Similar articles for PMID: 8978852

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1

Discovery of 1,5-benzodiazepines with peripheral cholecystokinin (CCK-A) receptor agonist activity (II): Optimization of the C3 amino substituent.

Hirst GC, Aquino C, Birkemo L, Croom DK, Dezube M, Dougherty RW Jr, Ervin GN, Grizzle MK, Henke B, James MK, Johnson MF, Momtahen T, Queen KL, Sherrill RG, Szewczyk J, Willson TM, Sugg EE. Hirst GC, et al. J Med Chem. 1996 Dec 20;39(26):5236-45. doi: 10.1021/jm9601664. J Med Chem. 1996. PMID: 8978852

2

Discovery of 1,5-benzodiazepines with peripheral cholecystokinin (CCK-A) receptor agonist activity. 1. Optimization of the agonist "trigger".

Aquino CJ, Armour DR, Berman JM, Birkemo LS, Carr RA, Croom DK, Dezube M, Dougherty RW Jr, Ervin GN, Grizzle MK, Head JE, Hirst GC, James MK, Johnson MF, Miller LJ, Queen KL, Rimele TJ, Smith DN, Sugg EE. Aquino CJ, et al. J Med Chem. 1996 Jan 19;39(2):562-9. doi: 10.1021/jm950626d. J Med Chem. 1996. PMID: 8558528

3

Optimization of 3-(1H-indazol-3-ylmethyl)-1,5-benzodiazepines as potent, orally active CCK-A agonists.

Henke BR, Aquino CJ, Birkemo LS, Croom DK, Dougherty RW Jr, Ervin GN, Grizzle MK, Hirst GC, James MK, Johnson MF, Queen KL, Sherrill RG, Sugg EE, Suh EM, Szewczyk JW, Unwalla RJ, Yingling J, Willson TM. Henke BR, et al. J Med Chem. 1997 Aug 15;40(17):2706-25. doi: 10.1021/jm970265x. J Med Chem. 1997. PMID: 9276016

4

Modification of receptor selectivity and functional activity in cholecystokinin peptoid ligands.

Dezube M, Sugg EE, Birkemo LS, Croom DK, Dougherty RW Jr, Ervin GN, Grizzle MK, James MK, Johnson MF, Mosher JT, et al. Dezube M, et al. J Med Chem. 1995 Aug 18;38(17):3384-90. doi: 10.1021/jm00017a022. J Med Chem. 1995. PMID: 7650691

5

Structure-based design of new constrained cyclic agonists of the cholecystokinin CCK-B receptor.

Blommaert AG, Dhôtel H, Ducos B, Durieux C, Goudreau N, Bado A, Garbay C, Roques BP. Blommaert AG, et al. J Med Chem. 1997 Feb 28;40(5):647-58. doi: 10.1021/jm9603072. J Med Chem. 1997. PMID: 9057851

6

SR146131: a new potent, orally active, and selective nonpeptide cholecystokinin subtype 1 receptor agonist. I. In vitro studies.

Bignon E, Bachy A, Boigegrain R, Brodin R, Cottineau M, Gully D, Herbert JM, Keane P, Labie C, Molimard JC, Olliero D, Oury-Donat F, Petereau C, Prabonnaud V, Rockstroh MP, Schaeffer P, Servant O, Thurneyssen O, Soubrié P, Pascal M, Maffrand JP, Le Fur G. Bignon E, et al. J Pharmacol Exp Ther. 1999 May;289(2):742-51. J Pharmacol Exp Ther. 1999. PMID: 10215648

7

Protein kinase C-mediated inhibition of transmembrane signalling through CCK(A) and CCK(B) receptors.

Smeets RL, Fouraux MA, van Emst-de Vries SE, De Pont JJ, Willems PH. Smeets RL, et al. Br J Pharmacol. 1998 Mar;123(6):1189-97. doi: 10.1038/sj.bjp.0701713. Br J Pharmacol. 1998. PMID: 9559904 Free PMC article.

8

1,4-Benzodiazepine peripheral cholecystokinin (CCK-A) receptor agonists.

Sherrill RG, Berman JM, Birkemo L, Croom DK, Dezube M, Ervin GN, Grizzle MK, James MK, Johnson MF, Queen KL, Rimele TJ, Vanmiddlesworth F, Sugg EE. Sherrill RG, et al. Bioorg Med Chem Lett. 2001 May 7;11(9):1145-8. doi: 10.1016/s0960-894x(01)00164-0. Bioorg Med Chem Lett. 2001. PMID: 11354363

9

3-[2-(N-phenylacetamide)]-1,5-benzodiazepines: orally active, binding selective CCK-A agonists.

Willson TM, Henke BR, Momtahen TM, Myers PL, Sugg EE, Unwalla RJ, Croom DK, Dougherty RW, Grizzle MK, Johnson MF, Queen KL, Rimele TJ, Yingling JD, James MK. Willson TM, et al. J Med Chem. 1996 Jul 19;39(15):3030-4. doi: 10.1021/jm960205b. J Med Chem. 1996. PMID: 8709137

10

Synthesis and biological properties of new constrained CCK-B antagonists: discrimination of two affinity states of the CCK-B receptor on transfected CHO cells.

Bellier B, McCort-Tranchepain I, Ducos B, Danascimento S, Meudal H, Noble F, Garbay C, Roques BP. Bellier B, et al. J Med Chem. 1997 Nov 21;40(24):3947-56. doi: 10.1021/jm970439a. J Med Chem. 1997. PMID: 9397175

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