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Items: 1 to 20 of 115

1.

Total synthesis and stereochemical assignment of baringolin.

Just-Baringo X, Bruno P, Ottesen LK, Cañedo LM, Albericio F, Álvarez M.

Angew Chem Int Ed Engl. 2013 Jul 22;52(30):7818-21. doi: 10.1002/anie.201302372. Epub 2013 Jun 18.

PMID:
23780649
2.

Total synthesis and biological evaluation of the antibiotic lysocin E and its enantiomeric, epimeric, and N-demethylated analogues.

Murai M, Kaji T, Kuranaga T, Hamamoto H, Sekimizu K, Inoue M.

Angew Chem Int Ed Engl. 2015 Jan 26;54(5):1556-60. doi: 10.1002/anie.201410270. Epub 2014 Dec 11.

PMID:
25504563
3.

Structure determination and total synthesis of bottromycin A2: a potent antibiotic against MRSA and VRE.

Shimamura H, Gouda H, Nagai K, Hirose T, Ichioka M, Furuya Y, Kobayashi Y, Hirono S, Sunazuka T, Omura S.

Angew Chem Int Ed Engl. 2009;48(5):914-7. doi: 10.1002/anie.200804138. No abstract available.

PMID:
19115340
4.

Total synthesis of the thiopeptide amythiamicin D.

Hughes RA, Thompson SP, Alcaraz L, Moody CJ.

Chem Commun (Camb). 2004 Apr 21;(8):946-8. Epub 2004 Mar 16.

PMID:
15069488
5.

Synthesis, in vitro, and in vivo antibacterial activity of nocathiacin I thiol-Michael adducts.

Naidu BN, Sorenson ME, Bronson JJ, Pucci MJ, Clark JM, Ueda Y.

Bioorg Med Chem Lett. 2005 Apr 15;15(8):2069-72.

PMID:
15808470
6.

Total synthesis of thiopeptide antibiotics GE2270A, GE2270T, and GE2270C1.

Nicolaou KC, Dethe DH, Leung GY, Zou B, Chen DY.

Chem Asian J. 2008 Feb 1;3(2):413-29. doi: 10.1002/asia.200700361.

PMID:
18188863
7.

The synthesis of phenylalanine-derived C5-substituted rhodanines and their activity against selected methicillin-resistant Staphylococcus aureus (MRSA) strains.

Hardej D, Ashby CR Jr, Khadtare NS, Kulkarni SS, Singh S, Talele TT.

Eur J Med Chem. 2010 Dec;45(12):5827-32. doi: 10.1016/j.ejmech.2010.09.045. Epub 2010 Sep 25.

PMID:
20947220
8.

Glycopeptides--important treatment option for methicillin-resistant Staphylococcus aureus.

Arora S, Arora U.

Indian J Med Microbiol. 2011 Jul-Sep;29(3):313-4. doi: 10.4103/0255-0857.83922. No abstract available.

9.

Thiol activated prodrugs of sulfur dioxide (SO2) as MRSA inhibitors.

Pardeshi KA, Malwal SR, Banerjee A, Lahiri S, Rangarajan R, Chakrapani H.

Bioorg Med Chem Lett. 2015 Jul 1;25(13):2694-7. doi: 10.1016/j.bmcl.2015.04.046. Epub 2015 Apr 23.

PMID:
25981687
10.

In vitro and in vivo activities of novel, semisynthetic thiopeptide inhibitors of bacterial elongation factor Tu.

Leeds JA, LaMarche MJ, Brewer JT, Bushell SM, Deng G, Dewhurst JM, Dzink-Fox J, Gangl E, Jain A, Lee L, Lilly M, Manni K, Mullin S, Neckermann G, Osborne C, Palestrant D, Patane MA, Raimondi A, Ranjitkar S, Rann EM, Sachdeva M, Shao J, Tiamfook S, Whitehead L, Yu D.

Antimicrob Agents Chemother. 2011 Nov;55(11):5277-83. doi: 10.1128/AAC.00582-11. Epub 2011 Aug 8.

11.

Dissecting the structure of thiopeptides: assessment of thiazoline and tail moieties of baringolin and antibacterial activity optimization.

Just-Baringo X, Bruno P, Pitart C, Vila J, Albericio F, Álvarez M.

J Med Chem. 2014 May 22;57(10):4185-95. doi: 10.1021/jm500062g. Epub 2014 Apr 30.

