Format
Sort by
Items per page

Send to

Choose Destination

Links from PubMed

Items: 1 to 20 of 95

1.

1-Phenyl-1H- and 2-phenyl-2H-1,2,3-triazol derivatives: design, synthesis and inhibitory effect on alpha-glycosidases.

Gonzaga D, Senger MR, da Silva Fde C, Ferreira VF, Silva FP Jr.

Eur J Med Chem. 2014 Mar 3;74:461-76. doi: 10.1016/j.ejmech.2013.12.039. Epub 2014 Jan 8.

PMID:
24487194
2.

Kinetics studies on the inhibition mechanism of pancreatic α-amylase by glycoconjugated 1H-1,2,3-triazoles: a new class of inhibitors with hypoglycemiant activity.

Senger MR, Gomes Lda C, Ferreira SB, Kaiser CR, Ferreira VF, Silva FP Jr.

Chembiochem. 2012 Jul 23;13(11):1584-93. doi: 10.1002/cbic.201200272. Epub 2012 Jun 29.

PMID:
22753086
3.

Synthesis, biological activity, and molecular modeling studies of 1H-1,2,3-triazole derivatives of carbohydrates as alpha-glucosidases inhibitors.

Ferreira SB, Sodero AC, Cardoso MF, Lima ES, Kaiser CR, Silva FP, Ferreira VF.

J Med Chem. 2010 Mar 25;53(6):2364-75. doi: 10.1021/jm901265h.

PMID:
20170190
4.

Synthesis of 1,2,3-triazole glycoconjugates as inhibitors of α-glucosidases.

da Rocha DR, Santos WC, Lima ES, Ferreira VF.

Carbohydr Res. 2012 Mar 1;350:14-9. doi: 10.1016/j.carres.2011.12.026. Epub 2012 Jan 3.

PMID:
22269981
5.

Application of click chemistry towards an efficient synthesis of 1,2,3-1H-triazolyl glycohybrids as enzyme inhibitors.

Anand N, Jaiswal N, Pandey SK, Srivastava AK, Tripathi RP.

Carbohydr Res. 2011 Jan 3;346(1):16-25. doi: 10.1016/j.carres.2010.10.017. Epub 2010 Oct 26.

PMID:
21129735
6.

Inhibition of α-glucosidase and α-amylase by diaryl derivatives of imidazole-thione and 1,2,4-triazole-thiol.

Balba M, El-Hady NA, Taha N, Rezki N, El Ashry el SH.

Eur J Med Chem. 2011 Jun;46(6):2596-601. doi: 10.1016/j.ejmech.2011.03.051. Epub 2011 Mar 31.

PMID:
21497424
7.

Anti-diabetic and anti-hypertensive potential of sprouted and solid-state bioprocessed soybean.

McCue P, Kwon YI, Shetty K.

Asia Pac J Clin Nutr. 2005;14(2):145-52.

8.

Synthesis, biological evaluation and molecular modeling studies of some novel thiazolidinediones with triazole ring.

Chinthala Y, Kumar Domatti A, Sarfaraz A, Singh SP, Kumar Arigari N, Gupta N, Satya SK, Kotesh Kumar J, Khan F, Tiwari AK, Paramjit G.

Eur J Med Chem. 2013;70:308-14. doi: 10.1016/j.ejmech.2013.10.005. Epub 2013 Oct 10.

PMID:
24177357
9.

Synthesis and glycosidase inhibitory activity of novel (2-phenyl-4H-benzopyrimedo[2,1-b]-thiazol-4-yliden)acetonitrile derivatives.

Patil VS, Nandre KP, Ghosh S, Rao VJ, Chopade BA, Bhosale SV, Bhosale SV.

Bioorg Med Chem Lett. 2012 Dec 1;22(23):7011-4. doi: 10.1016/j.bmcl.2012.10.025. Epub 2012 Oct 13.

PMID:
23102653
10.
11.

Homonojirimycin isomers and N-alkylated homonojirimycins: structural and conformational basis of inhibition of glycosidases.

