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Items: 1 to 20 of 119

1.

No evidence for histamine H4 receptor in human monocytes.

Werner K, Neumann D, Buschauer A, Seifert R.

J Pharmacol Exp Ther. 2014 Dec;351(3):519-26. doi: 10.1124/jpet.114.218107. Epub 2014 Oct 1.

2.

Conformational Restriction and Enantioseparation Increase Potency and Selectivity of Cyanoguanidine-Type Histamine H4 Receptor Agonists.

Geyer R, Nordemann U, Strasser A, Wittmann HJ, Buschauer A.

J Med Chem. 2016 Apr 14;59(7):3452-70. doi: 10.1021/acs.jmedchem.6b00120. Epub 2016 Apr 5.

PMID:
27007611
3.

Histamine H4 receptor stimulation suppresses IL-12p70 production and mediates chemotaxis in human monocyte-derived dendritic cells.

Gutzmer R, Diestel C, Mommert S, Köther B, Stark H, Wittmann M, Werfel T.

J Immunol. 2005 May 1;174(9):5224-32.

4.

Synthesis and structure-activity relationships of cyanoguanidine-type and structurally related histamine H4 receptor agonists.

Igel P, Geyer R, Strasser A, Dove S, Seifert R, Buschauer A.

J Med Chem. 2009 Oct 22;52(20):6297-313. doi: 10.1021/jm900526h.

PMID:
19791743
5.

Incomplete activation of human eosinophils via the histamine H4-receptor: evidence for ligand-specific receptor conformations.

Reher TM, Neumann D, Buschauer A, Seifert R.

Biochem Pharmacol. 2012 Jul 15;84(2):192-203. doi: 10.1016/j.bcp.2012.04.004. Epub 2012 Apr 11.

PMID:
22516788
6.

Role of H4 receptor in histamine-mediated responses in human melanoma.

Massari NA, Medina VA, Martinel Lamas DJ, Cricco GP, Croci M, Sambuco L, Bergoc RM, Rivera ES.

Melanoma Res. 2011 Oct;21(5):395-404. doi: 10.1097/CMR.0b013e328347ee53.

PMID:
21691231
7.

Compared pharmacology of human histamine H3 and H4 receptors: structure-activity relationships of histamine derivatives.

Gbahou F, Vincent L, Humbert-Claude M, Tardivel-Lacombe J, Chabret C, Arrang JM.

Br J Pharmacol. 2006 Apr;147(7):744-54.

8.

Histamine H4 receptor agonists have more activities than H4 agonism in antigen-specific human T-cell responses.

Sugata Y, Okano M, Fujiwara T, Matsumoto R, Hattori H, Yamamoto M, Nishibori M, Nishizaki K.

Immunology. 2007 Jun;121(2):266-75. Epub 2007 Mar 7.

10.

Pleiotropic effect of histamine H4 receptor modulation in the central nervous system.

Galeotti N, Sanna MD, Ghelardini C.

Neuropharmacology. 2013 Aug;71:141-7. doi: 10.1016/j.neuropharm.2013.03.026. Epub 2013 Apr 11.

PMID:
23583928
11.

Synthesis and functional characterization of imbutamine analogs as histamine H3 and H4 receptor ligands.

Geyer R, Kaske M, Baumeister P, Buschauer A.

Arch Pharm (Weinheim). 2014 Feb;347(2):77-88. doi: 10.1002/ardp.201300316. Epub 2013 Nov 12.

PMID:
24493592
12.

Histamine downregulates monocyte CCL2 production through the histamine H4 receptor.

Dijkstra D, Leurs R, Chazot P, Shenton FC, Stark H, Werfel T, Gutzmer R.

J Allergy Clin Immunol. 2007 Aug;120(2):300-7. Epub 2007 May 15.

PMID:
17507084
13.

Profiling of histamine H4 receptor agonists in native human monocytes.

Gschwandtner M, Koether B, Werfel T, Stark H, Gutzmer R.

Br J Pharmacol. 2013 Sep;170(1):136-43. doi: 10.1111/bph.12237.

14.

Functional characterization of histamine H4 receptor on human mast cells.

Jemima EA, Prema A, Thangam EB.

Mol Immunol. 2014 Nov;62(1):19-28. doi: 10.1016/j.molimm.2014.05.007. Epub 2014 Jun 14.

PMID:
24934979
15.

Pharmacological characterization of the new histamine H4 receptor agonist VUF 8430.

Lim HD, Adami M, Guaita E, Werfel T, Smits RA, de Esch IJ, Bakker RA, Gutzmer R, Coruzzi G, Leurs R.

Br J Pharmacol. 2009 May;157(1):34-43. doi: 10.1111/j.1476-5381.2009.00200.x.

16.

Functional expression of H4 histamine receptor in human natural killer cells, monocytes, and dendritic cells.

Damaj BB, Becerra CB, Esber HJ, Wen Y, Maghazachi AA.

J Immunol. 2007 Dec 1;179(11):7907-15.

17.

Histamine induces proliferation in keratinocytes from patients with atopic dermatitis through the histamine 4 receptor.

Glatzer F, Gschwandtner M, Ehling S, Rossbach K, Janik K, Klos A, Bäumer W, Kietzmann M, Werfel T, Gutzmer R.

J Allergy Clin Immunol. 2013 Dec;132(6):1358-67. doi: 10.1016/j.jaci.2013.06.023. Epub 2013 Aug 9.

18.

Cellular analysis of the histamine H4 receptor in human myeloid cells.

Capelo R, Lehmann C, Ahmad K, Snodgrass R, Diehl O, Ringleb J, Flamand N, Weigert A, Stark H, Steinhilber D, Kahnt AS.

Biochem Pharmacol. 2016 Mar 1;103:74-84. doi: 10.1016/j.bcp.2016.01.007. Epub 2016 Jan 13.

PMID:
26774453
19.

2,4-Diaminopyrimidines as dual ligands at the histamine H1 and H4 receptor-H1/H4-receptor selectivity.

Hammer SG, Gobleder S, Naporra F, Wittmann HJ, Elz S, Heinrich MR, Strasser A.

Bioorg Med Chem Lett. 2016 Jan 15;26(2):292-300. doi: 10.1016/j.bmcl.2015.12.035. Epub 2015 Dec 11.

PMID:
26718844
20.

The H1 receptor agonist 2-(3-chlorophenyl)histamine activates Gi proteins in HL-60 cells through a mechanism that is independent of known histamine receptor subtypes.

Seifert R, Hagelüken A, Höer A, Höer D, Grünbaum L, Offermanns S, Schwaner I, Zingel V, Schunack W, Schultz G.

Mol Pharmacol. 1994 Apr;45(4):578-86.

PMID:
7514261

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