Format
Sort by

Send to

Choose Destination

Links from PubMed

Items: 1 to 20 of 98

1.

Utilization of [11C]phosgene for radiosynthesis of N-(2-{3-[3,5-bis(trifluoromethyl)]phenyl[11C]ureido}ethyl)glycyrrhetinamide, an inhibitory agent for proteasome and kinase in tumors.

Asakawa C, Ogawa M, Fujinaga M, Kumata K, Xie L, Yamasaki T, Yui J, Fukumura T, Zhang MR.

Bioorg Med Chem Lett. 2012 Jun 1;22(11):3594-7. doi: 10.1016/j.bmcl.2012.04.049.

PMID:
22546673
2.

N-(2-{3-[3,5-bis(trifluoromethyl)phenyl]ureido}ethyl)-glycyrrhetinamide (6b): a novel anticancer glycyrrhetinic acid derivative that targets the proteasome and displays anti-kinase activity.

Lallemand B, Chaix F, Bury M, Bruyère C, Ghostin J, Becker JP, Delporte C, Gelbcke M, Mathieu V, Dubois J, Prévost M, Jabin I, Kiss R.

J Med Chem. 2011 Oct 13;54(19):6501-13. doi: 10.1021/jm200285z.

PMID:
21888390
3.

Radiosynthesis of three [11C]ureido-substituted benzenesulfonamides as PET probes for carbonic anhydrase IX in tumors.

Asakawa C, Ogawa M, Kumata K, Fujinaga M, Yamasaki T, Xie L, Yui J, Kawamura K, Fukumura T, Zhang MR.

Bioorg Med Chem Lett. 2011 Dec 1;21(23):7017-20. doi: 10.1016/j.bmcl.2011.09.102.

PMID:
22014831
4.

Radiosynthesis of [2-(11)C-carbonyl]dantrolene using [(11)C]phosgene for PET.

Takada Y, Ogawa M, Suzuki H, Fukumura T.

Appl Radiat Isot. 2010 Sep;68(9):1715-20. doi: 10.1016/j.apradiso.2010.03.012.

PMID:
20395154
5.

[11C]sorafenib: radiosynthesis and preliminary PET study of brain uptake in P-gp/Bcrp knockout mice.

Asakawa C, Ogawa M, Kumata K, Fujinaga M, Kato K, Yamasaki T, Yui J, Kawamura K, Hatori A, Fukumura T, Zhang MR.

Bioorg Med Chem Lett. 2011 Apr 15;21(8):2220-3. doi: 10.1016/j.bmcl.2011.03.002.

PMID:
21419625
6.

Synthesis and plasma pharmacokinetics in CD-1 mice of a 18β-glycyrrhetinic acid derivative displaying anti-cancer activity.

Lallemand B, Ouedraogo M, Wauthoz N, Lamkami T, Mathieu V, Jabin I, Amighi K, Kiss R, Dubois J, Goole J.

J Pharm Pharmacol. 2013 Mar;65(3):402-10. doi: 10.1111/j.2042-7158.2012.01603.x.

PMID:
23356849
7.

An automated radiosynthesis of 2-[11C]thymidine using anhydrous [11C]urea derived from [11C]phosgene.

Steel CJ, Brady F, Luthra SK, Brown G, Khan I, Poole KG, Sergis A, Jones T, Price PM.

Appl Radiat Isot. 1999 Oct;51(4):377-88.

PMID:
10464914
9.

A simplified and improved synthesis of [11C]phosgene with iron and iron (III) oxide.

Nishijima K, Kuge Y, Seki K, Ohkura K, Motoki N, Nagatsu K, Tanaka A, Tsukamoto E, Tamaki N.

Nucl Med Biol. 2002 Apr;29(3):345-50.

PMID:
11929705
10.
11.

Radiosynthesis of [13N]dantrolene, a positron emission tomography probe for breast cancer resistant protein, using no-carrier-added [13N]ammonia.

Kumata K, Ogawa M, Takei M, Fujinaga M, Yoshida Y, Nengaki N, Fukumura T, Suzuki K, Zhang MR.

Bioorg Med Chem. 2012 Jan 1;20(1):305-10. doi: 10.1016/j.bmc.2011.10.077.

PMID:
22115838
12.

Synthesis and biological evaluation of novel spin labeled 18β-glycyrrhetinic acid derivatives.

Liu Y, Qian K, Wang CY, Chen CH, Yang X, Lee KH.

Bioorg Med Chem Lett. 2012 Dec 15;22(24):7530-3. doi: 10.1016/j.bmcl.2012.10.041.

PMID:
23122524
13.
14.

[(11)C-carbonyl]CEP-32496: radiosynthesis, biodistribution and PET study of brain uptake in P-gp/BCRP knockout mice.

Shimoda Y, Yui J, Fujinaga M, Xie L, Kumata K, Ogawa M, Yamasaki T, Hatori A, Kawamura K, Zhang MR.

Bioorg Med Chem Lett. 2014 Aug 1;24(15):3574-7. doi: 10.1016/j.bmcl.2014.05.045.

PMID:
24930831
15.

A novel and efficient synthesis of [2-11C]5-fluorouracil for prognosis of cancer chemotherapy.

Seki K, Nishijima K, Kuge Y, Tamaki N, Wiebe LI, Ohkura K.

J Pharm Pharm Sci. 2007;10(2):212-6.

16.

Synthesis and proteasome inhibition of glycyrrhetinic acid derivatives.

Huang L, Yu D, Ho P, Qian K, Lee KH, Chen CH.

Bioorg Med Chem. 2008 Jul 15;16(14):6696-701. doi: 10.1016/j.bmc.2008.05.078.

17.

[11C]-dimethylamine as a labeling agent for PET biomarkers.

Jacobson O, Mishani E.

Appl Radiat Isot. 2008 Feb;66(2):188-93.

PMID:
17923410
18.

Synthesis, radiolabeling and initial in vivo evaluation of [(11)C]KSM-01 for imaging PPAR-α receptors.

Solingapuram Sai KK, Kil KE, Tu Z, Chu W, Finck BN, Rothfuss JM, Shoghi KI, Welch MJ, Gropler RJ, Mach RH.

Bioorg Med Chem Lett. 2012 Oct 1;22(19):6233-6. doi: 10.1016/j.bmcl.2012.08.010.

19.

An efficient and expedient method for the synthesis of 11C-labeled α-aminoisobutyric acid: a tumor imaging agent potentially useful for cancer diagnosis.

Kato K, Tsuji AB, Saga T, Zhang MR.

Bioorg Med Chem Lett. 2011 Apr 15;21(8):2437-40. doi: 10.1016/j.bmcl.2011.02.065.

PMID:
21392981
20.

Two routes to [11C-carbonyl]organo-isocyanates utilizing [11C]phosgene ([11C]organo-isocyanates from [11C]phosgene).

Brown GD, Henderson D, Steel C, Luthra S, Price PM, Brady F.

Nucl Med Biol. 2001 Nov;28(8):991-8.

PMID:
11711319
Items per page

Supplemental Content

Support Center