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Items: 1 to 20 of 96

1.

Synthesis of 5-enamine-4-thiazolidinone derivatives with trypanocidal and anticancer activity.

Holota S, Kryshchyshyn A, Derkach H, Trufin Y, Demchuk I, Gzella A, Grellier P, Lesyk R.

Bioorg Chem. 2019 May;86:126-136. doi: 10.1016/j.bioorg.2019.01.045. Epub 2019 Jan 22.

PMID:
30690336
2.

Isothiochromenothiazoles-A Class of Fused Thiazolidinone Derivatives with Established Anticancer Activity That Inhibits Growth of Trypanosoma brucei brucei.

Kryshchyshyn A, Kaminskyy D, Nektegayev I, Grellier P, Lesyk R.

Sci Pharm. 2018 Oct 19;86(4). pii: E47. doi: 10.3390/scipharm86040047.

3.

Synthesis of pyrazoline-thiazolidinone hybrids with trypanocidal activity.

Havrylyuk D, Zimenkovsky B, Karpenko O, Grellier P, Lesyk R.

Eur J Med Chem. 2014 Oct 6;85:245-54. doi: 10.1016/j.ejmech.2014.07.103. Epub 2014 Jul 30.

PMID:
25089808
4.

Synthesis and biological activity evaluation of 5-pyrazoline substituted 4-thiazolidinones.

Havrylyuk D, Zimenkovsky B, Vasylenko O, Day CW, Smee DF, Grellier P, Lesyk R.

Eur J Med Chem. 2013 Aug;66:228-37. doi: 10.1016/j.ejmech.2013.05.044. Epub 2013 Jun 6.

PMID:
23811085
5.

Trypanocidal and cysteine protease inhibitory activity of isopentyl caffeate is not linked in Trypanosoma brucei.

Steverding D, da Nóbrega FR, Rushworth SA, de Sousa DP.

Parasitol Res. 2016 Nov;115(11):4397-4403. Epub 2016 Aug 18.

PMID:
27535679
6.

Isothiocoumarin-3-carboxylic acid derivatives: synthesis, anticancer and antitrypanosomal activity evaluation.

Kaminskyy D, Kryshchyshyn A, Nektegayev I, Vasylenko O, Grellier P, Lesyk R.

Eur J Med Chem. 2014 Mar 21;75:57-66. doi: 10.1016/j.ejmech.2014.01.028. Epub 2014 Jan 25.

PMID:
24530491
7.

5-Ene-4-thiazolidinones induce apoptosis in mammalian leukemia cells.

Senkiv J, Finiuk N, Kaminskyy D, Havrylyuk D, Wojtyra M, Kril I, Gzella A, Stoika R, Lesyk R.

Eur J Med Chem. 2016 Jul 19;117:33-46. doi: 10.1016/j.ejmech.2016.03.089. Epub 2016 Apr 2.

PMID:
27089210
8.

In vitro trypanocidal activity of dibutyltin dichloride and its fatty acid derivatives.

Shuaibu MN, Kanbara H, Yanagi T, Ichinose A, Ameh DA, Bonire JJ, Nok AJ.

Parasitol Res. 2003 Sep;91(1):5-11. Epub 2003 Jul 8.

PMID:
12851812
9.

In vitro antitrypanosomal and antiplasmodial activities of crude extracts and essential oils of Ocimum gratissimum Linn from Benin and influence of vegetative stage.

Kpadonou Kpoviessi BG, Kpoviessi SD, Yayi Ladekan E, Gbaguidi F, Frédérich M, Moudachirou M, Quetin-Leclercq J, Accrombessi GC, Bero J.

J Ethnopharmacol. 2014 Sep 29;155(3):1417-23. doi: 10.1016/j.jep.2014.07.014. Epub 2014 Jul 21.

PMID:
25058875
10.

8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases.

Fersing C, Boudot C, Pedron J, Hutter S, Primas N, Castera-Ducros C, Bourgeade-Delmas S, Sournia-Saquet A, Moreau A, Cohen A, Stigliani JL, Pratviel G, Crozet MD, Wyllie S, Fairlamb A, Valentin A, Rathelot P, Azas N, Courtioux B, Verhaeghe P, Vanelle P.

Eur J Med Chem. 2018 Sep 5;157:115-126. doi: 10.1016/j.ejmech.2018.07.064. Epub 2018 Aug 1.

PMID:
30092366
11.

Synthesis of 2-(5-((5-(4-chlorophenyl)furan-2-yl)methylene)-4-oxo-2-thioxothiazolidin-3-yl)acetic acid derivatives and evaluation of their cytotoxicity and induction of apoptosis in human leukemia cells.

