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Items: 1 to 20 of 180

1.

Synthesis and evaluation of antimalarial properties of novel 4-aminoquinoline hybrid compounds.

Fisher GM, Tanpure RP, Douchez A, Andrews KT, Poulsen SA.

Chem Biol Drug Des. 2014 Oct;84(4):462-72. doi: 10.1111/cbdd.12335.

PMID:
24720445
2.

Antimalarial activity of compounds comprising a primary benzene sulfonamide fragment.

Andrews KT, Fisher GM, Sumanadasa SD, Skinner-Adams T, Moeker J, Lopez M, Poulsen SA.

Bioorg Med Chem Lett. 2013 Nov 15;23(22):6114-7. doi: 10.1016/j.bmcl.2013.09.015.

PMID:
24084158
3.

Synthesis, antimalarial activity and molecular docking of hybrid 4-aminoquinoline-1,3,5-triazine derivatives.

Bhat HR, Singh UP, Thakur A, Kumar Ghosh S, Gogoi K, Prakash A, Singh RK.

Exp Parasitol. 2015 Oct;157:59-67. doi: 10.1016/j.exppara.2015.06.016.

PMID:
26164360
4.

Antiplasmodial activity of new 4-aminoquinoline derivatives against chloroquine resistant strain.

Sinha M, Dola VR, Agarwal P, Srivastava K, Haq W, Puri SK, Katti SB.

Bioorg Med Chem. 2014 Jul 15;22(14):3573-86. doi: 10.1016/j.bmc.2014.05.024.

PMID:
24906512
5.

A medicinal chemistry perspective on 4-aminoquinoline antimalarial drugs.

O'Neill PM, Ward SA, Berry NG, Jeyadevan JP, Biagini GA, Asadollaly E, Park BK, Bray PG.

Curr Top Med Chem. 2006;6(5):479-507. Review.

PMID:
16719804
6.

Quinoline-pyrimidine hybrids: synthesis, antiplasmodial activity, SAR, and mode of action studies.

Singh K, Kaur H, Smith P, de Kock C, Chibale K, Balzarini J.

J Med Chem. 2014 Jan 23;57(2):435-48. doi: 10.1021/jm4014778.

PMID:
24354322
7.

Synthesis and bioevaluation of novel 4-aminoquinoline-tetrazole derivatives as potent antimalarial agents.

Pandey S, Agarwal P, Srivastava K, Rajakumar S, Puri SK, Verma P, Saxena JK, Sharma A, Lal J, Chauhan PM.

Eur J Med Chem. 2013 Aug;66:69-81. doi: 10.1016/j.ejmech.2013.05.023.

PMID:
23792317
8.

β-amino-alcohol tethered 4-aminoquinoline-isatin conjugates: synthesis and antimalarial evaluation.

Nisha, Gut J, Rosenthal PJ, Kumar V.

Eur J Med Chem. 2014 Sep 12;84:566-73. doi: 10.1016/j.ejmech.2014.07.064.

PMID:
25062007
9.

Novel hybrid molecules based on 15-membered azalide as potential antimalarial agents.

Starčević K, Pešić D, Toplak A, Landek G, Alihodžić S, Herreros E, Ferrer S, Spaventi R, Perić M.

Eur J Med Chem. 2012 Mar;49:365-78. doi: 10.1016/j.ejmech.2012.01.039.

PMID:
22321992
10.
11.
12.

Design and synthesis of new antimalarial agents from 4-aminoquinoline.

Solomon VR, Puri SK, Srivastava K, Katti SB.

Bioorg Med Chem. 2005 Mar 15;13(6):2157-65.

PMID:
15727868
13.

4-Aminoquinoline derivatives: Synthesis, in vitro and in vivo antiplasmodial activity against chloroquine-resistant parasites.

Singh S, Agarwal D, Sharma K, Sharma M, Nielsen MA, Alifrangis M, Singh AK, Gupta RD, Awasthi SK.

Eur J Med Chem. 2016 Oct 21;122:394-407. doi: 10.1016/j.ejmech.2016.06.033.

PMID:
27394399
14.

Synthesis and in vitro evaluation of new chloroquine-chalcone hybrids against chloroquine-resistant strain of Plasmodium falciparum.

Sashidhara KV, Avula SR, Palnati GR, Singh SV, Srivastava K, Puri SK, Saxena JK.

Bioorg Med Chem Lett. 2012 Sep 1;22(17):5455-9. doi: 10.1016/j.bmcl.2012.07.028.

PMID:
22850213
15.

Synthesis, Docking, In Vitro and In Vivo Antimalarial Activity of Hybrid 4-aminoquinoline-1,3,5-triazine Derivatives Against Wild and Mutant Malaria Parasites.

Bhat HR, Singh UP, Gahtori P, Ghosh SK, Gogoi K, Prakash A, Singh RK.

Chem Biol Drug Des. 2015 Sep;86(3):265-71. doi: 10.1111/cbdd.12490.

PMID:
25487527
16.

Novel conjugated quinoline-indoles compromise Plasmodium falciparum mitochondrial function and show promising antimalarial activity.

Teguh SC, Klonis N, Duffy S, Lucantoni L, Avery VM, Hutton CA, Baell JB, Tilley L.

J Med Chem. 2013 Aug 8;56(15):6200-15. doi: 10.1021/jm400656s.

PMID:
23837878
17.

Overcoming drug resistance to heme-targeted antimalarials by systematic side chain variation of 7-chloro-4-aminoquinolines.

Yearick K, Ekoue-Kovi K, Iwaniuk DP, Natarajan JK, Alumasa J, de Dios AC, Roepe PD, Wolf C.

J Med Chem. 2008 Apr 10;51(7):1995-8. doi: 10.1021/jm800106u.

18.

Synthesis of aminoquinoline-based aminoalcohols and oxazolidinones and their antiplasmodial activity.

Kobarfard F, Yardley V, Little S, Daryaee F, Chibale K.

Chem Biol Drug Des. 2012 Mar;79(3):326-31. doi: 10.1111/j.1747-0285.2011.01278.x.

PMID:
22129095
19.

Synthesis and antiplasmodial activity of new heteroaryl derivatives of 7-chloro-4-aminoquinoline.

Casagrande M, Barteselli A, Basilico N, Parapini S, Taramelli D, Sparatore A.

Bioorg Med Chem. 2012 Oct 1;20(19):5965-79. doi: 10.1016/j.bmc.2012.07.040.

PMID:
22917857
20.

Synthesis and evaluation of 7-substituted 4-aminoquinoline analogues for antimalarial activity.

Hwang JY, Kawasuji T, Lowes DJ, Clark JA, Connelly MC, Zhu F, Guiguemde WA, Sigal MS, Wilson EB, Derisi JL, Guy RK.

J Med Chem. 2011 Oct 27;54(20):7084-93. doi: 10.1021/jm200636z.

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