Similar articles for PMID: 24809953

Year	Number of Results
2003	1
2004	2
2005	5
2006	8
2007	6
2008	2
2009	3
2010	4
2011	9
2012	15
2013	14
2014	22
2015	30
2016	24
2017	19
2018	25
2019	23
2020	13
2021	18
2022	17
2023	2
2024	0

1

Novel N-linked aminopiperidine-based gyrase inhibitors with improved hERG and in vivo efficacy against Mycobacterium tuberculosis.

Hameed P S, Patil V, Solapure S, Sharma U, Madhavapeddi P, Raichurkar A, Chinnapattu M, Manjrekar P, Shanbhag G, Puttur J, Shinde V, Menasinakai S, Rudrapatana S, Achar V, Awasthy D, Nandishaiah R, Humnabadkar V, Ghosh A, Narayan C, Ramya VK, Kaur P, Sharma S, Werngren J, Hoffner S, Panduga V, Kumar CN, Reddy J, Kumar K N M, Ganguly S, Bharath S, Bheemarao U, Mukherjee K, Arora U, Gaonkar S, Coulson M, Waterson D, Sambandamurthy VK, de Sousa SM. Hameed P S, et al. J Med Chem. 2014 Jun 12;57(11):4889-905. doi: 10.1021/jm500432n. Epub 2014 May 23. J Med Chem. 2014. PMID: 24809953

2

Development of acridine derivatives as selective Mycobacterium tuberculosis DNA gyrase inhibitors.

Medapi B, Meda N, Kulkarni P, Yogeeswari P, Sriram D. Medapi B, et al. Bioorg Med Chem. 2016 Feb 15;24(4):877-85. doi: 10.1016/j.bmc.2016.01.011. Epub 2016 Jan 7. Bioorg Med Chem. 2016. PMID: 26787274

3

Novel N-linked aminopiperidine inhibitors of bacterial topoisomerase type II with reduced pK(a): antibacterial agents with an improved safety profile.

Reck F, Alm RA, Brassil P, Newman JV, Ciaccio P, McNulty J, Barthlow H, Goteti K, Breen J, Comita-Prevoir J, Cronin M, Ehmann DE, Geng B, Godfrey AA, Fisher SL. Reck F, et al. J Med Chem. 2012 Aug 9;55(15):6916-33. doi: 10.1021/jm300690s. Epub 2012 Jul 20. J Med Chem. 2012. PMID: 22779424

4

Replacement of cardiotoxic aminopiperidine linker with piperazine moiety reduces cardiotoxicity? Mycobacterium tuberculosis novel bacterial topoisomerase inhibitors.

Bobesh KA, Renuka J, Srilakshmi RR, Yellanki S, Kulkarni P, Yogeeswari P, Sriram D. Bobesh KA, et al. Bioorg Med Chem. 2016 Jan 1;24(1):42-52. doi: 10.1016/j.bmc.2015.11.039. Epub 2015 Nov 28. Bioorg Med Chem. 2016. PMID: 26678175

5

Thiazole-aminopiperidine hybrid analogues: design and synthesis of novel Mycobacterium tuberculosis GyrB inhibitors.

Jeankumar VU, Renuka J, Santosh P, Soni V, Sridevi JP, Suryadevara P, Yogeeswari P, Sriram D. Jeankumar VU, et al. Eur J Med Chem. 2013;70:143-53. doi: 10.1016/j.ejmech.2013.09.025. Epub 2013 Oct 3. Eur J Med Chem. 2013. PMID: 24148991

6

WQ-3810: A new fluoroquinolone with a high potential against fluoroquinolone-resistant Mycobacterium tuberculosis.

Ouchi Y, Mukai T, Koide K, Yamaguchi T, Park JH, Kim H, Yokoyama K, Tamaru A, Gordon SV, Nakajima C, Suzuki Y. Ouchi Y, et al. Tuberculosis (Edinb). 2020 Jan;120:101891. doi: 10.1016/j.tube.2019.101891. Epub 2019 Nov 18. Tuberculosis (Edinb). 2020. PMID: 31778929 Free article.

7

Extending the N-linked aminopiperidine class to the mycobacterial gyrase domain: pharmacophore mapping from known antibacterial leads.

Bobesh KA, Renuka J, Jeankumar VU, Shruti SK, Sridevi JP, Yogeeswari P, Sriram D. Bobesh KA, et al. Eur J Med Chem. 2014 Oct 6;85:593-604. doi: 10.1016/j.ejmech.2014.08.018. Epub 2014 Aug 7. Eur J Med Chem. 2014. PMID: 25127151

8

Development of novel N-linked aminopiperidine-based mycobacterial DNA gyrase B inhibitors: scaffold hopping from known antibacterial leads.

Jeankumar VU, Renuka J, Pulla VK, Soni V, Sridevi JP, Suryadevara P, Shravan M, Medishetti R, Kulkarni P, Yogeeswari P, Sriram D. Jeankumar VU, et al. Int J Antimicrob Agents. 2014 Mar;43(3):269-78. doi: 10.1016/j.ijantimicag.2013.12.006. Epub 2013 Dec 25. Int J Antimicrob Agents. 2014. PMID: 24434114

9

Design and synthesis of novel quinoline-aminopiperidine hybrid analogues as Mycobacterium tuberculosis DNA gyraseB inhibitors.

Medapi B, Renuka J, Saxena S, Sridevi JP, Medishetti R, Kulkarni P, Yogeeswari P, Sriram D. Medapi B, et al. Bioorg Med Chem. 2015 May 1;23(9):2062-78. doi: 10.1016/j.bmc.2015.03.004. Epub 2015 Mar 9. Bioorg Med Chem. 2015. PMID: 25801151

10

Design, synthesis, biological evaluation of substituted benzofurans as DNA gyraseB inhibitors of Mycobacterium tuberculosis.

Renuka J, Reddy KI, Srihari K, Jeankumar VU, Shravan M, Sridevi JP, Yogeeswari P, Babu KS, Sriram D. Renuka J, et al. Bioorg Med Chem. 2014 Sep 1;22(17):4924-34. doi: 10.1016/j.bmc.2014.06.041. Epub 2014 Jun 27. Bioorg Med Chem. 2014. PMID: 25129171

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

227 results

Results by year