anticancer Agents Med Chem. 2021;21(11):1379-1402. doi: 10.2174/1871520620666200728133017. Anticancer Agents Med Chem. 2021. PMID: 32723259 Review.
Fused thiazole scaffold containing drugs are available in market as a promising group of anticancer agents. ...Various synthetic strategies for fused thiazole are also summarized in this article. Novel thiazole and its fused congener showed anticancer activit …
Fused thiazole scaffold containing drugs are available in market as a promising group of anticancer agents. ...Various synthetic stra …
A Comprehensive Review on the Therapeutic Versatility of Imidazo [2,1-b]thiazoles.
Shareef MA, Khan I, Babu BN, Kamal A. Shareef MA, et al. Curr Med Chem. 2020;27(40):6864-6887. doi: 10.2174/0929867326666190729152440. Curr Med Chem. 2020. PMID: 31362648 Review.
BACKGROUND: Imidazo[2,1-b]thiazole, a well-known fused five-membered hetrocycle is one of the most promising and versatile moieties in the area of medicinal chemistry. Derivatives of imidazo[2,1-b]thiazole have been investigated for the development of new derivative …
BACKGROUND: Imidazo[2,1-b]thiazole, a well-known fused five-membered hetrocycle is one of the most promising and versatile moieties i …
4-Adamantyl-(2-(arylidene)hydrazinyl)thiazoles as potential antidiabetic agents: experimental and docking studies.
Iqbal Y, Akhtar T, Haroon M, Mehmood H, Nizami T, Tahir E, Ehsan M. Iqbal Y, et al. Future Med Chem. 2023 Apr;15(7):599-613. doi: 10.4155/fmc-2023-0010. Epub 2023 May 4. Future Med Chem. 2023. PMID: 37140092
The compounds 4-adamantyl-(2-(4-chlorobenzylidene)hydrazinyl)thiazole and 4-adamantyl-(2-(2-chlorobenzylidene)hydrazinyl)thiazole showed the highest potency. The compounds 4-adamantyl-(2-(4-bromobenzylidene)hydrazinyl)thiazole and 4-adamantyl-(2-(2-hydroxyben …
The compounds 4-adamantyl-(2-(4-chlorobenzylidene)hydrazinyl)thiazole and 4-adamantyl-(2-(2-chlorobenzylidene)hydrazinyl)thiazole …
One-Pot Synthesis of Novel Thiazoles as Potential Anti-Cancer Agents.
Sayed AR, Gomha SM, Taher EA, Muhammad ZA, El-Seedi HR, Gaber HM, Ahmed MM. Sayed AR, et al. Drug Des Devel Ther. 2020 Apr 3;14:1363-1375. doi: 10.2147/DDDT.S221263. eCollection 2020. Drug Des Devel Ther. 2020. PMID: 32308369 Free PMC article.
BACKGROUND: Thiazole and thiosemicarbazone derivatives are known to have potential anticancer activity with a mechanism of action related to inhibition of matrix metallo-proteinases, kinases and anti-apoptotic BCL2 family proteins. MATERIALS AND METHODS: A novel three seri …
BACKGROUND: Thiazole and thiosemicarbazone derivatives are known to have potential anticancer activity with a mechanism of action rel …
Camalexin.
Glawischnig E. Glawischnig E. Phytochemistry. 2007 Feb;68(4):401-6. doi: 10.1016/j.phytochem.2006.12.005. Epub 2007 Jan 10. Phytochemistry. 2007. PMID: 17217970 Review.
Camalexin (3-thiazol-2'-yl-indole) is the characteristic phytoalexin of Arabidopsis thaliana, which is induced by a great variety of plant pathogens. ...
Camalexin (3-thiazol-2'-yl-indole) is the characteristic phytoalexin of Arabidopsis thaliana, which is induced by a great variety of …
Thiazole Ring-A Biologically Active Scaffold.
Petrou A, Fesatidou M, Geronikaki A. Petrou A, et al. Molecules. 2021 May 25;26(11):3166. doi: 10.3390/molecules26113166. Molecules. 2021. PMID: 34070661 Free PMC article. Review.
BACKGROUND: Thiazole is a good pharmacophore nucleus due to its various pharmaceutical applications. ...RESULTS: Nearly 124 research articles were found, critically analyzed, and arranged regarding the synthesis and biological activities of thiazoles derivatives in …
BACKGROUND: Thiazole is a good pharmacophore nucleus due to its various pharmaceutical applications. ...RESULTS: Nearly 124 research …
Thiazole Compounds as Antiviral Agents: An Update.
Singh IP, Gupta S, Kumar S. Singh IP, et al. Med Chem. 2020;16(1):4-23. doi: 10.2174/1573406415666190614101253. Med Chem. 2020. PMID: 31203807 Review.
Thiazole containing compounds (thiazoles) have shown various biological activities like antioxidant, analgesic, antibacterial, anticancer, antiallergic, antihypertensive, antiinflammatory, antimalarial, antifungal and antipsychotic. ...Further filters were applied f …
Thiazole containing compounds (thiazoles) have shown various biological activities like antioxidant, analgesic, antibacterial, …
Organolithium-mediated diversification of peptide thiazoles.
Deng S, Taunton J. Deng S, et al. Org Lett. 2005 Jan 20;7(2):299-301. doi: 10.1021/ol047660j. Org Lett. 2005. PMID: 15646982
[Reaction: see text] We report a one-step, racemization-free method for the diversification of peptide thiazoles via direct lithiation of the thiazole ring. The method is compatible with N-Boc, N-trityl, carboxylic ester, and carboxamide protecting groups and has be …
[Reaction: see text] We report a one-step, racemization-free method for the diversification of peptide thiazoles via direct lithiatio …
109,885 results
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