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Items: 1 to 20 of 50

1.

Characterization of AN317, a novel selective agonist of α6β2-containing nicotinic acetylcholine receptors.

Sandager-Nielsen K, Ahring PK, Klein J, van Hout M, Thaneshwaran S, Dos Santos AB, Jacobsen TA, Amrutkar DV, Peters D, Jensen AA, Kohlmeier KA, Christophersen P, Dyhring T.

Biochem Pharmacol. 2019 Dec 27:113786. doi: 10.1016/j.bcp.2019.113786. [Epub ahead of print]

PMID:
31887288
2.

In vivo characterization of a novel norepinephrine transporter PET tracer [18F]NS12137 in adult and immature Sprague-Dawley rats.

López-Picón FR, Kirjavainen AK, Forsback S, Takkinen JS, Peters D, Haaparanta-Solin M, Solin O.

Theranostics. 2019 Jan 1;9(1):11-19. doi: 10.7150/thno.29740. eCollection 2019.

3.

Synthesis and radiofluorination of novel fluoren-9-one based derivatives for the imaging of α7 nicotinic acetylcholine receptor with PET.

Teodoro R, Scheunemann M, Wenzel B, Peters D, Deuther-Conrad W, Brust P.

Bioorg Med Chem Lett. 2018 May 15;28(9):1471-1475. doi: 10.1016/j.bmcl.2018.03.081. Epub 2018 Mar 29.

PMID:
29628323
4.

18F-labeled norepinephrine transporter tracer [18F]NS12137: radiosynthesis and preclinical evaluation.

Kirjavainen AK, Forsback S, López-Picón FR, Marjamäki P, Takkinen J, Haaparanta-Solin M, Peters D, Solin O.

Nucl Med Biol. 2018 Jan;56:39-46. doi: 10.1016/j.nucmedbio.2017.10.005. Epub 2017 Oct 24.

PMID:
29172120
5.

Tos-Nos-Mos: Synthesis of different aryl sulfonate precursors for the radiosynthesis of the alpha7 nicotinic acetylcholine receptor radioligand [(18)F]NS14490.

Rötering S, Scheunemann M, Günther R, Löser R, Hiller A, Dan Peters, Brust P, Fischer S, Steinbach J.

Appl Radiat Isot. 2016 Aug;114:57-62. doi: 10.1016/j.apradiso.2016.04.028. Epub 2016 Apr 28.

PMID:
27183376
6.

[¹¹C]NS9531, [¹¹C]NS9762 and [¹¹C]NS6417, specific SERT tracers: pre-clinical evaluation in pigs and optimization of synthesis conditions using [¹¹C]methyl triflate.

Dam JH, Bender D, Peters D, Någren K.

Nucl Med Biol. 2016 Jan;43(1):42-51. doi: 10.1016/j.nucmedbio.2015.10.004. Epub 2015 Oct 21.

PMID:
26702786
7.

A Promising PET Tracer for Imaging of α₇ Nicotinic Acetylcholine Receptors in the Brain: Design, Synthesis, and in Vivo Evaluation of a Dibenzothiophene-Based Radioligand.

Teodoro R, Scheunemann M, Deuther-Conrad W, Wenzel B, Fasoli FM, Gotti C, Kranz M, Donat CK, Patt M, Hillmer A, Zheng MQ, Peters D, Steinbach J, Sabri O, Huang Y, Brust P.

Molecules. 2015 Oct 9;20(10):18387-421. doi: 10.3390/molecules201018387.

8.

Radiosynthesis and in vitro validation of (3)H-NS14492 as a novel high affinity alpha7 nicotinic receptor radioligand.

Magnussen JH, Ettrup A, Donat CK, Peters D, Pedersen MH, Knudsen GM, Mikkelsen JD.

Eur J Pharmacol. 2015 Sep 5;762:35-41. doi: 10.1016/j.ejphar.2015.04.036. Epub 2015 May 1.

PMID:
25941084
9.

Engineered α4β2 nicotinic acetylcholine receptors as models for measuring agonist binding and effect at the orthosteric low-affinity α4-α4 interface.

Ahring PK, Olsen JA, Nielsen EØ, Peters D, Pedersen MH, Rohde LA, Kastrup JS, Shahsavar A, Indurthi DC, Chebib M, Gajhede M, Balle T.

Neuropharmacology. 2015 May;92:135-45. doi: 10.1016/j.neuropharm.2014.12.035. Epub 2015 Jan 13.

PMID:
25595102
10.

A high-yield automated radiosynthesis of the alpha-7 nicotinic receptor radioligand [18F]NS10743.

