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Items: 1 to 20 of 128

1.

Convergent diversity-oriented side-chain macrocyclization scan for unprotected polypeptides.

Zou Y, Spokoyny AM, Zhang C, Simon MD, Yu H, Lin YS, Pentelute BL.

Org Biomol Chem. 2014 Jan 28;12(4):566-73. doi: 10.1039/c3ob42168f.

2.

Synthesis of macrocyclic organo-peptide hybrids from ribosomal polypeptide precursors via CuAAC-/hydrazide-mediated cyclization.

Smith JM, Fasan R.

Methods Mol Biol. 2015;1248:23-38. doi: 10.1007/978-1-4939-2020-4_2. Review.

3.

Emerging strategies to access peptide macrocycles from genetically encoded polypeptides.

Smith JM, Frost JR, Fasan R.

J Org Chem. 2013 Apr 19;78(8):3525-31. doi: 10.1021/jo400119s. Epub 2013 Mar 29.

PMID:
23517465
5.

A diversity-oriented synthesis approach to macrocycles via oxidative ring expansion.

Kopp F, Stratton CF, Akella LB, Tan DS.

Nat Chem Biol. 2012 Mar 11;8(4):358-65. doi: 10.1038/nchembio.911.

6.

Macrocyclization of organo-peptide hybrids through a dual bio-orthogonal ligation: insights from structure-reactivity studies.

Frost JR, Vitali F, Jacob NT, Brown MD, Fasan R.

Chembiochem. 2013 Jan 2;14(1):147-60. doi: 10.1002/cbic.201200579. Epub 2012 Nov 30.

PMID:
23203912
7.

Bidirectional macrocyclization of peptides by double multicomponent reactions.

Ricardo MG, Morales FE, Garay H, Reyes O, Vasilev D, Wessjohann LA, Rivera DG.

Org Biomol Chem. 2015 Jan 14;13(2):438-46. doi: 10.1039/c4ob01915f.

PMID:
25371987
8.

Acetone-Linked Peptides: A Convergent Approach for Peptide Macrocyclization and Labeling.

Assem N, Ferreira DJ, Wolan DW, Dawson PE.

Angew Chem Int Ed Engl. 2015 Jul 20;54(30):8665-8. doi: 10.1002/anie.201502607. Epub 2015 Jun 11.

9.

Enzyme-catalyzed macrocyclization of long unprotected peptides.

Zhang C, Dai P, Spokoyny AM, Pentelute BL.

Org Lett. 2014 Jul 18;16(14):3652-5. doi: 10.1021/ol501609y. Epub 2014 Jul 8.

10.

The role of the amino acid-derived side chain in the preorganization of C₂-symmetric pseudopeptides: effect on S(N)2 macrocyclization reactions.

Martí-Centelles V, Burguete MI, Cativiela C, Luis SV.

J Org Chem. 2014 Jan 17;79(2):559-70. doi: 10.1021/jo4022309. Epub 2013 Dec 23.

PMID:
24328149
11.

A two-directional strategy for the diversity-oriented synthesis of macrocyclic scaffolds.

O'Connell KM, Beckmann HS, Laraia L, Horsley HT, Bender A, Venkitaraman AR, Spring DR.

Org Biomol Chem. 2012 Oct 7;10(37):7545-51. doi: 10.1039/c2ob26272j.

PMID:
22890306
12.

A diversity-oriented synthesis strategy enabling the combinatorial-type variation of macrocyclic peptidomimetic scaffolds.

Isidro-Llobet A, Hadje Georgiou K, Galloway WR, Giacomini E, Hansen MR, Méndez-Abt G, Tan YS, Carro L, Sore HF, Spring DR.

Org Biomol Chem. 2015 Apr 21;13(15):4570-80. doi: 10.1039/c5ob00371g.

13.

Synthesis of peptide macrocycles using unprotected amino aldehydes.

Rotstein BH, Rai V, Hili R, Yudin AK.

Nat Protoc. 2010 Nov;5(11):1813-22. doi: 10.1038/nprot.2010.127. Epub 2010 Oct 21.

PMID:
21030956
14.

A Thiol-Ene Coupling Approach to Native Peptide Stapling and Macrocyclization.

Wang Y, Chou DH.

Angew Chem Int Ed Engl. 2015 Sep 7;54(37):10931-4. doi: 10.1002/anie.201503975. Epub 2015 Jul 17.

PMID:
26189498
15.

Macrocyclic diketopiperazine receptors: effect of macrocyclization on the binding properties of two-armed receptors.

Bernard J, Wennemers H.

Org Lett. 2007 Oct 11;9(21):4283-6. Epub 2007 Sep 20.

PMID:
17880233
16.

Diversity-oriented synthesis of macrocyclic peptidomimetics.

Isidro-Llobet A, Murillo T, Bello P, Cilibrizzi A, Hodgkinson JT, Galloway WR, Bender A, Welch M, Spring DR.

Proc Natl Acad Sci U S A. 2011 Apr 26;108(17):6793-8. doi: 10.1073/pnas.1015267108. Epub 2011 Mar 7.

17.

Template-constrained macrocyclic peptides prepared from native, unprotected precursors.

Lawson KV, Rose TE, Harran PG.

Proc Natl Acad Sci U S A. 2013 Oct 1;110(40):E3753-60. doi: 10.1073/pnas.1311706110. Epub 2013 Sep 16.

18.

Direct comparison of linear and macrocyclic compound libraries as a source of protein ligands.

Gao Y, Kodadek T.

ACS Comb Sci. 2015 Mar 9;17(3):190-5. doi: 10.1021/co500161c. Epub 2015 Feb 14.

19.

Macrocyclization of Unprotected Peptide Isocyanates.

Vinogradov AA, Choo ZN, Totaro KA, Pentelute BL.

Org Lett. 2016 Mar 18;18(6):1226-9. doi: 10.1021/acs.orglett.5b03626. Epub 2016 Mar 7.

PMID:
26948900
20.

In vitro selection of multiple libraries created by genetic code reprogramming to discover macrocyclic peptides that antagonize VEGFR2 activity in living cells.

Kawakami T, Ishizawa T, Fujino T, Reid PC, Suga H, Murakami H.

ACS Chem Biol. 2013;8(6):1205-14. doi: 10.1021/cb300697h. Epub 2013 Apr 2.

PMID:
23517428

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