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Items: 1 to 20 of 88

1.

6-Bromo-8-(4-[(3)H]methoxybenzamido)-4-oxo-4H-chromene-2-carboxylic Acid: a powerful tool for studying orphan G protein-coupled receptor GPR35.

Thimm D, Funke M, Meyer A, Müller CE.

J Med Chem. 2013 Sep 12;56(17):7084-99. doi: 10.1021/jm4009373. Epub 2013 Aug 15.

PMID:
23888932
2.

8-Benzamidochromen-4-one-2-carboxylic acids: potent and selective agonists for the orphan G protein-coupled receptor GPR35.

Funke M, Thimm D, Schiedel AC, Müller CE.

J Med Chem. 2013 Jun 27;56(12):5182-97. doi: 10.1021/jm400587g. Epub 2013 Jun 17.

PMID:
23713606
3.

Novel diastereomeric opioid tetrapeptides exhibit differing pharmacological activity profiles.

Ioja E, Tourwé D, Kertész I, Tóth G, Borsodi A, Benyhe S.

Brain Res Bull. 2007 Sep 14;74(1-3):119-29. Epub 2007 Jun 8.

PMID:
17683797
4.
5.

[3H]Rauwolscine: an antagonist radioligand for the cloned human 5-hydroxytryptamine2b (5-HT2B) receptor.

Wainscott DB, Sasso DA, Kursar JD, Baez M, Lucaites VL, Nelson DL.

Naunyn Schmiedebergs Arch Pharmacol. 1998 Jan;357(1):17-24.

PMID:
9459568
6.

Use of an inverse agonist radioligand [3H]A-317920 reveals distinct pharmacological profiles of the rat histamine H3 receptor.

Yao BB, Witte DG, Miller TR, Carr TL, Kang CH, Cassar S, Faghih R, Bennani YL, Surber BW, Hancock AA, Esbenshade TA.

Neuropharmacology. 2006 Mar;50(4):468-78. Epub 2005 Nov 28.

PMID:
16316670
7.

Discovery of 2-(4-methylfuran-2(5H)-ylidene)malononitrile and thieno[3,2-b]thiophene-2-carboxylic acid derivatives as G protein-coupled receptor 35 (GPR35) agonists.

Deng H, Hu H, He M, Hu J, Niu W, Ferrie AM, Fang Y.

J Med Chem. 2011 Oct 27;54(20):7385-96. doi: 10.1021/jm200999f. Epub 2011 Oct 4.

8.

6-Bromo-3-hydr-oxy-4-oxo-2-phenyl-4H-chromene-8-carboxylic acid dimethyl-formamide disolvate.

Wen HL, Chen DD, Liu CB.

Acta Crystallogr Sect E Struct Rep Online. 2008 Jul 5;64(Pt 8):o1415. doi: 10.1107/S1600536808019454.

9.

1-Alkyl-benzotriazole-5-carboxylic acids are highly selective agonists of the human orphan G-protein-coupled receptor GPR109b.

Semple G, Skinner PJ, Cherrier MC, Webb PJ, Sage CR, Tamura SY, Chen R, Richman JG, Connolly DT.

J Med Chem. 2006 Feb 23;49(4):1227-30.

PMID:
16480258
10.

[N-methyl-3H3]AZ10419369 binding to the 5-HT1B receptor: in vitro characterization and in vivo receptor occupancy.

Maier DL, Sobotka-Briner C, Ding M, Powell ME, Jiang Q, Hill G, Heys JR, Elmore CS, Pierson ME, Mrzljak L.

J Pharmacol Exp Ther. 2009 Jul;330(1):342-51. doi: 10.1124/jpet.109.150722. Epub 2009 Apr 28.

11.

Novel heterocyclic trans olefin analogues of N-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl}arylcarboxamides as selective probes with high affinity for the dopamine D3 receptor.

Grundt P, Carlson EE, Cao J, Bennett CJ, McElveen E, Taylor M, Luedtke RR, Newman AH.

J Med Chem. 2005 Feb 10;48(3):839-48.

PMID:
15689168
12.

Characterisation of the binding of [3H]-SB-674042, a novel nonpeptide antagonist, to the human orexin-1 receptor.

Langmead CJ, Jerman JC, Brough SJ, Scott C, Porter RA, Herdon HJ.

Br J Pharmacol. 2004 Jan;141(2):340-6. Epub 2003 Dec 22.

13.

Discovery of 2H-Chromen-2-one Derivatives as G Protein-Coupled Receptor-35 Agonists.

Wei L, Wang J, Zhang X, Wang P, Zhao Y, Li J, Hou T, Qu L, Shi L, Liang X, Fang Y.

J Med Chem. 2017 Jan 12;60(1):362-372. doi: 10.1021/acs.jmedchem.6b01431. Epub 2016 Dec 28.

PMID:
27976894
14.

Selective and high affinity labeling of neuronal and recombinant nociceptin receptors with the hexapeptide radioprobe [(3)H]Ac-RYYRIK-ol.

Bojnik E, Farkas J, Magyar A, Tömböly C, Güçlü U, Gündüz O, Borsodi A, Corbani M, Benyhe S.

Neurochem Int. 2009 Dec;55(7):458-66. doi: 10.1016/j.neuint.2009.04.014. Epub 2009 May 4.

PMID:
19414055
15.

[3H] A-369508 ([2-[4-(2-cyanophenyl)-1-piperazinyl]-N-(3-methylphenyl) acetamide): an agonist radioligand selective for the dopamine D4 receptor.

Moreland RB, Terranova MA, Chang R, Uchic ME, Matulenko MA, Surber BW, Stewart AO, Brioni JD.

Eur J Pharmacol. 2004 Aug 23;497(2):147-54.

PMID:
15306199
16.

Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.

Klotz KN, Hessling J, Hegler J, Owman C, Kull B, Fredholm BB, Lohse MJ.

Naunyn Schmiedebergs Arch Pharmacol. 1998 Jan;357(1):1-9.

PMID:
9459566
17.

Development of [(3)H]2-Carboxy-4,6-dichloro-1H-indole-3-propionic Acid ([(3)H]PSB-12150): A Useful Tool for Studying GPR17.

Köse M, Ritter K, Thiemke K, Gillard M, Kostenis E, Müller CE.

ACS Med Chem Lett. 2014 Jan 16;5(4):326-30. doi: 10.1021/ml400399f. eCollection 2014 Apr 10.

18.

2-Phenylimidazo[2,1-i]purin-5-ones: structure-activity relationships and characterization of potent and selective inverse agonists at Human A3 adenosine receptors.

Ozola V, Thorand M, Diekmann M, Qurishi R, Schumacher B, Jacobson KA, Müller CE.

Bioorg Med Chem. 2003 Feb 6;11(3):347-56.

PMID:
12517430
20.

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