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Items: 1 to 20 of 99

1.

Identification of a selective inhibitor of murine intestinal alkaline phosphatase (ML260) by concurrent ultra-high throughput screening against human and mouse isozymes.

Ardecky RJ, Bobkova EV, Kiffer-Moreira T, Brown B, Ganji S, Zou J, Pass I, Narisawa S, Iano FG, Rosenstein C, Cheltsov A, Rascon J, Hedrick M, Gasior C, Forster A, Shi S, Dahl R, Vasile S, Su Y, Sergienko E, Chung TDY, Kaunitz J, Hoylaerts MF, Pinkerton AB, Millán JL.

Bioorg Med Chem Lett. 2014 Feb 1;24(3):1000-1004. doi: 10.1016/j.bmcl.2013.12.043. Epub 2013 Dec 19.

2.

A Selective Murine Intestinal Alkaline Phosphatase (muIAP) Inhibitor.

Ganji S, Zou J, Brown B, Bobkova EV, Ardecky R, Rosenstein C, Pass I, Dahl R, Vasile S, Sergienko E, Shi S, Stonich D, Cheltov A, Su Y, Mangravita-Novo A, Vicchiarelli M, McAnally D, Kim S, Nguyen H, Moreira TK, Smith LH, Zeng FY, Diwan J, Chung TDY, Pinkerton AB, Kaunitz J, Millán JL.

Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010-.
2011 Oct 31 [updated 2013 Mar 7].

3.

Modulators of intestinal alkaline phosphatase.

Bobkova EV, Kiffer-Moreira T, Sergienko EA.

Methods Mol Biol. 2013;1053:135-44. doi: 10.1007/978-1-62703-562-0_9.

PMID:
23860652
4.

Multisystemic functions of alkaline phosphatases.

Buchet R, Millán JL, Magne D.

Methods Mol Biol. 2013;1053:27-51. doi: 10.1007/978-1-62703-562-0_3. Review.

PMID:
23860646
5.

A novel phosphatase upregulated in Akp3 knockout mice.

Narisawa S, Hoylaerts MF, Doctor KS, Fukuda MN, Alpers DH, Millán JL.

Am J Physiol Gastrointest Liver Physiol. 2007 Nov;293(5):G1068-77. Epub 2007 Sep 27.

PMID:
17901166
6.

Synthesis, characterization and biological evaluation of novel chalcone sulfonamide hybrids as potent intestinal alkaline phosphatase inhibitors.

Ejaz SA, Saeed A, Siddique MN, Nisa ZU, Khan S, Lecka J, Sévigny J, Iqbal J.

Bioorg Chem. 2017 Feb;70:229-236. doi: 10.1016/j.bioorg.2017.01.003. Epub 2017 Jan 5.

PMID:
28110961
7.
8.

Diarylsulfonamides and their bioisosteres as dual inhibitors of alkaline phosphatase and carbonic anhydrase: Structure activity relationship and molecular modelling studies.

Al-Rashida M, Ejaz SA, Ali S, Shaukat A, Hamayoun M, Ahmed M, Iqbal J.

Bioorg Med Chem. 2015 May 15;23(10):2435-44. doi: 10.1016/j.bmc.2015.03.054. Epub 2015 Mar 27.

PMID:
25865133
9.

Facile dimethyl amino group triggered cyclic sulfonamides synthesis and evaluation as alkaline phosphatase inhibitors.

Bhatti HA, Khatoon M, Al-Rashida M, Bano H, Iqbal N, Zaib-Un-Nisa, Yousuf S, Khan KM, Hameed A, Iqbal J.

Bioorg Chem. 2017 Apr;71:10-18. doi: 10.1016/j.bioorg.2017.01.008. Epub 2017 Jan 18.

PMID:
28139246
10.

Structural evidence of functional divergence in human alkaline phosphatases.

Le Du MH, Millan JL.

J Biol Chem. 2002 Dec 20;277(51):49808-14. Epub 2002 Oct 7.

11.

Identification of novel chromone based sulfonamides as highly potent and selective inhibitors of alkaline phosphatases.

al-Rashida M, Raza R, Abbas G, Shah MS, Kostakis GE, Lecka J, Sévigny J, Muddassar M, Papatriantafyllopoulou C, Iqbal J.

Eur J Med Chem. 2013 Aug;66:438-49. doi: 10.1016/j.ejmech.2013.06.015. Epub 2013 Jun 19.

PMID:
23831808
12.

Isonicotinohydrazones as inhibitors of alkaline phosphatase and ecto-5'-nucleotidase.

Channar PA, Shah SJ, Hassan S, Nisa ZU, Lecka J, Sévigny J, Bajorath J, Saeed A, Iqbal J.

Chem Biol Drug Des. 2017 Mar;89(3):365-370. doi: 10.1111/cbdd.12861. Epub 2016 Oct 26.

PMID:
27589035
13.

Heterogeneity in alkaline phosphatase isozyme expression in human testicular germ cell tumours: An enzyme-/immunohistochemical and molecular analysis.

Roelofs H, Manes T, Janszen T, Millán JL, Oosterhuis JW, Looijenga LH.

J Pathol. 1999 Oct;189(2):236-44.

PMID:
10547581
15.

Identification of pulmonary surfactant that bears intestinal-type and tissue-nonspecific-type alkaline phosphatase in endotoxin-induced rat bronchoalveolar fluid.

Harada T, Koyama I, Shimoi A, Alpers DH, Komoda T.

Cell Tissue Res. 2002 Jan;307(1):69-77. Epub 2001 Oct 30.

PMID:
11810315
16.

Crystal structure of rat intestinal alkaline phosphatase--role of crown domain in mammalian alkaline phosphatases.

Ghosh K, Mazumder Tagore D, Anumula R, Lakshmaiah B, Kumar PP, Singaram S, Matan T, Kallipatti S, Selvam S, Krishnamurthy P, Ramarao M.

J Struct Biol. 2013 Nov;184(2):182-92. doi: 10.1016/j.jsb.2013.09.017. Epub 2013 Sep 27.

PMID:
24076154
17.

A method for direct assessment of tissue-nonspecific alkaline phosphatase (TNAP) inhibitors in blood samples.

Sergienko EA, Sun Q, Ma CT.

Methods Mol Biol. 2013;1053:103-13. doi: 10.1007/978-1-62703-562-0_6.

PMID:
23860649
18.

Synthesis, alkaline phosphatase inhibition studies and molecular docking of novel derivatives of 4-quinolones.

Miliutina M, Ejaz SA, Khan SU, Iaroshenko VO, Villinger A, Iqbal J, Langer P.

Eur J Med Chem. 2017 Jan 27;126:408-420. doi: 10.1016/j.ejmech.2016.11.036. Epub 2016 Nov 17.

PMID:
27907877
19.

Expression and regulation of alkaline phosphatases in human breast cancer MCF-7 cells.

Tsai LC, Hung MW, Chen YH, Su WC, Chang GG, Chang TC.

Eur J Biochem. 2000 Mar;267(5):1330-9.

20.

Design and synthesis of selective inhibitors of placental alkaline phosphatase.

Lanier M, Sergienko E, Simão AM, Su Y, Chung T, Millán JL, Cashman JR.

Bioorg Med Chem. 2010 Jan 15;18(2):573-9. doi: 10.1016/j.bmc.2009.12.012. Epub 2009 Dec 11.

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