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Items: 1 to 20 of 143

1.

Synthesis and biological evaluation of 2-substituted-5-(4-nitrophenylsulfonamido)benzoxazoles as human GST P1-1 inhibitors, and description of the binding site features.

Ertan-Bolelli T, Musdal Y, Bolelli K, Yilmaz S, Aksoy Y, Yildiz I, Aki-Yalcin E, Yalcin I.

ChemMedChem. 2014 May;9(5):984-92. doi: 10.1002/cmdc.201400010. Epub 2014 Mar 26.

PMID:
24677708
2.

Identifying and characterizing binding sites on the irreversible inhibition of human glutathione S-transferase P1-1 by S-thiocarbamoylation.

Quesada-Soriano I, Primavera A, Casas-Solvas JM, Téllez-Sanz R, Barón C, Vargas-Berenguel A, Lo Bello M, García-Fuentes L.

Chembiochem. 2012 Jul 23;13(11):1594-604. doi: 10.1002/cbic.201200210. Epub 2012 Jun 27.

PMID:
22740430
3.

Sulphonamide-based bombesin prodrug analogues for glutathione transferase, useful in targeted cancer chemotherapy.

Axarli I, Labrou NE, Petrou C, Rassias N, Cordopatis P, Clonis YD.

Eur J Med Chem. 2009 May;44(5):2009-16. doi: 10.1016/j.ejmech.2008.10.009. Epub 2008 Oct 17.

PMID:
19019494
4.

FDA-approved drugs and other compounds tested as inhibitors of human glutathione transferase P1-1.

Musdal Y, Hegazy UM, Aksoy Y, Mannervik B.

Chem Biol Interact. 2013 Sep 5;205(1):53-62. doi: 10.1016/j.cbi.2013.06.003. Epub 2013 Jun 13.

PMID:
23769903
5.

Role of human glutathione S-transferases in the inactivation of reactive metabolites of clozapine.

Dragovic S, Boerma JS, van Bergen L, Vermeulen NP, Commandeur JN.

Chem Res Toxicol. 2010 Sep 20;23(9):1467-76. doi: 10.1021/tx100131f.

PMID:
20849150
6.

Inhibition of cellular enzymes by equine catechol estrogens in human breast cancer cells: specificity for glutathione S-transferase P1-1.

Yao J, Chang M, Li Y, Pisha E, Liu X, Yao D, Elguindi EC, Blond SY, Bolton JL.

Chem Res Toxicol. 2002 Jul;15(7):935-42.

PMID:
12119004
7.

Inhibition of human glutathione transferases by multidrug resistance chemomodulators in vitro.

Hayeshi R, Chinyanga F, Chengedza S, Mukanganyama S.

J Enzyme Inhib Med Chem. 2006 Oct;21(5):581-7.

PMID:
17194031
8.

Design and synthesis of 2-substituted-5-(4-trifluoromethylphenyl-sulphonamido)benzoxazole derivatives as human GST P1-1 inhibitors.

Ertan-Bolelli T, Bolelli K, Musdal Y, Yildiz I, Aki-Yalcin E, Mannervik B, Yalcin I.

Artif Cells Nanomed Biotechnol. 2017 May 14:1-8. doi: 10.1080/21691401.2017.1324464. [Epub ahead of print]

PMID:
28503938
9.

Potent isozyme-selective inhibition of human glutathione S-transferase A1-1 by a novel glutathione S-conjugate.

Cacciatore I, Caccuri AM, Cocco A, De Maria F, Di Stefano A, Luisi G, Pinnen F, Ricci G, Sozio P, Turella P.

Amino Acids. 2005 Nov;29(3):255-61. Epub 2005 Aug 8.

PMID:
16082503
10.

A novel method for screening the glutathione transferase inhibitors.

Wang Z, Jin L, Wegrzyn G, Wegrzyn A.

BMC Biochem. 2009 Mar 16;10:6. doi: 10.1186/1471-2091-10-6.

11.

Nitrobenzoxadiazole-based GSTP1-1 inhibitors containing the full peptidyl moiety of (pseudo)glutathione.

Luisi G, Mollica A, Carradori S, Lenoci A, De Luca A, Caccuri AM.

J Enzyme Inhib Med Chem. 2016 Dec;31(6):924-30. doi: 10.3109/14756366.2015.1070845. Epub 2015 Sep 2.

PMID:
26329912
12.

Assembly of ligands interaction models for glutathione-S-transferases from Plasmodium falciparum, human and mouse using enzyme kinetics and molecular docking.

Al-Qattan MN, Mordi MN, Mansor SM.

Comput Biol Chem. 2016 Oct;64:237-249. doi: 10.1016/j.compbiolchem.2016.07.007. Epub 2016 Jul 25.

PMID:
27475235
13.

Human theta class glutathione transferase: the crystal structure reveals a sulfate-binding pocket within a buried active site.

Rossjohn J, McKinstry WJ, Oakley AJ, Verger D, Flanagan J, Chelvanayagam G, Tan KL, Board PG, Parker MW.

Structure. 1998 Mar 15;6(3):309-22.

14.

Interactions of glutathione S-transferase-pi with ethacrynic acid and its glutathione conjugate.

Awasthi S, Srivastava SK, Ahmad F, Ahmad H, Ansari GA.

Biochim Biophys Acta. 1993 Jul 10;1164(2):173-8.

PMID:
8329448
15.

Peptidomimetic glutathione analogues as novel gammaGT stable GST inhibitors.

Burg D, Filippov DV, Hermanns R, van der Marel GA, van Boom JH, Mulder GJ.

Bioorg Med Chem. 2002 Jan;10(1):195-205.

PMID:
11738622
16.

Design and synthesis of 2-substituted benzoxazoles as novel PTP1B inhibitors.

Chandrasekharappa AP, Badiger SE, Dubey PK, Panigrahi SK, Manukonda SR.

Bioorg Med Chem Lett. 2013 May 1;23(9):2579-84. doi: 10.1016/j.bmcl.2013.02.109. Epub 2013 Mar 7.

PMID:
23528300
17.

Human cytosolic glutathione transferases: structure, function, and drug discovery.

Wu B, Dong D.

Trends Pharmacol Sci. 2012 Dec;33(12):656-68. doi: 10.1016/j.tips.2012.09.007. Epub 2012 Oct 31. Review.

PMID:
23121834
18.

A homology model for rat mu class glutathione S-transferase 4-4.

de Groot MJ, Vermeulen NP, Mullenders DL, Donné-Op den Kelder GM.

Chem Res Toxicol. 1996 Jan-Feb;9(1):28-40.

PMID:
8924604
19.

The inhibition of human glutathione S-transferases activity by plant polyphenolic compounds ellagic acid and curcumin.

Hayeshi R, Mutingwende I, Mavengere W, Masiyanise V, Mukanganyama S.

Food Chem Toxicol. 2007 Feb;45(2):286-95. Epub 2006 Aug 30.

PMID:
17046132
20.

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