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Items: 1 to 20 of 158

1.

Effect of C7 modifications on benzothiadiazine-1,1-dioxide derivatives on their inhibitory activity and selectivity toward aldose reductase.

Zhang S, Chen X, Parveen S, Hussain S, Yang Y, Jing C, Zhu C.

ChemMedChem. 2013 Apr;8(4):603-13. doi: 10.1002/cmdc.201200386. Epub 2012 Nov 7.

PMID:
23136050
2.

Correlation of binding constants and molecular modelling of inhibitors in the active sites of aldose reductase and aldehyde reductase.

Carbone V, Zhao HT, Chung R, Endo S, Hara A, El-Kabbani O.

Bioorg Med Chem. 2009 Feb 1;17(3):1244-50. doi: 10.1016/j.bmc.2008.12.024. Epub 2008 Dec 24.

PMID:
19121944
3.

Acetic acid derivatives of 3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxide as a novel class of potent aldose reductase inhibitors.

Chen X, Zhu C, Guo F, Qiu X, Yang Y, Zhang S, He M, Parveen S, Jing C, Li Y, Ma B.

J Med Chem. 2010 Dec 9;53(23):8330-44. doi: 10.1021/jm100962a. Epub 2010 Nov 9.

PMID:
21062005
4.

Discovery of new inhibitors of aldose reductase from molecular docking and database screening.

Rastelli G, Ferrari AM, Costantino L, Gamberini MC.

Bioorg Med Chem. 2002 May;10(5):1437-50.

PMID:
11886806
5.

Coumarin-thiazole and -oxadiazole derivatives: Synthesis, bioactivity and docking studies for aldose/aldehyde reductase inhibitors.

Ibrar A, Tehseen Y, Khan I, Hameed A, Saeed A, Furtmann N, Bajorath J, Iqbal J.

Bioorg Chem. 2016 Oct;68:177-86. doi: 10.1016/j.bioorg.2016.08.005. Epub 2016 Aug 6.

PMID:
27544072
6.

6,7-Dihydroxy-4-phenylcoumarin as inhibitor of aldose reductase 2.

Kato A, Kobayashi K, Narukawa K, Minoshima Y, Adachi I, Hirono S, Nash RJ.

Bioorg Med Chem Lett. 2010 Oct 1;20(19):5630-3. doi: 10.1016/j.bmcl.2010.08.038. Epub 2010 Aug 12.

PMID:
20805028
7.

Pyridothiadiazine derivatives as aldose reductase inhibitors having antioxidant activity.

Zhu S, Zhang S, Hao X, Qin X, Parveen S, Yang S, Ma B, Zhu C.

J Enzyme Inhib Med Chem. 2016;31(sup1):126-130. Epub 2016 May 6.

PMID:
27153454
8.

Synthesis and structure-activity relationship studies of quinoxaline derivatives as aldose reductase inhibitors.

Wu B, Yang Y, Qin X, Zhang S, Jing C, Zhu C, Ma B.

ChemMedChem. 2013 Dec;8(12):1913-7. doi: 10.1002/cmdc.201300324. Epub 2013 Oct 2.

PMID:
24115741
9.

Synthesis and structure-activity relationship of 2-phenyliminochromene derivatives as inhibitors for aldo-keto reductase (AKR) 1B10.

Endo S, Hu D, Suyama M, Matsunaga T, Sugimoto K, Matsuya Y, El-Kabbani O, Kuwata K, Hara A, Kitade Y, Toyooka N.

Bioorg Med Chem. 2013 Nov 1;21(21):6378-84. doi: 10.1016/j.bmc.2013.08.059. Epub 2013 Sep 6.

PMID:
24071447
10.

Synthesis of benzothiadiazine derivatives exhibiting dual activity as aldose reductase inhibitors and antioxidant agents.

Zhu S, Hao X, Zhang S, Qin X, Chen X, Zhu C.

Bioorg Med Chem Lett. 2016 Jun 15;26(12):2880-2885. doi: 10.1016/j.bmcl.2016.04.047. Epub 2016 Apr 20.