Asano N, Nishida M, Kato A, Kizu H, Matsui K, Shimada Y, Itoh T, Baba M, Watson AA, Nash RJ, Lilley PM, Watkin DJ, Fleet GW.

J Med Chem. 1998 Jul 2;41(14):2565-71.

PMID:
9651160
12.

Synthesis of novel indenoquinoxaline derivatives as potent α-glucosidase inhibitors.

Khan MS, Munawar MA, Ashraf M, Alam U, Ata A, Asiri AM, Kousar S, Khan MA.

Bioorg Med Chem. 2014 Feb 1;22(3):1195-200. doi: 10.1016/j.bmc.2013.12.024. Epub 2013 Dec 21.

PMID:
24398385
13.

A novel competitive class of α-glucosidase inhibitors: (E)-1-phenyl-3-(4-styrylphenyl)urea derivatives.

Kim JY, Lee JW, Kim YS, Lee Y, Ryu YB, Kim S, Ryu HW, Curtis-Long MJ, Lee KW, Lee WS, Park KH.

Chembiochem. 2010 Oct 18;11(15):2125-31. doi: 10.1002/cbic.201000376.

PMID:
20827790
14.

Synthesis and evaluation of the alpha-glucosidase inhibitory activity of 3-[4-(phenylsulfonamido)benzoyl]-2H-1-benzopyran-2-one derivatives.

Wang S, Yan J, Wang X, Yang Z, Lin F, Zhang T.

Eur J Med Chem. 2010 Mar;45(3):1250-5. doi: 10.1016/j.ejmech.2009.12.031. Epub 2009 Dec 22.

PMID:
20045223
15.

Synthesis and biological evaluation of phenyl substituted 1H-1,2,4-triazoles as non-steroidal inhibitors of 17β-hydroxysteroid dehydrogenase type 2.

Al-Soud YA, Marchais-Oberwinkler S, Frotscher M, Hartmann RW.

Arch Pharm (Weinheim). 2012 Aug;345(8):610-21. doi: 10.1002/ardp.201200025. Epub 2012 Apr 25.

PMID:
22532378
16.

The synthesis and biological evaluation of 1-C-alkyl-L-arabinoiminofuranoses, a novel class of α-glucosidase inhibitors.

Natori Y, Imahori T, Murakami K, Yoshimura Y, Nakagawa S, Kato A, Adachi I, Takahata H.

Bioorg Med Chem Lett. 2011 Jan 15;21(2):738-41. doi: 10.1016/j.bmcl.2010.11.112. Epub 2010 Nov 30.

PMID:
21185187
17.

Inhibition of some hepatic glycosidases by the diseco nucleoside, 4-amino-3-(D-glucopentitol-1-yl)-5-mercapto-1,2,4-triazole and its 3-methyl analog.

Balbaa M, Mansour H, El-Sawy H, El-Ashry el-SH.

Nucleosides Nucleotides Nucleic Acids. 2002 Oct;21(10):695-708.

PMID:
12502284
19.

Discovery of novel inhibitors for human intestinal maltase: virtual screening in a WISDOM environment and in vitro evaluation.

Nguyen TT, Ryu HJ, Lee SH, Hwang S, Cha J, Breton V, Kim D.

Biotechnol Lett. 2011 Nov;33(11):2185-91. doi: 10.1007/s10529-011-0675-8. Epub 2011 Jul 7.

PMID:
21735260
20.

Synthesis and evaluation of 1,ω-bis(1,2,3,5-thiatriazol-5-yl)alkanes as in vitro and in vivo α-amylase and lipase inhibitors.

Hamzaoui S, Hamden K, Ben Salem A, Mourer M, Regnouf-De-Vains JB, Kossentini M.

Arch Pharm (Weinheim). 2013 Apr;346(4):321-9. doi: 10.1002/ardp.201200312. Epub 2013 Feb 28.

PMID:
23447412

Supplemental Content

Support Center