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Items: 1 to 20 of 85

1.

Design and synthesis of biphenyl and biphenyl ether inhibitors of sulfatases.

Reuillon T, Alhasan SF, Beale GS, Bertoli A, Brennan A, Cano C, Reeves HL, Newell DR, Golding BT, Miller DC, Griffin RJ.

Chem Sci. 2016 Apr 21;7(4):2821-2826. doi: 10.1039/c5sc03612g. Epub 2016 Jan 11.

3.

Steroidal and nonsteroidal sulfamates as potent inhibitors of steroid sulfatase.

Woo LW, Howarth NM, Purohit A, Hejaz HA, Reed MJ, Potter BV.

J Med Chem. 1998 Mar 26;41(7):1068-83.

PMID:
9544207
4.

Inhibition of placental estrone sulfatase activity and MCF-7 breast cancer cell proliferation by estrone-3-amino derivatives.

Selcer KW, Jagannathan S, Rhodes ME, Li PK.

J Steroid Biochem Mol Biol. 1996 Sep;59(1):83-91.

PMID:
9009241
5.
6.

Dual aromatase-sulfatase inhibitors based on the anastrozole template: synthesis, in vitro SAR, molecular modelling and in vivo activity.

Jackson T, Woo LW, Trusselle MN, Chander SK, Purohit A, Reed MJ, Potter BV.

Org Biomol Chem. 2007 Sep 21;5(18):2940-52. Epub 2007 Aug 7. Erratum in: Org Biomol Chem. 2007 Oct 21;5(20):3368. Corrected and republished in: Org Biomol Chem. 2007 Oct 21;5(20):2940-52.

PMID:
17728860
7.

Synthesis and sulfatase inhibitory activities of non-steroidal estrone sulfatase inhibitors.

Li PK, Milano S, Kluth L, Rhodes ME.

J Steroid Biochem Mol Biol. 1996 Sep;59(1):41-8.

PMID:
9009236
8.

Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates.

Okada M, Nakagawa T, Iwashita S, Takegawa S, Fujii T, Koizumi N.

J Steroid Biochem Mol Biol. 2003 Nov;87(2-3):141-8.

PMID:
14672734
9.

Aryl sulfamates are broad spectrum inactivators of sulfatases: effects on sulfatases from various sources.

Bojarová P, Williams SJ.

Bioorg Med Chem Lett. 2009 Jan 15;19(2):477-80. doi: 10.1016/j.bmcl.2008.11.059. Epub 2008 Nov 20.

PMID:
19058962
10.

Development of (p-O-sulfamoyl)-N-alkanoyl-phenylalkyl amines as non-steroidal estrone sulfatase inhibitors.

Kolli A, Chu GH, Rhodes ME, Inoue K, Selcer KW, Li PK.

J Steroid Biochem Mol Biol. 1999 Jan;68(1-2):31-40.

PMID:
10215035
12.
13.

Highly potent first examples of dual aromatase-steroid sulfatase inhibitors based on a biphenyl template.

Woo LW, Jackson T, Putey A, Cozier G, Leonard P, Acharya KR, Chander SK, Purohit A, Reed MJ, Potter BV.

J Med Chem. 2010 Mar 11;53(5):2155-70. doi: 10.1021/jm901705h.

PMID:
20148564
14.

Stimulation of aryl sulfatase in rat peritoneal macrophages exposed to bone in vitro.

Gies JP, Dorey CK.

Calcif Tissue Int. 1981;33(2):181-4.

PMID:
6783275
15.

Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES).

Ahmed S, James K, Owen CP, Patel CK.

Bioorg Med Chem Lett. 2002 May 20;12(10):1343-6.

PMID:
11992773
16.

Synthesis and Biological Evaluation of Fluorinated 3-Phenylcoumarin-7-O-Sulfamate Derivatives as Steroid Sulfatase Inhibitors.

Demkowicz S, Daśko M, Kozak W, Krawczyk K, Witt D, Masłyk M, Kubiński K, Rachon J.

Chem Biol Drug Des. 2016 Feb;87(2):233-8. doi: 10.1111/cbdd.12652. Epub 2015 Sep 14.

PMID:
26280898
19.

Synthesis of aromatase inhibitors and dual aromatase steroid sulfatase inhibitors by linking an arylsulfamate motif to 4-(4H-1,2,4-triazol-4-ylamino)benzonitrile: SAR, crystal structures, in vitro and in vivo activities.

Bubert C, Woo LW, Sutcliffe OB, Mahon MF, Chander SK, Purohit A, Reed MJ, Potter BV.

ChemMedChem. 2008 Nov;3(11):1708-30. doi: 10.1002/cmdc.200800164.

PMID:
18816537
20.

Nonsteroidal compounds designed to mimic potent steroid sulfatase inhibitors.

Ciobanu LC, Luu-The V, Poirier D.

J Steroid Biochem Mol Biol. 2002 Mar;80(3):339-53.

PMID:
11948019

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