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Items: 1 to 20 of 98

1.

Synthesis of novel benzothiazole amides: Evaluation of PPAR activity and anti-proliferative effects in paraganglioma, pancreatic and colorectal cancer cell lines.

Ammazzalorso A, De Lellis L, Florio R, Laghezza A, De Filippis B, Fantacuzzi M, Giampietro L, Maccallini C, Tortorella P, Veschi S, Loiodice F, Cama A, Amoroso R.

Bioorg Med Chem Lett. 2019 Aug 15;29(16):2302-2306. doi: 10.1016/j.bmcl.2019.06.020. Epub 2019 Jun 18.

PMID:
31272790
2.

Eco-friendly synthesis, in vitro anti-proliferative evaluation, and 3D-QSAR analysis of a novel series of monocationic 2-aryl/heteroaryl-substituted 6-(2-imidazolinyl)benzothiazole mesylates.

Racané L, Ptiček L, Sedić M, Grbčić P, Kraljević Pavelić S, Bertoša B, Sović I, Karminski-Zamola G.

Mol Divers. 2018 Aug;22(3):723-741. doi: 10.1007/s11030-018-9827-2. Epub 2018 Apr 17.

PMID:
29667008
3.

Benzothiazole-based N-(phenylsulfonyl)amides as a novel family of PPARα antagonists.

Ammazzalorso A, Giancristofaro A, D'Angelo A, Filippis BD, Fantacuzzi M, Giampietro L, Maccallini C, Amoroso R.

Bioorg Med Chem Lett. 2011 Aug 15;21(16):4869-72. doi: 10.1016/j.bmcl.2011.06.028.

PMID:
21742490
4.

Synthesis of 2-Substituted Benzothiazole Derivatives and Their In Vitro Anticancer Effects and Antioxidant Activities Against Pancreatic Cancer Cells.

Uremis N, Uremis MM, Tolun FI, Ceylan M, Doganer A, Kurt AH.

Anticancer Res. 2017 Nov;37(11):6381-6389.

PMID:
29061823
5.

Cytotoxic effect of a family of peroxisome proliferator-activated receptor antagonists in colorectal and pancreatic cancer cell lines.

Ammazzalorso A, De Lellis L, Florio R, Bruno I, De Filippis B, Fantacuzzi M, Giampietro L, Maccallini C, Perconti S, Verginelli F, Cama A, Amoroso R.

Chem Biol Drug Des. 2017 Nov;90(5):1029-1035. doi: 10.1111/cbdd.13026. Epub 2017 Jul 19.

PMID:
28544586
6.

Synthesis, structure-activity relationships and preliminary antitumor evaluation of benzothiazole-2-thiol derivatives as novel apoptosis inducers.

Wang Z, Shi XH, Wang J, Zhou T, Xu YZ, Huang TT, Li YF, Zhao YL, Yang L, Yang SY, Yu LT, Wei YQ.

Bioorg Med Chem Lett. 2011 Feb 15;21(4):1097-101. doi: 10.1016/j.bmcl.2010.12.124. Epub 2010 Dec 31.

PMID:
21262571
7.

Synthesis and Investigation of the Role of Benzopyran Dihydropyrimidinone Hybrids in Cell Proliferation, Migration and Tumor Growth.

Dash AK, Nayak D, Hussain N, Mintoo MJ, Bano S, Katoch A, Mondhe DM, Goswami A, Mukherjee D.

Anticancer Agents Med Chem. 2019;19(2):276-288. doi: 10.2174/1871520618666180903101422.

PMID:
30179143
8.

SKLB316, a novel small-molecule inhibitor of cell-cycle progression, induces G2/M phase arrest and apoptosis in vitro and inhibits tumor growth in vivo.

Xia Y, Lei Q, Zhu Y, Ye T, Wang N, Li G, Shi X, Liu Y, Shao B, Yin T, Zhao L, Wu W, Song X, Xiong Y, Wei Y, Yu L.

Cancer Lett. 2014 Dec 28;355(2):297-309. doi: 10.1016/j.canlet.2014.09.042. Epub 2014 Oct 7.

PMID:
25301449
9.

Novel pyrazolo[3,4-d]pyrimidines as potential cytotoxic agents: Design, synthesis, molecular docking and CDK2 inhibition.

Maher M, Kassab AE, Zaher AF, Mahmoud Z.

Anticancer Agents Med Chem. 2019 Apr 17. doi: 10.2174/1871520619666190417153350. [Epub ahead of print]

PMID:
31038080
10.

