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Items: 1 to 20 of 91

1.

Discovery of the first irreversible small molecule inhibitors of the interaction between the vitamin D receptor and coactivators.

Nandhikonda P, Lynt WZ, McCallum MM, Ara T, Baranowski AM, Yuan NY, Pearson D, Bikle DD, Guy RK, Arnold LA.

J Med Chem. 2012 May 24;55(10):4640-51. doi: 10.1021/jm300460c. Epub 2012 May 16.

2.

Inhibitors for the Vitamin D Receptor-Coregulator Interaction.

Teske KA, Yu O, Arnold LA.

Vitam Horm. 2016;100:45-82. doi: 10.1016/bs.vh.2015.10.002. Epub 2015 Nov 30. Review.

3.

Development of novel Vitamin D Receptor-Coactivator Inhibitors.

Sidhu PS, Nassif N, McCallum MM, Teske K, Feleke B, Yuan NY, Nandhikonda P, Cook JM, Singh RK, Bikle DD, Arnold LA.

ACS Med Chem Lett. 2014 Feb 13;5(2):199-204.

4.

Vitamin D receptor and coactivators SRC2 and 3 regulate epidermis-specific sphingolipid production and permeability barrier formation.

Oda Y, Uchida Y, Moradian S, Crumrine D, Elias PM, Bikle DD.

J Invest Dermatol. 2009 Jun;129(6):1367-78. doi: 10.1038/jid.2008.380. Epub 2008 Dec 4.

5.

Ternary complexes and cooperative interplay between NCoA-62/Ski-interacting protein and steroid receptor coactivators in vitamin D receptor-mediated transcription.

Zhang C, Baudino TA, Dowd DR, Tokumaru H, Wang W, MacDonald PN.

J Biol Chem. 2001 Nov 2;276(44):40614-20. Epub 2001 Aug 20.

6.

Vitamin D analogue-specific recruitment of vitamin D receptor coactivators.

Issa LL, Leong GM, Sutherland RL, Eisman JA.

J Bone Miner Res. 2002 May;17(5):879-90.

7.

Nuclear coactivator-62 kDa/Ski-interacting protein is a nuclear matrix-associated coactivator that may couple vitamin D receptor-mediated transcription and RNA splicing.

Zhang C, Dowd DR, Staal A, Gu C, Lian JB, van Wijnen AJ, Stein GS, MacDonald PN.

J Biol Chem. 2003 Sep 12;278(37):35325-36. Epub 2003 Jul 2.

8.

The vitamin D hormone and its nuclear receptor: molecular actions and disease states.

Haussler MR, Haussler CA, Jurutka PW, Thompson PD, Hsieh JC, Remus LS, Selznick SH, Whitfield GK.

J Endocrinol. 1997 Sep;154 Suppl:S57-73. Review.

9.

Coactivator-vitamin D receptor interactions mediate inhibition of the atrial natriuretic peptide promoter.

Chen S, Cui J, Nakamura K, Ribeiro RC, West BL, Gardner DG.

J Biol Chem. 2000 May 19;275(20):15039-48.

10.

Peroxisome proliferation-activated receptor δ agonist GW0742 interacts weakly with multiple nuclear receptors, including the vitamin D receptor.

Nandhikonda P, Yasgar A, Baranowski AM, Sidhu PS, McCallum MM, Pawlak AJ, Teske K, Feleke B, Yuan NY, Kevin C, Bikle DD, Ayers SD, Webb P, Rai G, Simeonov A, Jadhav A, Maloney D, Arnold LA.

Biochemistry. 2013 Jun 18;52(24):4193-203. doi: 10.1021/bi400321p. Epub 2013 Jun 10.

11.

Development of stapled short helical peptides capable of inhibiting vitamin D receptor (VDR)-coactivator interactions.

Demizu Y, Nagoya S, Shirakawa M, Kawamura M, Yamagata N, Sato Y, Doi M, Kurihara M.

Bioorg Med Chem Lett. 2013 Aug 1;23(15):4292-6. doi: 10.1016/j.bmcl.2013.06.002. Epub 2013 Jun 10.

PMID:
23806555
13.

Evidence for ligand-dependent intramolecular folding of the AF-2 domain in vitamin D receptor-activated transcription and coactivator interaction.

Masuyama H, Brownfield CM, St-Arnaud R, MacDonald PN.

Mol Endocrinol. 1997 Sep;11(10):1507-17.

PMID:
9280066
14.

LXXLL peptide mimetics as inhibitors of the interaction of vitamin D receptor with coactivators.

Mita Y, Dodo K, Noguchi-Yachide T, Miyachi H, Makishima M, Hashimoto Y, Ishikawa M.

Bioorg Med Chem Lett. 2010 Mar 1;20(5):1712-7. doi: 10.1016/j.bmcl.2010.01.079. Epub 2010 Jan 21.

PMID:
20144545
15.
16.
17.

Sequential regulation of keratinocyte differentiation by 1,25(OH)2D3, VDR, and its coregulators.

Bikle D, Teichert A, Hawker N, Xie Z, Oda Y.

J Steroid Biochem Mol Biol. 2007 Mar;103(3-5):396-404. Epub 2007 Jan 16.

PMID:
17229570
18.

Vitamin D receptor and nuclear receptor coactivators: crucial interactions in vitamin D-mediated transcription.

MacDonald PN, Baudino TA, Tokumaru H, Dowd DR, Zhang C.

Steroids. 2001 Mar-May;66(3-5):171-6. Review.

PMID:
11179724
19.

The 1,25(OH)2D3-regulated transcription factor MN1 stimulates vitamin D receptor-mediated transcription and inhibits osteoblastic cell proliferation.

Sutton AL, Zhang X, Ellison TI, Macdonald PN.

Mol Endocrinol. 2005 Sep;19(9):2234-44. Epub 2005 May 12.

PMID:
15890672
20.

Regulation of human epidermal keratinocyte differentiation by the vitamin D receptor and its coactivators DRIP205, SRC2, and SRC3.

Hawker NP, Pennypacker SD, Chang SM, Bikle DD.

J Invest Dermatol. 2007 Apr;127(4):874-80. Epub 2006 Nov 2.

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