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Items: 1 to 20 of 81

1.

Design, synthesis, antiviral activity, and pre-formulation development of poly-L-arginine-fatty acyl derivatives of nucleoside reverse transcriptase inhibitors.

Pemmaraju BP, Malekar S, Agarwal HK, Tiwari RK, Oh D, Doncel GF, Worthen DR, Parang K.

Nucleosides Nucleotides Nucleic Acids. 2015;34(1):1-15. doi: 10.1080/15257770.2014.945649.

2.

Synthesis and anti-HIV activities of unsymmetrical long chain dicarboxylate esters of dinucleoside reverse transcriptase inhibitors.

Agarwal HK, Chhikara BS, Doncel GF, Parang K.

Bioorg Med Chem Lett. 2017 May 1;27(9):1934-1937. doi: 10.1016/j.bmcl.2017.03.031. Epub 2017 Mar 16.

3.

Synthesis and anti-HIV activities of symmetrical dicarboxylate esters of dinucleoside reverse transcriptase inhibitors.

Agarwal HK, Buckheit KW, Buckheit RW Jr, Parang K.

Bioorg Med Chem Lett. 2012 Sep 1;22(17):5451-4. doi: 10.1016/j.bmcl.2012.07.037. Epub 2012 Jul 17.

4.

Synthesis and anti-HIV activities of glutamate and peptide conjugates of nucleoside reverse transcriptase inhibitors.

Agarwal HK, Chhikara BS, Quiterio M, Doncel GF, Parang K.

J Med Chem. 2012 Mar 22;55(6):2672-87. doi: 10.1021/jm201551m. Epub 2012 Mar 6.

PMID:
22352809
5.

A comparison of the phenotypic susceptibility profiles of emtricitabine and lamivudine.

Borroto-Esoda K, Parkin N, Miller MD.

Antivir Chem Chemother. 2007;18(5):297-300.

PMID:
18046962
6.

Cytosine deoxyribonucleoside anti-HIV analogues: a small chemical substitution allows relevant activities.

Scaglione F, Berrino L.

Int J Antimicrob Agents. 2012 Jun;39(6):458-63. doi: 10.1016/j.ijantimicag.2011.11.013. Epub 2012 Jan 23.

PMID:
22269860
7.

Deoxyribonucleoside 2'- or 3'-mixed disulfides: prodrugs to target ribonucleotide reductase and/or to inhibit HIV reverse transcription.

Roy B, Chambert S, Lepoivre M, Aubertin AM, Balzarini J, Décout JL.

J Med Chem. 2003 Jun 19;46(13):2565-8.

PMID:
12801219
8.

Partial selective inhibition of HIV-1 reverse transcriptase and human DNA polymerases γ and β by thiated 3'-fluorothymidine analogue 5'-triphosphates.

Wińska P, Miazga A, Poznański J, Kulikowski T.

Antiviral Res. 2010 Nov;88(2):176-81. doi: 10.1016/j.antiviral.2010.08.011. Epub 2010 Aug 23.

PMID:
20739003
9.

Molecular design, synthesis and biological evaluation of BP-O-DAPY and O-DAPY derivatives as non-nucleoside HIV-1 reverse transcriptase inhibitors.

Yang S, Pannecouque C, Daelemans D, Ma XD, Liu Y, Chen FE, De Clercq E.

Eur J Med Chem. 2013 Jul;65:134-43. doi: 10.1016/j.ejmech.2013.04.052. Epub 2013 May 3.

PMID:
23707918
10.
11.
12.

2'-Fluoro-4'-thio-2',3'-unsaturated nucleosides: anti-HIV activity, resistance profile, and molecular modeling studies.

Chong Y, Choo H, Schinazi RF, Chu CK.

Nucleosides Nucleotides Nucleic Acids. 2003 May-Aug;22(5-8):611-5.

PMID:
14565238
13.

Drug resistance and drug combination features of the human immunodeficiency virus inhibitor, BCH-10652 [(+/-)-2'-deoxy-3'-oxa-4'-thiocytidine, dOTC].

Taylor DL, Ahmed PS, Tyms AS, Wood LJ, Kelly LA, Chambers P, Clarke J, Bedard J, Bowlin TL, Rando RF.

Antivir Chem Chemother. 2000 Jul;11(4):291-301.

PMID:
10950391
14.

Synthesis and Biological Evaluation of 5'-O-Dicarboxylic Fatty Acyl Monoester Derivatives of Anti-HIV Nucleoside Reverse Transcriptase Inhibitors.

Pemmaraju B, Agarwal HK, Oh D, Buckheit KW, Buckheit RW Jr, Tiwari R, Parang K.

Tetrahedron Lett. 2014 Mar 19;55(12):1983-1986.

15.

D- and L-2',3'-didehydro-2',3'-dideoxy-3'-fluoro-carbocyclic nucleosides: synthesis, anti-HIV activity and mechanism of resistance.

Wang J, Jin Y, Rapp KL, Schinazi RF, Chu CK.

J Med Chem. 2007 Apr 19;50(8):1828-39. Epub 2007 Mar 21.

16.

Thiated analogues of 2',3'-dideoxy-3'-fluorothymidine and their phosphorylated and phosphonylated derivatives: synthesis, interaction with HIV reverse transcriptase, and in vitro anti-HIV activity.

Miazga A, Felczak K, Bretner M, Siwecka MA, Piasek A, Kulikowski T.

Nucleosides Nucleotides Nucleic Acids. 2003 May-Aug;22(5-8):973-5. No abstract available.

PMID:
14565324
17.

Thiated derivatives of 2',3'-dideoxy-3'-fluorothymidine: synthesis, in vitro anti-HIV-1 activity and interaction with recombinant drug resistant HIV-1 reverse transcriptase forms.

Miazga A, Hamy F, Louvel S, Klimkait T, Pietrusiewicz Z, Kurzyńska-Kokorniak A, Figlerowicz M, Wińska P, Kulikowski T.

Antiviral Res. 2011 Oct;92(1):57-63. doi: 10.1016/j.antiviral.2011.05.012. Epub 2011 Jun 6.

PMID:
21683097
18.

Synthesis and anti-HIV activity of [d4U]-[trovirdine analogue] and [d4T]-[trovirdine analogue] heterodimers as inhibitors of HIV-1 reverse transcriptase.

Gavriliu D, Fossey C, Ciurea A, Delbederi Z, Sugeac E, Ladurée D, Schmidt S, Laumond G, Aubertin AM.

Nucleosides Nucleotides Nucleic Acids. 2002;21(8-9):505-33.

PMID:
12484448
19.

Synthesis and biological evaluation of N4-(hetero)arylsulfonylquinoxalinones as HIV-1 reverse transcriptase inhibitors.

Xu B, Sun Y, Guo Y, Cao Y, Yu T.

Bioorg Med Chem. 2009 Apr 1;17(7):2767-74. doi: 10.1016/j.bmc.2009.02.039. Epub 2009 Feb 25.

PMID:
19269831
20.

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