Similar articles for PMID: 30743173

Year	Number of Results
1940	1
1941	1
1943	1
2000	2
2005	1
2006	3
2007	2
2008	7
2009	4
2010	8
2011	5
2012	21
2013	17
2014	19
2015	13
2016	14
2017	14
2018	18
2019	35
2020	51
2021	36
2022	20
2023	15
2024	0

1

Toward a treatment of diabesity: Rational design, synthesis and biological evaluation of benzene-sulfonamide derivatives as a new class of PTP-1B inhibitors.

Ghareb N, El-Sayed NM, Abdelhameed R, Yamada K, Elgawish MS. Ghareb N, et al. Bioorg Chem. 2019 May;86:322-338. doi: 10.1016/j.bioorg.2019.01.052. Epub 2019 Jan 31. Bioorg Chem. 2019. PMID: 30743173

2

Discovery of potent, selective and orally bioavailable triaryl-sulfonamide based PTP1B inhibitors.

Patel D, Jain M, Shah SR, Bahekar R, Jadav P, Joharapurkar A, Dhanesha N, Shaikh M, Sairam KV, Kapadnis P. Patel D, et al. Bioorg Med Chem Lett. 2012 Jan 15;22(2):1111-7. doi: 10.1016/j.bmcl.2011.11.122. Epub 2011 Dec 6. Bioorg Med Chem Lett. 2012. PMID: 22189136

3

Design, synthesis and biological evaluation of some tetrazole acetamide derivatives as novel non-carboxylic PTP1B inhibitors.

Maheshwari N, Karthikeyan C, Bhadada SV, Verma AK, Sahi C, Moorthy NSHN, Trivedi P. Maheshwari N, et al. Bioorg Chem. 2019 Nov;92:103221. doi: 10.1016/j.bioorg.2019.103221. Epub 2019 Aug 30. Bioorg Chem. 2019. PMID: 31499261

4

A Library of Thiazolidin-4-one Derivatives as Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitors: An Attempt To Discover Novel Antidiabetic Agents.

Patel AD, Pasha TY, Lunagariya P, Shah U, Bhambharoliya T, Tripathi RKP. Patel AD, et al. ChemMedChem. 2020 Jul 3;15(13):1229-1242. doi: 10.1002/cmdc.202000055. Epub 2020 Jun 3. ChemMedChem. 2020. PMID: 32390300

5

Synthesis, biological evaluation and in silico studies of 5-(3-methoxybenzylidene)thiazolidine-2,4-dione analogues as PTP1B inhibitors.

Mahapatra MK, Kumar R, Kumar M. Mahapatra MK, et al. Bioorg Chem. 2017 Apr;71:1-9. doi: 10.1016/j.bioorg.2017.01.007. Epub 2017 Jan 17. Bioorg Chem. 2017. PMID: 28126289

6

Design, synthesis, kinetic, molecular dynamics, and hypoglycemic effect characterization of new and potential selective benzimidazole derivatives as Protein Tyrosine Phosphatase 1B inhibitors.

Campos-Almazán MI, Flores-Ramos M, Hernández-Campos A, Castillo R, Sierra-Campos E, Torgeson K, Peti W, Valdez-Solana M, Oria-Hernández J, Méndez ST, Castillo-Villanueva A, Jiménez-de Jesús H, Avitia-Domínguez C, Téllez-Valencia A. Campos-Almazán MI, et al. Bioorg Med Chem. 2021 Oct 15;48:116418. doi: 10.1016/j.bmc.2021.116418. Epub 2021 Sep 17. Bioorg Med Chem. 2021. PMID: 34563877

7

[Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].

Du X, Zhang SE, Liu JZ, Nie FL, Ye F, Tian JY, Xiao ZY. Du X, et al. Yao Xue Xue Bao. 2012 Mar;47(3):367-73. Yao Xue Xue Bao. 2012. PMID: 22645761 Chinese.

8

Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties.

Jiang B, Luo J, Guo S, Wang L. Jiang B, et al. Bioorg Chem. 2021 Mar;108:104648. doi: 10.1016/j.bioorg.2021.104648. Epub 2021 Jan 12. Bioorg Chem. 2021. PMID: 33493928

9

Discovery of novel high potent and cellular active ADC type PTP1B inhibitors with selectivity over TC-PTP via modification interacting with C site.

Du Y, Zhang Y, Ling H, Li Q, Shen J. Du Y, et al. Eur J Med Chem. 2018 Jan 20;144:692-700. doi: 10.1016/j.ejmech.2017.12.064. Epub 2017 Dec 20. Eur J Med Chem. 2018. PMID: 29289892

10

Molecular Docking, In-Silico ADMET Study and Development of 1,6- Dihydropyrimidine Derivative as Protein Tyrosine Phosphatase Inhibitor: An Approach to Design and Develop Antidiabetic Agents.

Patel AD, Barot R, Parmar I, Panchal I, Shah U, Patel M, Mishtry B. Patel AD, et al. Curr Comput Aided Drug Des. 2018;14(4):349-362. doi: 10.2174/1573409914666180426125721. Curr Comput Aided Drug Des. 2018. PMID: 29701158

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