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Items: 1 to 20 of 125

1.

Synthesis of 1,2,3-triazoles from xylosyl and 5-thioxylosyl azides: evaluation of the xylose scaffold for the design of potential glycogen phosphorylase inhibitors.

Goyard D, Baron M, Skourti PV, Chajistamatiou AS, Docsa T, Gergely P, Chrysina ED, Praly JP, Vidal S.

Carbohydr Res. 2012 Dec 15;364:28-40. doi: 10.1016/j.carres.2012.09.020. Epub 2012 Oct 5.

PMID:
23147043
2.

Synthesis of 5-halogenated 1,2,3-triazoles under stoichiometric Cu(I)-mediated azide-alkyne cycloaddition (CuAAC or 'Click Chemistry').

Goyard D, Praly JP, Vidal S.

Carbohydr Res. 2012 Nov 15;362:79-83. doi: 10.1016/j.carres.2012.08.014. Epub 2012 Sep 11.

PMID:
23124169
3.

Efficient atropodiastereoselective access to 5,5'-bis-1,2,3-triazoles: studies on 1-glucosylated 5-halogeno 1,2,3-triazoles and their 5-substituted derivatives as glycogen phosphorylase inhibitors.

Goyard D, Chajistamatiou AS, Sotiropoulou AI, Chrysina ED, Praly JP, Vidal S.

Chemistry. 2014 Apr 25;20(18):5423-32. doi: 10.1002/chem.201304989. Epub 2014 Mar 27.

PMID:
24677199
4.

Application of click chemistry towards an efficient synthesis of 1,2,3-1H-triazolyl glycohybrids as enzyme inhibitors.

Anand N, Jaiswal N, Pandey SK, Srivastava AK, Tripathi RP.

Carbohydr Res. 2011 Jan 3;346(1):16-25. doi: 10.1016/j.carres.2010.10.017. Epub 2010 Oct 26.

PMID:
21129735
5.

Synthesis of 4-amidomethyl-1-glucosyl-1,2,3-triazoles and evaluation as glycogen phosphorylase inhibitors.

Goyard D, Docsa T, Gergely P, Praly JP, Vidal S.

Carbohydr Res. 2015 Jan 30;402:245-51. doi: 10.1016/j.carres.2014.10.009. Epub 2014 Oct 27.

PMID:
25498027
6.

New synthesis of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4-triazoles, nanomolar inhibitors of glycogen phosphorylase.

Kun S, Bokor É, Varga G, Szőcs B, Páhi A, Czifrák K, Tóth M, Juhász L, Docsa T, Gergely P, Somsák L.

Eur J Med Chem. 2014 Apr 9;76:567-79. doi: 10.1016/j.ejmech.2014.02.041. Epub 2014 Feb 15.

PMID:
24608000
7.
8.

Toward analogues of MraY natural inhibitors: synthesis of 5'-triazole-substituted-aminoribosyl uridines through a Cu-catalyzed azide-alkyne cycloaddition.

Fer MJ, Olatunji S, Bouhss A, Calvet-Vitale S, Gravier-Pelletier C.

J Org Chem. 2013 Oct 18;78(20):10088-105. doi: 10.1021/jo4014035. Epub 2013 Oct 7.

PMID:
24044436
9.

Synthesis of C-xylopyranosyl- and xylopyranosylidene-spiro-heterocycles as potential inhibitors of glycogen phosphorylase.

Somsák L, Bokor É, Czibere B, Czifrák K, Koppány C, Kulcsár L, Kun S, Szilágyi E, Tóth M, Docsa T, Gergely P.

Carbohydr Res. 2014 Nov 18;399:38-48. doi: 10.1016/j.carres.2014.05.020. Epub 2014 Jun 4.

PMID:
25081322
10.

C-Glucopyranosyl-1,2,4-triazol-5-ones: synthesis and inhibition of glycogen phosphorylase.

Bokor É, Széles Z, Docsa T, Gergely P, Somsák L.

Carbohydr Res. 2016 Jun 24;429:128-34. doi: 10.1016/j.carres.2015.12.005. Epub 2015 Dec 24.

PMID:
26818133
11.

Synthesis of novel steroidal 17α-triazolyl derivatives via Cu(I)-catalyzed azide-alkyne cycloaddition, and an evaluation of their cytotoxic activity in vitro.

Frank É, Molnár J, Zupkó I, Kádár Z, Wölfling J.

Steroids. 2011 Sep-Oct;76(10-11):1141-8. doi: 10.1016/j.steroids.2011.05.002. Epub 2011 May 10.

PMID:
21600229
12.

Synthesis of 1-(D-glucopyranosyl)-1,2,3-triazoles and their evaluation as glycogen phosphorylase inhibitors.

Bokor E, Docsa T, Gergely P, Somsák L.

Bioorg Med Chem. 2010 Feb;18(3):1171-80. doi: 10.1016/j.bmc.2009.12.043. Epub 2009 Dec 22.

PMID:
20080412
13.

Synthesis of heterocyclic N-(β-D-glucopyranosyl)carboxamides for inhibition of glycogen phosphorylase.

Kónya B, Docsa T, Gergely P, Somsák L.

Carbohydr Res. 2012 Apr 1;351:56-63. doi: 10.1016/j.carres.2012.01.020. Epub 2012 Jan 31.

PMID:
22365837
14.

Kinetic and crystallographic studies of glucopyranose spirohydantoin and glucopyranosylamine analogs inhibitors of glycogen phosphorylase.

Watson KA, Chrysina ED, Tsitsanou KE, Zographos SE, Archontis G, Fleet GW, Oikonomakos NG.

Proteins. 2005 Dec 1;61(4):966-83.

PMID:
16222658
15.

Synthesis of variously coupled conjugates of D-glucose, 1,3,4-oxadiazole, and 1,2,3-triazole for inhibition of glycogen phosphorylase.

Kun S, Nagy GZ, Tóth M, Czecze L, Van Nhien AN, Docsa T, Gergely P, Charavgi MD, Skourti PV, Chrysina ED, Patonay T, Somsák L.

Carbohydr Res. 2011 Sep 6;346(12):1427-38. doi: 10.1016/j.carres.2011.03.004. Epub 2011 Mar 8.

PMID:
21470596
16.

Synthesis of oleanolic acid dimers as inhibitors of glycogen phosphorylase.

Cheng K, Liu J, Sun H, Xie J.

Chem Biodivers. 2010 Mar;7(3):690-7. doi: 10.1002/cbdv.200900086.

PMID:
20232331
17.
18.

Glucose analog inhibitors of glycogen phosphorylases as potential antidiabetic agents: recent developments.

Somsák L, Nagya V, Hadady Z, Docsa T, Gergely P.

Curr Pharm Des. 2003;9(15):1177-89. Review.

PMID:
12769745
19.

Quick and highly efficient copper-catalyzed cycloaddition of organic azides with terminal alkynes.

Wang D, Zhao M, Liu X, Chen Y, Li N, Chen B.

Org Biomol Chem. 2012 Jan 14;10(2):229-31. doi: 10.1039/c1ob06190a. Epub 2011 Oct 24.

PMID:
22024945
20.

Reversible and competitive cinnamoyl triazole inhibitors of tissue transglutaminase.

Pardin C, Roy I, Lubell WD, Keillor JW.

Chem Biol Drug Des. 2008 Sep;72(3):189-96. doi: 10.1111/j.1747-0285.2008.00696.x. Epub 2008 Aug 19.

PMID:
18715232

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