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Items: 1 to 20 of 138

1.

Switching the stereochemical outcome of 6-endo-trig cyclizations; synthesis of 2,6-cis-6-substituted 4-oxopipecolic acids.

Daly M, Cant AA, Fowler LS, Simpson GL, Senn HM, Sutherland A.

J Org Chem. 2012 Nov 16;77(22):10001-9. doi: 10.1021/jo3022583. Epub 2012 Nov 8.

PMID:
23126509
2.

A one-pot, reductive amination/6-endo-trig cyclisation for the stereoselective synthesis of 6-substituted-4-oxopipecolic acids.

Fowler LS, Thomas LH, Ellis D, Sutherland A.

Chem Commun (Camb). 2011 Jun 21;47(23):6569-71. doi: 10.1039/c1cc11916h. Epub 2011 May 13.

PMID:
21573277
3.

Synthesis of enantiopure 4-hydroxypipecolate and 4-hydroxylysine derivatives from a common 4,6-dioxopiperidinecarboxylate precursor.

Marin J, Didierjean C, Aubry A, Casimir JR, Briand JP, Guichard G.

J Org Chem. 2004 Jan 9;69(1):130-41.

PMID:
14703388
4.

6-Alkynyl- and 6-aryl-substituted (R)-pipecolic acid derivatives.

Sadiq A, Sewald N.

Org Lett. 2013 Jun 7;15(11):2720-2. doi: 10.1021/ol4010728. Epub 2013 May 29.

PMID:
23718275
5.

Enantioselective synthesis of trans-4-methylpipecolic acid.

Alegret C, Santacana F, Riera A.

J Org Chem. 2007 Sep 28;72(20):7688-92. Epub 2007 Sep 6.

PMID:
17803317
6.

Synthesis of 2-substituted indoles and indolines via Suzuki-Miyaura coupling/5-endo-trig cyclization strategies.

Fuwa H, Sasaki M.

J Org Chem. 2009 Jan 2;74(1):212-21. doi: 10.1021/jo801985a.

PMID:
19007181
7.
8.

The vinylfluoro group as an acetonyl cation equivalent: stereoselective synthesis of 6-substituted 4-hydroxy pipecolic acid derivatives.

Purkayastha N, Shendage DM, Fröhlich R, Haufe G.

J Org Chem. 2010 Jan 1;75(1):222-5. doi: 10.1021/jo901872a.

PMID:
19968262
9.
10.

Recycling the versatile Pipecolic linker.

Zajdel P, Masurier N, Sanchez P, Pawlowski M, Kreiter A, Nomezine G, Enjalbal C, Amblard M, Martinez J, Subra G.

J Comb Chem. 2010 Sep 13;12(5):747-53. doi: 10.1021/cc100099z.

PMID:
20715810
11.

Synthesis of methyl N-Boc-(2S,4R)-4-methylpipecolate.

Hung KY, Harris PW, Brimble MA.

J Org Chem. 2010 Dec 17;75(24):8728-31. doi: 10.1021/jo102038q. Epub 2010 Nov 23.

PMID:
21090804
12.

Intramolecular reductive cyclization strategy to the synthesis of (-)-6-methyl-3-hydroxy-piperidine-2-carboxylic acid, (+)-6-methyl-(2-hydroxymethyl)-piperidine-3-ol and their glycosidase inhibitory activity.

Pawar VU, Chavan ST, Sabharwal SG, Shinde VS.

Bioorg Med Chem. 2010 Nov 15;18(22):7799-803. doi: 10.1016/j.bmc.2010.09.055. Epub 2010 Oct 21.

PMID:
20971014
13.

Synthesis of phosphonic analogues of 4-hydroxyproline and 5-hydroxypipecolic acid.

El Khalabi R, El Hallaoui A, Ouazzani F, Elachqar A, Atmani A, Roumestant ML, Viallefont P, Martinez J.

Prep Biochem Biotechnol. 2000 Nov;30(4):295-304.

PMID:
11065274
14.

Conformationally restricted nonchiral pipecolic acid analogues.

Radchenko DS, Kopylova N, Grygorenko OO, Komarov IV.

J Org Chem. 2009 Aug 7;74(15):5541-4. doi: 10.1021/jo900842w.

PMID:
19518120
15.

Stereoselective access to fluorinated and non-fluorinated quaternary piperidines: synthesis of pipecolic acid and iminosugar derivatives.

Fustero S, Albert L, Mateu N, Chiva G, Miró J, González J, Aceña JL.

Chemistry. 2012 Mar 19;18(12):3753-64. doi: 10.1002/chem.201102351. Epub 2012 Feb 14.

PMID:
22334380
16.

Asymmetric synthesis of a C-3 substituted pipecolic acid.

Souers AJ, Ellman JA.

J Org Chem. 2000 Feb 25;65(4):1222-4. No abstract available.

PMID:
10814077
17.

Diastereoselective synthesis of (2S,5R)-5-hydroxypipecolic acid and 6-substituted derivatives.

Botman PN, Dommerholt FJ, de Gelder R, Broxterman QB, Schoemaker HE, Rutjes FP, Blaauw RH.

Org Lett. 2004 Dec 23;6(26):4941-4.

PMID:
15606105
18.

Stereoconvergent approach for synthesizing enantiopure 5, 6-dialkylpipecolic acids.

Swarbrick ME, Lubell WD.

Chirality. 2000 Jun;12(5-6):366-73.

PMID:
10824154
19.

Controlling the regiochemistry of radical cyclizations.

Ishibashi H.

Chem Rec. 2006;6(1):23-31. Review.

PMID:
16470801
20.

Cationic cyclization of 2-alkenyl-1,3-dithiolanes: diastereoselective synthesis of trans-decalins.

Goncalves S, Santoro S, Nicolas M, Wagner A, Maillos P, Himo F, Baati R.

J Org Chem. 2011 May 6;76(9):3274-85. doi: 10.1021/jo2001116. Epub 2011 Apr 13.

PMID:
21446693

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