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Items: 1 to 20 of 89

1.

Γ-aminobutyric acid(C) (GABAC) selective antagonists derived from the bioisosteric modification of 4-aminocyclopent-1-enecarboxylic acid: amides and hydroxamates.

Locock KE, Yamamoto I, Tran P, Hanrahan JR, Chebib M, Johnston GA, Allan RD.

J Med Chem. 2013 Jul 11;56(13):5626-30. doi: 10.1021/jm4006548. Epub 2013 Jun 27.

PMID:
23755849
3.

Structural determinants for antagonist pharmacology that distinguish the rho1 GABAC receptor from GABAA receptors.

Zhang J, Xue F, Chang Y.

Mol Pharmacol. 2008 Oct;74(4):941-51. doi: 10.1124/mol.108.048710. Epub 2008 Jul 3.

4.

The effects of cyclopentane and cyclopentene analogues of GABA at recombinant GABA(C) receptors.

Chebib M, Duke RK, Allan RD, Johnston GA.

Eur J Pharmacol. 2001 Nov 2;430(2-3):185-92.

PMID:
11711030
5.

Mixed antagonistic effects of bilobalide at rho1 GABAC receptor.

Huang SH, Duke RK, Chebib M, Sasaki K, Wada K, Johnston GA.

Neuroscience. 2006;137(2):607-17. Epub 2005 Nov 21.

PMID:
16300902
6.

Permeability and single channel conductance of human homomeric rho1 GABAC receptors.

Wotring VE, Chang Y, Weiss DS.

J Physiol. 1999 Dec 1;521 Pt 2:327-36.

7.

Medicinal chemistry of ρ GABAC receptors.

Ng CK, Kim HL, Gavande N, Yamamoto I, Kumar RJ, Mewett KN, Johnston GA, Hanrahan JR, Chebib M.

Future Med Chem. 2011 Feb;3(2):197-209. doi: 10.4155/fmc.10.286. Review.

PMID:
21428815
8.
9.

Unsaturated phosphinic analogues of gamma-aminobutyric acid as GABA(C) receptor antagonists.

Chebib M, Vandenberg RJ, Froestl W, Johnston GA.

Eur J Pharmacol. 1997 Jun 25;329(2-3):223-9.

PMID:
9226416
10.

(3-Aminocyclopentyl)methylphosphinic acids: novel GABA(C) receptor antagonists.

Chebib M, Hanrahan JR, Kumar RJ, Mewett KN, Morriss G, Wooller S, Johnston GA.

Neuropharmacology. 2007 Mar;52(3):779-87. Epub 2006 Nov 13.

PMID:
17098260
11.

Agonist pharmacology of two Drosophila GABA receptor splice variants.

Hosie AM, Sattelle DB.

Br J Pharmacol. 1996 Dec;119(8):1577-85.

12.
13.

Neuroactive steroids and human recombinant rho1 GABAC receptors.

Li W, Jin X, Covey DF, Steinbach JH.

J Pharmacol Exp Ther. 2007 Oct;323(1):236-47. Epub 2007 Jul 17.

15.

Novel gamma-aminobutyric acid rho1 receptor antagonists; synthesis, pharmacological activity and structure-activity relationships.

Kumar RJ, Chebib M, Hibbs DE, Kim HL, Johnston GA, Salam NK, Hanrahan JR.

J Med Chem. 2008 Jul 10;51(13):3825-40. doi: 10.1021/jm7015842. Epub 2008 Jun 5.

PMID:
18528996
16.

5-Substituted imidazole-4-acetic acid analogues: synthesis, modeling, and pharmacological characterization of a series of novel gamma-aminobutyric acid(C) receptor agonists.

Madsen C, Jensen AA, Liljefors T, Kristiansen U, Nielsen B, Hansen CP, Larsen M, Ebert B, Bang-Andersen B, Krogsgaard-Larsen P, Frølund B.

J Med Chem. 2007 Aug 23;50(17):4147-61. Epub 2007 Jul 26.

PMID:
17655213
18.

Actions of cyclic esters, S-esters, and amides of phenyl- and phenylthiophosphonic acids on mammalian and insect GABA-gated chloride channels.

Ozoe Y, Niina K, Matsumoto K, Ikeda I, Mochida K, Ogawa C, Matsuno A, Miki M, Yanagi K.

Bioorg Med Chem. 1998 Jan;6(1):73-83.

PMID:
9502107
19.

Differential effects of quercetin glycosides on GABAC receptor channel activity.

Kim HJ, Lee BH, Choi SH, Jung SW, Kim HS, Lee JH, Hwang SH, Pyo MK, Kim HC, Nah SY.

Arch Pharm Res. 2015 Jan;38(1):108-14. doi: 10.1007/s12272-014-0409-2. Epub 2014 Jun 4.

PMID:
24895146
20.

The enantiomers of syn-2,3-difluoro-4-aminobutyric acid elicit opposite responses at the GABA(C) receptor.

Yamamoto I, Jordan MJ, Gavande N, Doddareddy MR, Chebib M, Hunter L.

Chem Commun (Camb). 2012 Jan 21;48(6):829-31. doi: 10.1039/c1cc15816c. Epub 2011 Dec 5.

PMID:
22143050

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