Format
Sort by
Items per page

Send to

Choose Destination

Links from PubMed

Items: 1 to 20 of 106

1.

Microwave assisted solid phase synthesis of highly functionalized N-alkylated oligobenzamide α-helix mimetics.

Long K, Edwards TA, Wilson AJ.

Bioorg Med Chem. 2013 Jul 15;21(14):4034-40. doi: 10.1016/j.bmc.2012.09.053. Epub 2012 Oct 3.

2.

Synthesis and screening of small-molecule α-helix mimetic libraries targeting protein-protein interactions.

Moon H, Lim HS.

Curr Opin Chem Biol. 2015 Feb;24:38-47. doi: 10.1016/j.cbpa.2014.10.023. Epub 2014 Nov 15. Review.

PMID:
25461722
3.

Solid-phase synthesis of tris-benzamides as α-helix mimetics.

Lee TK, Ahn JM.

ACS Comb Sci. 2011 Mar 14;13(2):107-11. doi: 10.1021/co100056c. Epub 2010 Dec 1.

PMID:
21395339
4.

Design, solid-phase synthesis, and evaluation of a phenyl-piperazine-triazine scaffold as α-helix mimetics.

Moon H, Lee WS, Oh M, Lee H, Lee JH, Im W, Lim HS.

ACS Comb Sci. 2014 Dec 8;16(12):695-701. doi: 10.1021/co500114f. Epub 2014 Nov 3.

PMID:
25336412
5.

Synthesis of highly functionalized oligobenzamide proteomimetic foldamers by late stage introduction of sensitive groups.

Burslem GM, Kyle HF, Prabhakaran P, Breeze AL, Edwards TA, Warriner SL, Nelson A, Wilson AJ.

Org Biomol Chem. 2016 Apr 12;14(15):3782-6. doi: 10.1039/c6ob00078a.

6.

Solid-phase methodology for synthesis of O-alkylated aromatic oligoamide inhibitors of α-helix-mediated protein-protein interactions.

Murphy NS, Prabhakaran P, Azzarito V, Plante JP, Hardie MJ, Kilner CA, Warriner SL, Wilson AJ.

Chemistry. 2013 Apr 26;19(18):5546-50. doi: 10.1002/chem.201204098. Epub 2013 Mar 18.

7.

2-O-alkylated para-benzamide α-helix mimetics: the role of scaffold curvature.

Azzarito V, Prabhakaran P, Bartlett AI, Murphy NS, Hardie MJ, Kilner CA, Edwards TA, Warriner SL, Wilson AJ.

Org Biomol Chem. 2012 Aug 28;10(32):6469-72. doi: 10.1039/c2ob26262b. Epub 2012 Jul 11.

PMID:
22785578
8.

N-alkylated oligoamide alpha-helical proteomimetics.

Campbell F, Plante JP, Edwards TA, Warriner SL, Wilson AJ.

Org Biomol Chem. 2010 May 21;8(10):2344-51. doi: 10.1039/c001164a. Epub 2010 Mar 18.

PMID:
20448891
9.

Comprehensive peptidomimetic libraries targeting protein-protein interactions.

Whitby LR, Boger DL.

Acc Chem Res. 2012 Oct 16;45(10):1698-709. doi: 10.1021/ar300025n. Epub 2012 Jul 16.

10.

Probing Protein Surfaces: QSAR Analysis with Helix Mimetics.

Azzarito V, Rowell P, Barnard A, Edwards TA, Macdonald A, Warriner SL, Wilson AJ.

Chembiochem. 2016 Apr 15;17(8):768-73. doi: 10.1002/cbic.201500504. Epub 2016 Jan 21.

PMID:
26690307
11.

Synthesis of Pyridazine-Based α-Helix Mimetics.

Londregan AT, Piotrowski DW, Wei L.

ACS Comb Sci. 2016 Oct 10;18(10):651-654. Epub 2016 Sep 14.

PMID:
27571162
12.

Oligophenylenaminones as scaffolds for α-helix mimicry.

Adler MJ, Hamilton AD.

J Org Chem. 2011 Sep 2;76(17):7040-7. doi: 10.1021/jo200917d. Epub 2011 Aug 3.

PMID:
21739975
13.

Small-molecule proteomimetic inhibitors of the HIF-1α-p300 protein-protein interaction.

Burslem GM, Kyle HF, Breeze AL, Edwards TA, Nelson A, Warriner SL, Wilson AJ.

Chembiochem. 2014 May 26;15(8):1083-7. doi: 10.1002/cbic.201400009. Epub 2014 Apr 29.

14.

Traceless solid-phase synthesis of 2,4,6-trisubstituted thiazolo[4,5-d]pyrimidine-5,7-dione derivatives.

Lee T, Park JH, Lee DH, Gong YD.

J Comb Chem. 2009 May-Jun;11(3):495-9. doi: 10.1021/cc900023s.

PMID:
19338271
15.

Disrupting protein-protein interactions with non-peptidic, small molecule alpha-helix mimetics.

Cummings CG, Hamilton AD.

Curr Opin Chem Biol. 2010 Jun;14(3):341-6. doi: 10.1016/j.cbpa.2010.04.001. Epub 2010 Apr 27. Review.

PMID:
20430687
16.

Converting One-Face α-Helix Mimetics into Amphiphilic α-Helix Mimetics as Potent Inhibitors of Protein-Protein Interactions.

Lee JH, Oh M, Kim HS, Lee H, Im W, Lim HS.

ACS Comb Sci. 2016 Jan 11;18(1):36-42. doi: 10.1021/acscombsci.5b00080. Epub 2015 Dec 22.

PMID:
26651509
17.

Non-peptidic α-helical mimetics as protein-protein interaction inhibitors.

Dewal MB, Firestine SM.

Curr Med Chem. 2011;18(16):2420-8. Review.

PMID:
21568916
18.

Microwave-assisted diastereoselective two-step three-component synthesis for rapid access to drug-like libraries of substituted 3-amino-β-lactams.

Janssen GV, van den Heuvel JAC, Megens RP, Benningshof JCJ, Ovaa H.

Bioorg Med Chem. 2018 Jan 1;26(1):41-49. doi: 10.1016/j.bmc.2017.11.014. Epub 2017 Nov 16.

19.

Synthesis of isoxazolo[5,4-b]pyridines by microwave-assisted multi-component reactions in water.

Tu SJ, Zhang XH, Han ZG, Cao XD, Wu SS, Yan S, Hao WJ, Zhang G, Ma N.

J Comb Chem. 2009 May-Jun;11(3):428-32. doi: 10.1021/cc800212v.

PMID:
19364093
20.

Microwave-assisted solid-phase synthesis of antifreeze glycopeptides.

Izumi R, Matsushita T, Fujitani N, Naruchi K, Shimizu H, Tsuda S, Hinou H, Nishimura S.

Chemistry. 2013 Mar 18;19(12):3913-20. doi: 10.1002/chem.201203731. Epub 2013 Feb 10.

PMID:
23401082

Supplemental Content

Support Center