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Items: 1 to 20 of 49

1.

Analytical method for simultaneously measuring ex vivo drug receptor occupancy and dissociation rate: application to (R)-dimethindene occupancy of central histamine H1 receptors.

Malany S, Hernandez LM, Smith WF, Crowe PD, Hoare SR.

J Recept Signal Transduct Res. 2009;29(2):84-93. doi: 10.1080/10799890902721339.

PMID:
19308787
2.

Pharmacologic methods for identification of receptors.

Tallarida RJ.

Life Sci. 1988;43(26):2169-76. Review.

PMID:
2850427
4.

[Molecular imaging of histamine receptors in the human brain].

Tashiro M, Yanai K.

Brain Nerve. 2007 Mar;59(3):221-31. Review. Japanese.

PMID:
17370648
5.

[Mutagenesis of the human histamine H1 receptor and design of new antihistamine agents].

Differding E, Gillard M, Moguilevsky N, Varsalona F, Noyer M, Daliers J, Goldstein S, Neuwels M, Lassoie MA, Guillaume JP, Bascour M, Bollen A, Hénichart JP.

J Pharm Belg. 1996 May-Jun;51(3):155-60. Review. French.

PMID:
8778348
6.
7.

The pharmacological basis of receptor binding.

Schütz W.

Wien Klin Wochenschr. 1991;103(15):438-42. Review.

PMID:
1656614
8.

In vitro receptor binding assays: general methods and considerations.

Bigott-Hennkens HM, Dannoon S, Lewis MR, Jurisson SS.

Q J Nucl Med Mol Imaging. 2008 Sep;52(3):245-53. Epub 2008 May 13. Review.

9.

Kinetic versus allosteric mechanisms to explain insurmountable antagonism and delayed ligand dissociation.

Vauquelin G, Szczuka A.

Neurochem Int. 2007 Oct;51(5):254-60. Epub 2007 May 21. Review.

PMID:
17606314
10.

Measuring drug-related receptor occupancy with positron emission tomography.

Passchier J, Gee A, Willemsen A, Vaalburg W, van Waarde A.

Methods. 2002 Jul;27(3):278-86. Review.

PMID:
12183116
11.

Molecular properties and signalling pathways of the histamine H1 receptor.

Smit MJ, Hoffmann M, Timmerman H, Leurs R.

Clin Exp Allergy. 1999 Jul;29 Suppl 3:19-28. Review.

PMID:
10444208
13.

Two-point kinetic experiments to quantify allosteric effects on radioligand dissociation.

Kostenis E, Mohr K.

Trends Pharmacol Sci. 1996 Aug;17(8):280-3. Review.

PMID:
8810873
14.

Positron emission tomography evaluation of sedative properties of antihistamines.

Yanai K, Zhang D, Tashiro M, Yoshikawa T, Naganuma F, Harada R, Nakamura T, Shibuya K, Okamura N.

Expert Opin Drug Saf. 2011 Jul;10(4):613-22. doi: 10.1517/14740338.2011.562889. Epub 2011 Apr 27. Review.

PMID:
21521134
15.
16.

[Histamine receptors and antagonists. New interesting views].

Naess K.

Tidsskr Nor Laegeforen. 1974 Aug 10;94(21-22):1333-4. Review. Norwegian. No abstract available.

PMID:
4153213
17.

The role of receptor binding in drug discovery.

Sweetnam PM, Caldwell L, Lancaster J, Bauer C Jr, McMillan B, Kinnier WJ, Price CH.

J Nat Prod. 1993 Apr;56(4):441-55. Review.

PMID:
8496700
18.

Studying neurotransmitter receptors: binding and biological assays.

Richelson E.

Monogr Neural Sci. 1984;10:4-19. Review. No abstract available.

PMID:
6321972
19.

[Structure of histamine H1 receptor].

Shimamura T.

Seikagaku. 2012 Sep;84(9):772-6. Review. Japanese. No abstract available.

PMID:
23198586
20.

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