Similar articles for PMID: 25596758

Year	Number of Results
1955	3
1956	2
1960	2
1961	3
1962	1
1968	2
1971	7
1974	1
1980	1
1988	1
1993	1
1994	1
1998	1
1999	1
2000	1
2003	3
2005	6
2006	5
2007	8
2008	9
2009	4
2010	10
2011	12
2012	19
2013	16
2014	28
2015	21
2016	29
2017	16
2018	20
2019	16
2020	13
2021	9
2022	7
2023	3
2024	0

1

Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors.

Consalvi S, Alfonso S, Di Capua A, Poce G, Pirolli A, Sabatino M, Ragno R, Anzini M, Sartini S, La Motta C, Di Cesare Mannelli L, Ghelardini C, Biava M. Consalvi S, et al. Bioorg Med Chem. 2015 Feb 15;23(4):810-20. doi: 10.1016/j.bmc.2014.12.041. Epub 2014 Dec 26. Bioorg Med Chem. 2015. PMID: 25596758

2

Cyclooxygenase-2 inhibitors. 1,5-diarylpyrrol-3-acetic esters with enhanced inhibitory activity toward cyclooxygenase-2 and improved cyclooxygenase-2/cyclooxygenase-1 selectivity.

Biava M, Porretta GC, Poce G, Supino S, Forli S, Rovini M, Cappelli A, Manetti F, Botta M, Sautebin L, Rossi A, Pergola C, Ghelardini C, Vivoli E, Makovec F, Anzellotti P, Patrignani P, Anzini M. Biava M, et al. J Med Chem. 2007 Nov 1;50(22):5403-11. doi: 10.1021/jm0707525. Epub 2007 Oct 4. J Med Chem. 2007. PMID: 17915854 Free article.

3

Synthesis, anti-inflammatory, analgesic, COX-1/2 inhibitory activities and molecular docking studies of substituted 2-mercapto-4(3H)-quinazolinones.

Abdel-Aziz AA, Abou-Zeid LA, ElTahir KEH, Ayyad RR, El-Sayed MA, El-Azab AS. Abdel-Aziz AA, et al. Eur J Med Chem. 2016 Oct 4;121:410-421. doi: 10.1016/j.ejmech.2016.05.066. Epub 2016 Jun 1. Eur J Med Chem. 2016. PMID: 27318118

4

Synthesis and biological evaluation of 3-[4-(amino/methylsulfonyl)phenyl]methylene-indolin-2-one derivatives as novel COX-1/2 and 5-LOX inhibitors.

Lai Y, Ma L, Huang W, Yu X, Zhang Y, Ji H, Tian J. Lai Y, et al. Bioorg Med Chem Lett. 2010 Dec 15;20(24):7349-53. doi: 10.1016/j.bmcl.2010.10.056. Epub 2010 Oct 20. Bioorg Med Chem Lett. 2010. PMID: 21055929

5

Synthesis, biological evaluation, and enzyme docking simulations of 1,5-diarylpyrrole-3-alkoxyethyl ethers as selective cyclooxygenase-2 inhibitors endowed with anti-inflammatory and antinociceptive activity.

Anzini M, Rovini M, Cappelli A, Vomero S, Manetti F, Botta M, Sautebin L, Rossi A, Pergola C, Ghelardini C, Norcini M, Giordani A, Makovec F, Anzellotti P, Patrignani P, Biava M. Anzini M, et al. J Med Chem. 2008 Aug 14;51(15):4476-81. doi: 10.1021/jm800084s. Epub 2008 Jul 4. J Med Chem. 2008. PMID: 18598017

6

Design, synthesis, and biological evaluation of linear 1-(4-, 3- or 2-methylsulfonylphenyl)-2-phenylacetylenes: a novel class of cyclooxygenase-2 inhibitors.

Chen QH, Rao PN, Knaus EE. Chen QH, et al. Bioorg Med Chem. 2005 Dec 1;13(23):6425-34. doi: 10.1016/j.bmc.2005.06.064. Epub 2005 Aug 15. Bioorg Med Chem. 2005. PMID: 16099663

7

Novel analgesic/anti-inflammatory agents: diarylpyrrole acetic esters endowed with nitric oxide releasing properties.

Biava M, Porretta GC, Poce G, Battilocchio C, Alfonso S, Rovini M, Valenti S, Giorgi G, Calderone V, Martelli A, Testai L, Sautebin L, Rossi A, Papa G, Ghelardini C, Di Cesare Mannelli L, Giordani A, Anzellotti P, Bruno A, Patrignani P, Anzini M. Biava M, et al. J Med Chem. 2011 Nov 24;54(22):7759-71. doi: 10.1021/jm200715n. Epub 2011 Oct 31. J Med Chem. 2011. PMID: 21992176

8

Novel 2-(4-methylsulfonylphenyl)pyrimidine derivatives as highly potent and specific COX-2 inhibitors.

Orjales A, Mosquera R, López B, Olivera R, Labeaga L, Núñez MT. Orjales A, et al. Bioorg Med Chem. 2008 Mar 1;16(5):2183-99. doi: 10.1016/j.bmc.2007.11.079. Epub 2007 Dec 5. Bioorg Med Chem. 2008. PMID: 18158247

9

Synthesis and biological evaluation of N-substituted-3,5-diphenyl-2-pyrazoline derivatives as cyclooxygenase (COX-2) inhibitors.

Fioravanti R, Bolasco A, Manna F, Rossi F, Orallo F, Ortuso F, Alcaro S, Cirilli R. Fioravanti R, et al. Eur J Med Chem. 2010 Dec;45(12):6135-8. doi: 10.1016/j.ejmech.2010.10.005. Epub 2010 Oct 25. Eur J Med Chem. 2010. PMID: 20974503

10

Design, synthesis, and biological evaluation of new 1,4-diarylazetidin-2-one derivatives (β-lactams) as selective cyclooxygenase-2 inhibitors.

Arefi H, Naderi N, Shemirani ABI, Kiani Falavarjani M, Azami Movahed M, Zarghi A. Arefi H, et al. Arch Pharm (Weinheim). 2020 Mar;353(3):e1900293. doi: 10.1002/ardp.201900293. Epub 2020 Jan 9. Arch Pharm (Weinheim). 2020. PMID: 31917485

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

247 results

Results by year