Chandrappa S, Kavitha CV, Shahabuddin MS, Vinaya K, Ananda Kumar CS, Ranganatha SR, Raghavan SC, Rangappa KS.

Bioorg Med Chem. 2009 Mar 15;17(6):2576-84. doi: 10.1016/j.bmc.2009.01.016. Epub 2009 Jan 15.

PMID:
19243955
12.

3-(Oxazolo[4,5-b]pyridin-2-yl)anilides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei, the causative agent for human African trypanosomiasis.

Ferrins L, Rahmani R, Sykes ML, Jones AJ, Avery VM, Teston E, Almohaywi B, Yin J, Smith J, Hyland C, White KL, Ryan E, Campbell M, Charman SA, Kaiser M, Baell JB.

Eur J Med Chem. 2013 Aug;66:450-65. doi: 10.1016/j.ejmech.2013.05.007. Epub 2013 May 16.

PMID:
23831695
13.

5-Ene-4-thiazolidinones - An efficient tool in medicinal chemistry.

Kaminskyy D, Kryshchyshyn A, Lesyk R.

Eur J Med Chem. 2017 Nov 10;140:542-594. doi: 10.1016/j.ejmech.2017.09.031. Epub 2017 Sep 20. Review.

PMID:
28987611
14.

Synthesis and anticancer activity evaluation of 4-thiazolidinones containing benzothiazole moiety.

Havrylyuk D, Mosula L, Zimenkovsky B, Vasylenko O, Gzella A, Lesyk R.

Eur J Med Chem. 2010 Nov;45(11):5012-21. doi: 10.1016/j.ejmech.2010.08.008. Epub 2010 Aug 12.

PMID:
20810193
15.

Brazilian Cerrado Qualea grandiflora Mart. Leaves Exhibit Antiplasmodial and Trypanocidal Activities In vitro.

Cordeiro TM, Borghetti F, Caldas Oliveira SC, Bastos IMD, de Santana JM, Grellier P, Charneau S.

Pharmacogn Mag. 2017 Oct-Dec;13(52):668-672. doi: 10.4103/pm.pm_100_17. Epub 2017 Nov 13.

16.

Synthesis and antitrypanosomal activity of new 6,6,7-trisubstituted thiopyrano[2,3-d][1,3]thiazoles.

Zelisko N, Atamanyuk D, Vasylenko O, Grellier P, Lesyk R.

Bioorg Med Chem Lett. 2012 Dec 1;22(23):7071-4. doi: 10.1016/j.bmcl.2012.09.091. Epub 2012 Oct 2.

PMID:
23084895
17.

Tyrosol and hydroxytyrosol derivatives as antitrypanosomal and antileishmanial agents.

Belmonte-Reche E, Martínez-García M, Peñalver P, Gómez-Pérez V, Lucas R, Gamarro F, Pérez-Victoria JM, Morales JC.

Eur J Med Chem. 2016 Aug 25;119:132-40. doi: 10.1016/j.ejmech.2016.04.047. Epub 2016 Apr 26.

PMID:
27155468
18.

1,2-substituted 4-(1H)-quinolones: synthesis, antimalarial and antitrypanosomal activities in vitro.

Wube A, Hüfner A, Seebacher W, Kaiser M, Brun R, Bauer R, Bucar F.

Molecules. 2014 Sep 10;19(9):14204-20. doi: 10.3390/molecules190914204.

19.

Synthesis and evaluation of novel hybrids β-carboline-4-thiazolidinones as potential antitumor and antiviral agents.

Barbosa VA, Baréa P, Mazia RS, Ueda-Nakamura T, Costa WFD, Foglio MA, Goes Ruiz ALT, Carvalho JE, Vendramini-Costa DB, Nakamura CV, Sarragiotto MH.

Eur J Med Chem. 2016 Nov 29;124:1093-1104. doi: 10.1016/j.ejmech.2016.10.018. Epub 2016 Oct 11.

PMID:
27792980
20.

Novel ruthenium(II) cyclopentadienyl thiosemicarbazone compounds with antiproliferative activity on pathogenic trypanosomatid parasites.

Fernández M, Arce ER, Sarniguet C, Morais TS, Tomaz AI, Azar CO, Figueroa R, Diego Maya J, Medeiros A, Comini M, Helena Garcia M, Otero L, Gambino D.

J Inorg Biochem. 2015 Dec;153:306-314. doi: 10.1016/j.jinorgbio.2015.06.018. Epub 2015 Jun 30.

PMID:
26275470

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