Similar articles for PMID: 30846405

Year	Number of Results
2007	1
2008	3
2009	8
2010	7
2011	10
2012	7
2013	14
2014	16
2015	21
2016	14
2017	13
2018	23
2019	33
2020	35
2021	18
2022	10
2023	11
2024	1

1

Discovery of novel selective Janus kinase 2 (JAK2) inhibitors bearing a 1H-pyrazolo[3,4-d]pyrimidin-4-amino scaffold.

Yin Y, Chen CJ, Yu RN, Shu L, Zhang TT, Zhang DY. Yin Y, et al. Bioorg Med Chem. 2019 Apr 15;27(8):1562-1576. doi: 10.1016/j.bmc.2019.02.054. Epub 2019 Feb 28. Bioorg Med Chem. 2019. PMID: 30846405

2

Structure-based design and synthesis of 1H-pyrazolo[3,4-d]pyrimidin-4-amino derivatives as Janus kinase 3 inhibitors.

Yin Y, Chen CJ, Yu RN, Wang ZJ, Zhang TT, Zhang DY. Yin Y, et al. Bioorg Med Chem. 2018 Sep 15;26(17):4774-4786. doi: 10.1016/j.bmc.2018.04.005. Epub 2018 Apr 4. Bioorg Med Chem. 2018. PMID: 30139575

3

Design, synthesis and preliminary biological evaluation of 4-aminopyrazole derivatives as novel and potent JAKs inhibitors.

Liang X, Huang Y, Zang J, Gao Q, Wang B, Xu W, Zhang Y. Liang X, et al. Bioorg Med Chem. 2016 Jun 15;24(12):2660-72. doi: 10.1016/j.bmc.2016.04.030. Epub 2016 Apr 20. Bioorg Med Chem. 2016. PMID: 27137359

4

Identification of 4-(2-furanyl)pyrimidin-2-amines as Janus kinase 2 inhibitors.

Wang Y, Huang W, Xin M, Chen P, Gui L, Zhao X, Tang F, Wang J, Liu F. Wang Y, et al. Bioorg Med Chem. 2017 Jan 1;25(1):75-83. doi: 10.1016/j.bmc.2016.10.011. Epub 2016 Oct 11. Bioorg Med Chem. 2017. PMID: 27771180

5

2-Aminopyrazolo[1,5-a]pyrimidines as potent and selective inhibitors of JAK2.

Ledeboer MW, Pierce AC, Duffy JP, Gao H, Messersmith D, Salituro FG, Nanthakumar S, Come J, Zuccola HJ, Swenson L, Shlyakter D, Mahajan S, Hoock T, Fan B, Tsai WJ, Kolaczkowski E, Carrier S, Hogan JK, Zessis R, Pazhanisamy S, Bennani YL. Ledeboer MW, et al. Bioorg Med Chem Lett. 2009 Dec 1;19(23):6529-33. doi: 10.1016/j.bmcl.2009.10.053. Epub 2009 Oct 24. Bioorg Med Chem Lett. 2009. PMID: 19857967

6

Design, synthesis and anticancer evaluation of 1H-pyrazolo[3,4-d]pyrimidine derivatives as potent EGFR^WT and EGFR^T790M inhibitors and apoptosis inducers.

Gaber AA, Bayoumi AH, El-Morsy AM, Sherbiny FF, Mehany ABM, Eissa IH. Gaber AA, et al. Bioorg Chem. 2018 Oct;80:375-395. doi: 10.1016/j.bioorg.2018.06.017. Epub 2018 Jun 12. Bioorg Chem. 2018. PMID: 29986185

7

Discovery of 4-amino-1H-pyrazolo[3,4-d]pyrimidin derivatives as novel discoidin domain receptor 1 (DDR1) inhibitors.

Dong R, Zhou X, Wang M, Li W, Zhang JY, Zheng X, Tang KX, Sun LP. Dong R, et al. Bioorg Med Chem. 2021 Jan 1;29:115876. doi: 10.1016/j.bmc.2020.115876. Epub 2020 Nov 17. Bioorg Med Chem. 2021. PMID: 33246255

8

Structure-based design and synthesis of pyrimidine-4,6-diamine derivatives as Janus kinase 3 inhibitors.

Yu RN, Chen CJ, Shu L, Yin Y, Wang ZJ, Zhang TT, Zhang DY. Yu RN, et al. Bioorg Med Chem. 2019 Apr 15;27(8):1646-1657. doi: 10.1016/j.bmc.2019.03.009. Epub 2019 Mar 5. Bioorg Med Chem. 2019. PMID: 30853331

9

The discovery of 2,5-isomers of triazole-pyrrolopyrimidine as selective Janus kinase 2 (JAK2) inhibitors versus JAK1 and JAK3.

Lee SM, Yoon KB, Lee HJ, Kim J, Chung YK, Cho WJ, Mukai C, Choi S, Kang KW, Han SY, Ko H, Kim YC. Lee SM, et al. Bioorg Med Chem. 2016 Nov 1;24(21):5036-5046. doi: 10.1016/j.bmc.2016.08.008. Epub 2016 Aug 6. Bioorg Med Chem. 2016. PMID: 27555284

10

Synthesis, anticancer evaluation, and molecular docking studies of some novel 4,6-disubstituted pyrazolo[3,4-d]pyrimidines as cyclin-dependent kinase 2 (CDK2) inhibitors.

Cherukupalli S, Chandrasekaran B, Kryštof V, Aleti RR, Sayyad N, Merugu SR, Kushwaha ND, Karpoormath R. Cherukupalli S, et al. Bioorg Chem. 2018 Sep;79:46-59. doi: 10.1016/j.bioorg.2018.02.030. Epub 2018 Mar 17. Bioorg Chem. 2018. PMID: 29753773

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