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Items: 1 to 20 of 93

1.

GABA(B)-agonistic activity of certain baclofen homologues.

Attia MI, Herdeis C, Bräuner-Osborne H.

Molecules. 2013 Aug 22;18(9):10266-84. doi: 10.3390/molecules180910266.

2.

GABA(B) receptors do not internalize after baclofen treatment, possibly due to a lack of β-arrestin association: study with a real-time visualizing assay.

Sudo Y, Hojo M, Ando Y, Takada M, Murata H, Kurata S, Nishida N, Uezono Y.

Synapse. 2012 Sep;66(9):759-69. doi: 10.1002/syn.21565. Epub 2012 May 17.

PMID:
22517292
3.

Cytoskeletal rearrangement and Src and PI-3K-dependent Akt activation control GABA(B)R-mediated chemotaxis.

Barati MT, Scherzer J, Wu R, Rane MJ, Klein JB.

Cell Signal. 2015 Jun;27(6):1178-1185. doi: 10.1016/j.cellsig.2015.02.022. Epub 2015 Feb 26.

4.

Isovaline does not activate GABA(B) receptor-coupled potassium currents in GABA(B) expressing AtT-20 cells and cultured rat hippocampal neurons.

Pitman KA, Borgland SL, MacLeod B, Puil E.

PLoS One. 2015 Feb 23;10(2):e0118497. doi: 10.1371/journal.pone.0118497. eCollection 2015.

5.

Baclofen administration alters fear extinction and GABAergic protein levels.

Heaney CF, Bolton MM, Murtishaw AS, Sabbagh JJ, Magcalas CM, Kinney JW.

Neurobiol Learn Mem. 2012 Oct;98(3):261-71. doi: 10.1016/j.nlm.2012.09.005. Epub 2012 Sep 23.

6.

Synthesis and pharmacological evaluation of gamma-aminobutyric acid analogues. New ligand for GABAB sites.

Berthelot P, Vaccher C, Musadad A, Flouquet N, Debaert M, Luyckx M.

J Med Chem. 1987 Apr;30(4):743-6.

PMID:
3031294
7.

General, kappa, delta and mu opioid receptor antagonists mediate feeding elicited by the GABA-B agonist baclofen in the ventral tegmental area and nucleus accumbens shell in rats: reciprocal and regional interactions.

Miner P, Shimonova L, Khaimov A, Borukhova Y, Ilyayeva E, Ranaldi R, Bodnar RJ.

Brain Res. 2012 Mar 14;1443:34-51. doi: 10.1016/j.brainres.2012.01.015. Epub 2012 Jan 17.

PMID:
22305145
8.

Effects of GABAB receptor agonists and antagonists on glycemia regulation in mice.

Bonaventura MM, Crivello M, Ferreira ML, Repetto M, Cymeryng C, Libertun C, Lux-Lantos VA.

Eur J Pharmacol. 2012 Feb 29;677(1-3):188-96. doi: 10.1016/j.ejphar.2011.12.013. Epub 2011 Dec 21.

PMID:
22210053
9.

Differential effects of R-isovaline and the GABAB agonist, baclofen, in the guinea pig ileum.

Fung T, Asseri KA, Asiri YI, Wall RA, Schwarz SKW, Puil E, MacLeod BA.

Eur J Pharmacol. 2016 Nov 15;791:85-90. doi: 10.1016/j.ejphar.2016.08.005. Epub 2016 Aug 10.

PMID:
27521870
10.

Actions of thienyl analogs of baclofen at GABA(B) receptors in rat neocortical slices.

Ong J, Kerr DI, Vaccher C, Berthelot P.

Eur J Pharmacol. 1997 Jun 25;329(2-3):133-6.

PMID:
9226405
11.

[Studies of synthesis and structure-activity relationships of analogs of the muscle relaxant--baclofen].

Guo ZW, Tu SZ, Li WH, Chen J.

Yao Xue Xue Bao. 1990;25(1):11-7. Chinese.

PMID:
2163580
12.

GABA heteroreceptors modulate noradrenaline release in human dental pulp.

Parker DA, Marino V.

J Dent Res. 2013 Nov;92(11):1017-21. doi: 10.1177/0022034513505771. Epub 2013 Sep 20.

PMID:
24056226
13.

GABAB receptor subtypes differentially modulate synaptic inhibition in the dentate gyrus to enhance granule cell output.

Foster JD, Kitchen I, Bettler B, Chen Y.

Br J Pharmacol. 2013 Apr;168(8):1808-19. doi: 10.1111/bph.12073.

14.

Pharmacological modulation of GABA(B) receptors affects cocaine-induced seizures in mice.

Gasior M, Kaminski R, Witkin JM.

Psychopharmacology (Berl). 2004 Jul;174(2):211-9.

PMID:
14985936
15.

R-Isovaline: a subtype-specific agonist at GABA(B)-receptors?

Cooke JE, Mathers DA, Puil E.

Neuroscience. 2012 Jan 10;201:85-95. doi: 10.1016/j.neuroscience.2011.10.049. Epub 2011 Nov 4.

PMID:
22079439
16.

Discriminative stimulus effects of the GABAB receptor-positive modulator rac-BHFF: comparison with GABAB receptor agonists and drugs of abuse.

Koek W, Cheng K, Rice KC.

J Pharmacol Exp Ther. 2013 Mar;344(3):553-60. doi: 10.1124/jpet.112.202226. Epub 2012 Dec 28.

17.

In vitro and in vivo characterization of the novel GABAB receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE).

Perdona' E, Costantini VJ, Tessari M, Martinelli P, Carignani C, Valerio E, Mok MH, Zonzini L, Visentini F, Gianotti M, Gordon L, Rocheville M, Corsi M, Capelli AM.

Neuropharmacology. 2011 Oct-Nov;61(5-6):957-66. doi: 10.1016/j.neuropharm.2011.06.024. Epub 2011 Jul 5.

PMID:
21756923
18.

Pharmacological and autoradiographic studies on the pathophysiological role of GABA(B) receptors in the dystonic hamster: pronounced antidystonic effects of baclofen after striatal injections.

Sander SE, Richter F, Raymond R, Diwan M, Lange N, Nobrega JN, Richter A.

Neuroscience. 2009 Aug 18;162(2):423-30. doi: 10.1016/j.neuroscience.2009.05.007. Epub 2009 May 7.

PMID:
19427369
19.

Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid.

Karla R, Ebert B, Thorkildsen C, Herdeis C, Johansen TN, Nielsen B, Krogsgaard-Larsen P.

J Med Chem. 1999 Jun 3;42(11):2053-9.

PMID:
10354414
20.

The anti-spasticity drug baclofen alleviates collagen-induced arthritis and regulates dendritic cells.

Huang S, Mao J, Wei B, Pei G.

J Cell Physiol. 2015 Jul;230(7):1438-47. doi: 10.1002/jcp.24884.

PMID:
25556830

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