Effects of PPARα inhibition in head and neck paraganglioma cells.

Florio R, De Lellis L, di Giacomo V, Di Marcantonio MC, Cristiano L, Basile M, Verginelli F, Verzilli D, Ammazzalorso A, Prasad SC, Cataldi A, Sanna M, Cimini A, Mariani-Costantini R, Mincione G, Cama A.

PLoS One. 2017 Jun 8;12(6):e0178995. doi: 10.1371/journal.pone.0178995. eCollection 2017.

11.

Synthesis of Novel Benzothiazole-Piperazine Derivatives and Their Biological Evaluation as Acetylcholinesterase Inhibitors and Cytotoxic Agents.

Gurdal EE, Turgutalp B, Gulcan HO, Ercetin T, Sahin MF, Durmaz I, Atalay RC, Nguyen QD, Sippl W, Yarim M.

Anticancer Agents Med Chem. 2017;17(13):1837-1845. doi: 10.2174/1871520617666170412153604.

PMID:
28403780
12.

Design and synthesis of new potent anticancer benzothiazole amides and ureas featuring pyridylamide moiety and possessing dual B-Raf(V600E) and C-Raf kinase inhibitory activities.

El-Damasy AK, Lee JH, Seo SH, Cho NC, Pae AN, Keum G.

Eur J Med Chem. 2016 Jun 10;115:201-16. doi: 10.1016/j.ejmech.2016.02.039. Epub 2016 Feb 18.

PMID:
27017549
13.

[Design, synthesis and activities of novel benzothiazole derivatives containing arylpiperazine].

Liu WH, Chang JX, Liu Y, Luo JW, Zhang JW.

Yao Xue Xue Bao. 2013 Aug;48(8):1259-65. Chinese.

PMID:
24187833
14.

Melicope ptelefolia leaf extracts exhibit antioxidant activity and exert anti-proliferative effect with apoptosis induction on four different cancer cell lines.

Kabir MF, Mohd Ali J, Abolmaesoomi M, Hashim OH.

BMC Complement Altern Med. 2017 May 5;17(1):252. doi: 10.1186/s12906-017-1761-9.

15.

Synthesis and antitumor activity evaluation of new 2-(4-aminophenyl)benzothiazole derivatives bearing different heterocyclic rings.

Yurttaş L, Tay F, Demirayak Ş.

J Enzyme Inhib Med Chem. 2015 Jun;30(3):458-65. doi: 10.3109/14756366.2014.945168. Epub 2014 Sep 8.

PMID:
25198890
16.

New Ferrocene Compounds as Selective Cyclooxygenase (COX-2) Inhibitors: Design, Synthesis, Cytotoxicity and Enzyme-inhibitory Activity.

Farzaneh S, Zeinalzadeh E, Daraei B, Shahhosseini S, Zarghi A.

Anticancer Agents Med Chem. 2018;18(2):295-301. doi: 10.2174/1871520617666171003145533.

PMID:
28971779
17.

Synthesis and Evaluation of Antioxidant and Cytotoxicity of the N-Mannich Base of Berberine Bearing Benzothiazole Moieties.

Mistry BM, Shin HS, Keum YS, Pandurangan M, Kim DH, Moon SH, Kadam AA, Shinde SK, Patel RV.

Anticancer Agents Med Chem. 2017;17(12):1652-1660. doi: 10.2174/1871520617666170710180549.

PMID:
28699489
18.
19.

Synthesis of new diarylamides with pyrimidinyl pyridine scaffold and evaluation of their anti-proliferative effect on cancer cell lines.

Abdelazem AZ, Al-Sanea MM, Park HM, Lee SH.

Bioorg Med Chem Lett. 2016 Feb 15;26(4):1301-4. doi: 10.1016/j.bmcl.2016.01.014. Epub 2016 Jan 7.

PMID:
26786696
20.

Synthesis and Structural Elucidation of Novel Benzothiazole Derivatives as Anti-tubercular Agents: In-silico Screening for Possible Target Identification.

Venugopala KN, Chandrashekharappa S, Pillay M, Bhandary S, Kandeel M, Mahomoodally FM, Morsy MA, Chopra D, Aldhubiab BE, Attimarad M, Alwassil OI, Harsha S, Mlisana K, Odhav B.

Med Chem. 2019;15(3):311-326. doi: 10.2174/1573406414666180703121815.

PMID:
29968540

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