PMID:
27156769
11.

Novel, highly potent aldose reductase inhibitors: cyano(2-oxo-2,3-dihydroindol-3-yl)acetic acid derivatives.

Da Settimo F, Primofiore G, Da Settimo A, La Motta C, Simorini F, Novellino E, Greco G, Lavecchia A, Boldrini E.

J Med Chem. 2003 Apr 10;46(8):1419-28.

PMID:
12672241
12.

1,2-Benzothiazine 1,1-dioxide carboxylate derivatives as novel potent inhibitors of aldose reductase.

Chen X, Zhang S, Yang Y, Hussain S, He M, Gui D, Ma B, Jing C, Qiao Z, Zhu C, Yu Q.

Bioorg Med Chem. 2011 Dec 1;19(23):7262-9. doi: 10.1016/j.bmc.2011.07.051. Epub 2011 Jul 30.

PMID:
22036211
13.

Synthesis of derivatives of the keto-pyrrolyl-difluorophenol scaffold: some structural aspects for aldose reductase inhibitory activity and selectivity.

Kotsampasakou E, Demopoulos VJ.

Bioorg Med Chem. 2013 Feb 15;21(4):869-73. doi: 10.1016/j.bmc.2012.12.015. Epub 2012 Dec 20.

PMID:
23312612
14.

Structure-activity relationships studies of quinoxalinone derivatives as aldose reductase inhibitors.

Hussain S, Parveen S, Hao X, Zhang S, Wang W, Qin X, Yang Y, Chen X, Zhu S, Zhu C, Ma B.

Eur J Med Chem. 2014 Jun 10;80:383-92. doi: 10.1016/j.ejmech.2014.04.047. Epub 2014 Apr 21.

PMID:
24793885
15.

Synthesis and structure-activity relationship studies of phenolic hydroxyl derivatives based on quinoxalinone as aldose reductase inhibitors with antioxidant activity.

Hao X, Han Z, Li Y, Li C, Wang X, Zhang X, Yang Q, Ma B, Zhu C.

Bioorg Med Chem Lett. 2017 Feb 15;27(4):887-892. doi: 10.1016/j.bmcl.2017.01.006. Epub 2017 Jan 11.

PMID:
28109789
16.

In vitro evaluation of 5-arylidene-2-thioxo-4-thiazolidinones active as aldose reductase inhibitors.

Maccari R, Del Corso A, Giglio M, Moschini R, Mura U, Ottanà R.

Bioorg Med Chem Lett. 2011 Jan 1;21(1):200-3. doi: 10.1016/j.bmcl.2010.11.041. Epub 2010 Nov 12.

PMID:
21129963
17.

Design and synthesis of potent and selective aldose reductase inhibitors based on pyridylthiadiazine scaffold.

Chen X, Yang Y, Ma B, Zhang S, He M, Gui D, Hussain S, Jing C, Zhu C, Yu Q, Liu Y.

Eur J Med Chem. 2011 May;46(5):1536-44. doi: 10.1016/j.ejmech.2011.01.072. Epub 2011 Mar 1.

PMID:
21367494
18.

Structural bases for the inhibition of aldose reductase by phenolic compounds.

Rastelli G, Antolini L, Benvenuti S, Costantino L.

Bioorg Med Chem. 2000 May;8(5):1151-8.

PMID:
10882025
19.

Structure-based optimization of aldose reductase inhibitors originating from virtual screening.

Eisenmann M, Steuber H, Zentgraf M, Altenkämper M, Ortmann R, Perruchon J, Klebe G, Schlitzer M.

ChemMedChem. 2009 May;4(5):809-19. doi: 10.1002/cmdc.200800410.

PMID:
19301313
20.

[1,2,4]Triazino[4,3-a]benzimidazole acetic acid derivatives: a new class of selective aldose reductase inhibitors.

Da Settimo F, Primofiore G, Da Settimo A, La Motta C, Taliani S, Simorini F, Novellino E, Greco G, Lavecchia A, Boldrini E.

J Med Chem. 2001 Dec 6;44(25):4359-69.

PMID:
11728182

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