Teodoro R, Wenzel B, Oh-Nishi A, Fischer S, Peters D, Suhara T, Deuther-Conrad W, Brust P.

Appl Radiat Isot. 2015 Jan;95:76-84. doi: 10.1016/j.apradiso.2014.09.016. Epub 2014 Oct 8.

PMID:
25464181
11.

Imaging of α7 nicotinic acetylcholine receptors in brain and cerebral vasculature of juvenile pigs with [(18)F]NS14490.

Rötering S, Deuther-Conrad W, Cumming P, Donat CK, Scheunemann M, Fischer S, Xiong G, Steinbach J, Peters D, Sabri O, Bucerius J, Brust P.

EJNMMI Res. 2014 Aug 5;4:43. doi: 10.1186/s13550-014-0043-5. eCollection 2014.

12.

[11C]NS8880, a promising PET radiotracer targeting the norepinephrine transporter.

Vase KH, Peters D, Nielsen EØ, Alstrup AK, Bender D.

Nucl Med Biol. 2014 Oct;41(9):758-64. doi: 10.1016/j.nucmedbio.2014.06.004. Epub 2014 Jun 25.

PMID:
25127515
13.

One dentist's story: 'the future I never expected'.

Peters D.

J Mich Dent Assoc. 2014 Apr;96(4):40, 44-6. No abstract available.

PMID:
24968614
14.

Two distinct allosteric binding sites at α4β2 nicotinic acetylcholine receptors revealed by NS206 and NS9283 give unique insights to binding activity-associated linkage at Cys-loop receptors.

Olsen JA, Kastrup JS, Peters D, Gajhede M, Balle T, Ahring PK.

J Biol Chem. 2013 Dec 13;288(50):35997-6006. doi: 10.1074/jbc.M113.498618. Epub 2013 Oct 29.

15.

Biophysical and pharmacological characterization of α6-containing nicotinic acetylcholine receptors expressed in HEK293 cells.

Rasmussen AH, Strøbæk D, Dyhring T, Jensen ML, Peters D, Grunnet M, Timmermann DB, Ahring PK.

Brain Res. 2014 Jan 13;1542:1-11. doi: 10.1016/j.brainres.2013.10.024. Epub 2013 Oct 21.

PMID:
24157862
16.

Structural analysis of the positive AMPA receptor modulators CX516 and Me-CX516 in complex with the GluA2 ligand-binding domain.

Krintel C, Harpsøe K, Zachariassen LG, Peters D, Frydenvang K, Pickering DS, Gajhede M, Kastrup JS.

Acta Crystallogr D Biol Crystallogr. 2013 Sep;69(Pt 9):1645-52. doi: 10.1107/S0907444913011839. Epub 2013 Aug 15.

PMID:
23999288
17.

A combined α7 nicotinic acetylcholine receptor agonist and monoamine reuptake inhibitor, NS9775, represents a novel profile with potential benefits in emotional and cognitive disturbances.

Andreasen JT, Redrobe JP, Nielsen EØ, Christensen JK, Olsen GM, Peters D.

Neuropharmacology. 2013 Oct;73:183-91. doi: 10.1016/j.neuropharm.2013.04.060. Epub 2013 Jun 4.

PMID:
23748055
18.

Radiosynthesis and first evaluation in mice of [(18)F]NS14490 for molecular imaging of α7 nicotinic acetylcholine receptors.

Rötering S, Scheunemann M, Fischer S, Hiller A, Peters D, Deuther-Conrad W, Brust P.

Bioorg Med Chem. 2013 May 1;21(9):2635-42. doi: 10.1016/j.bmc.2013.02.018. Epub 2013 Feb 22.

PMID:
23507153
19.

Molecular determinants of subtype-selective efficacies of cytisine and the novel compound NS3861 at heteromeric nicotinic acetylcholine receptors.

Harpsøe K, Hald H, Timmermann DB, Jensen ML, Dyhring T, Nielsen EØ, Peters D, Balle T, Gajhede M, Kastrup JS, Ahring PK.

J Biol Chem. 2013 Jan 25;288(4):2559-70. doi: 10.1074/jbc.M112.436337. Epub 2012 Dec 10.

20.

Enantiomerically pure (1S,5R) and racemic 3-(1-benzothiophen-2-yl)-8-azoniabicyclo[3.2.1]oct-2-ene acetate.

Frøstrup B, Peters D, Bond AD.

Acta Crystallogr C. 2012 Aug;68(Pt 8):o298-301. doi: 10.1107/S0108270112030569. Epub 2012 Jul 13.

PMID:
22850855

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