PMID:
24738558
12.

Restoring methicillin-resistant Staphylococcus aureus susceptibility to β-lactam antibiotics.

Tan CM, Therien AG, Lu J, Lee SH, Caron A, Gill CJ, Lebeau-Jacob C, Benton-Perdomo L, Monteiro JM, Pereira PM, Elsen NL, Wu J, Deschamps K, Petcu M, Wong S, Daigneault E, Kramer S, Liang L, Maxwell E, Claveau D, Vaillancourt J, Skorey K, Tam J, Wang H, Meredith TC, Sillaots S, Wang-Jarantow L, Ramtohul Y, Langlois E, Landry F, Reid JC, Parthasarathy G, Sharma S, Baryshnikova A, Lumb KJ, Pinho MG, Soisson SM, Roemer T.

Sci Transl Med. 2012 Mar 21;4(126):126ra35. doi: 10.1126/scitranslmed.3003592.

13.

Synthesis and evaluation of novel sulfenamides as novel anti Methicillin-resistant Staphylococcus aureus agents.

Shang JL, Guo H, Li ZS, Ren B, Li ZM, Dai HQ, Zhang LX, Wang JG.

Bioorg Med Chem Lett. 2013 Feb 1;23(3):724-7. doi: 10.1016/j.bmcl.2012.11.103. Epub 2012 Dec 3.

PMID:
23265879
14.

Total synthesis and antibiotic activity of dehydrohomoplatencin.

Waalboer DC, Leenders SH, Schülin-Casonato T, van Delft FL, Rutjes FP.

Chemistry. 2010 Oct 4;16(37):11233-6. doi: 10.1002/chem.201001744. No abstract available.

PMID:
20715217
15.

The chemical synthesis and antibiotic activity of a diverse library of 2-aminobenzimidazole small molecules against MRSA and multidrug-resistant A. baumannii.

Huigens RW 3rd, Reyes S, Reed CS, Bunders C, Rogers SA, Steinhauer AT, Melander C.

Bioorg Med Chem. 2010 Jan 15;18(2):663-74. doi: 10.1016/j.bmc.2009.12.003. Epub 2009 Dec 6.

PMID:
20044260
16.

Codon randomization for rapid exploration of chemical space in thiopeptide antibiotic variants.

Young TS, Dorrestein PC, Walsh CT.

Chem Biol. 2012 Dec 21;19(12):1600-10. doi: 10.1016/j.chembiol.2012.10.013.

17.

In vitro susceptibility patterns of methicillin-resistant Staphylococcus aureus and coagulase-negative Staphylococcus corneal isolates to antibiotics.

Elsahn AF, Yildiz EH, Jungkind DL, Abdalla YF, Erdurmus M, Cremona FA, Rapuano CJ, Hammersmith KM, Cohen EJ.

Cornea. 2010 Oct;29(10):1131-5. doi: 10.1097/ICO.0b013e3181d2ce25. Erratum in: Cornea. 2010 Dec;29(12):1470.

PMID:
20595899
18.

Solid-phase synthesis and antibiotic activities of cyclodecapeptides on the scaffold of naturally occurring Laterocidin.

Xu C, Qin C, Zhang R, Niu W, Shang X.

Bioorg Med Chem Lett. 2010 Jan 1;20(1):164-7. doi: 10.1016/j.bmcl.2009.11.009. Epub 2009 Nov 10. Erratum in: Bioorg Med Chem Lett. 2010 Apr 1;20(7):2389.

PMID:
19932962
19.

Bottromycin derivatives: efficient chemical modifications of the ester moiety and evaluation of anti-MRSA and anti-VRE activities.

Kobayashi Y, Ichioka M, Hirose T, Nagai K, Matsumoto A, Matsui H, Hanaki H, Masuma R, Takahashi Y, Omura S, Sunazuka T.

Bioorg Med Chem Lett. 2010 Oct 15;20(20):6116-20. doi: 10.1016/j.bmcl.2010.08.037. Epub 2010 Aug 18.

PMID:
20833545
20.

Increasing levels of minimum inhibitory concentration vancomycin in methicillin resistant Staphylococcus aureus alarming bell for vancomycin abusers?

Veer P, Chande C, Chavan S, Wabale V, Chopdekar K, Bade J, Joshi A.

Indian J Med Microbiol. 2010 Oct-Dec;28(4):413-4. doi: 10.4103/0255-0857.71810. No abstract available.

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