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Items: 1 to 20 of 146

1.

Synthesis and biological evaluation of acridine derivatives as antimalarial agents.

Yu XM, Ramiandrasoa F, Guetzoyan L, Pradines B, Quintino E, Gadelle D, Forterre P, Cresteil T, Mahy JP, Pethe S.

ChemMedChem. 2012 Apr;7(4):587-605. doi: 10.1002/cmdc.201100554.

PMID:
22331612
2.

Antimalarial acridines: synthesis, in vitro activity against P. falciparum and interaction with hematin.

Guetzoyan L, Yu XM, Ramiandrasoa F, Pethe S, Rogier C, Pradines B, Cresteil T, Perrée-Fauvet M, Mahy JP.

Bioorg Med Chem. 2009 Dec 1;17(23):8032-9. doi: 10.1016/j.bmc.2009.10.005.

PMID:
19879150
3.

In vitro efficiency of new acridyl derivatives against Plasmodium falciparum.

Guetzoyan L, Ramiandrasoa F, Dorizon H, Desprez C, Bridoux A, Rogier C, Pradines B, Perrée-Fauvet M.

Bioorg Med Chem. 2007 May 1;15(9):3278-89.

PMID:
17339112
4.

Synthesis, antimalarial activity, and cellular toxicity of new arylpyrrolylaminoquinolines.

Casagrande M, Basilico N, Rusconi C, Taramelli D, Sparatore A.

Bioorg Med Chem. 2010 Sep 15;18(18):6625-33. doi: 10.1016/j.bmc.2010.08.001.

PMID:
20797868
5.

Design, synthesis, and structure-activity relationship studies of 4-quinolinyl- and 9-acrydinylhydrazones as potent antimalarial agents.

Fattorusso C, Campiani G, Kukreja G, Persico M, Butini S, Romano MP, Altarelli M, Ros S, Brindisi M, Savini L, Novellino E, Nacci V, Fattorusso E, Parapini S, Basilico N, Taramelli D, Yardley V, Croft S, Borriello M, Gemma S.

J Med Chem. 2008 Mar 13;51(5):1333-43. doi: 10.1021/jm7012375.

PMID:
18278859
6.

Synthesis of N1-arylidene-N2-quinolyl- and N2-acrydinylhydrazones as potent antimalarial agents active against CQ-resistant P. falciparum strains.

Gemma S, Kukreja G, Fattorusso C, Persico M, Romano MP, Altarelli M, Savini L, Campiani G, Fattorusso E, Basilico N, Taramelli D, Yardley V, Butini S.

Bioorg Med Chem Lett. 2006 Oct 15;16(20):5384-8.

PMID:
16890433
7.

Synthesis and antimalarial activity in vitro of potential metabolites of ferrochloroquine and related compounds.

Biot C, Delhaes L, N'Diaye CM, Maciejewski LA, Camus D, Dive D, Brocard JS.

Bioorg Med Chem. 1999 Dec;7(12):2843-7.

PMID:
10658588
8.

Synthesis and antimalarial activity of new heterocyclic hybrids based on chloroquine and thiazolidinone scaffolds.

Rojas Ruiz FA, García-Sánchez RN, Estupiñan SV, Gómez-Barrio A, Torres Amado DF, Pérez-Solórzano BM, Nogal-Ruiz JJ, Martínez-Fernández AR, Kouznetsov VV.

Bioorg Med Chem. 2011 Aug 1;19(15):4562-73. doi: 10.1016/j.bmc.2011.06.025.

PMID:
21723734
9.

Synthesis of new 4-aminoquinolines and quinoline-acridine hybrids as antimalarial agents.

Kumar A, Srivastava K, Kumar SR, Puri SK, Chauhan PM.

Bioorg Med Chem Lett. 2010 Dec 1;20(23):7059-63. doi: 10.1016/j.bmcl.2010.09.107.

PMID:
20951034
10.

Pharmacomodulation on the 3-acetylursolic acid skeleton: Design, synthesis, and biological evaluation of novel N-{3-[4-(3-aminopropyl)piperazinyl]propyl}-3-O-acetylursolamide derivatives as antimalarial agents.

Gnoatto SC, Susplugas S, Dalla Vechia L, Ferreira TB, Dassonville-Klimpt A, Zimmer KR, Demailly C, Da Nascimento S, Guillon J, Grellier P, Verli H, Gosmann G, Sonnet P.

Bioorg Med Chem. 2008 Jan 15;16(2):771-82.

PMID:
17967541
11.

Indolone-N-oxide derivatives: in vitro activity against fresh clinical isolates of Plasmodium falciparum, stage specificity and in vitro interactions with established antimalarial drugs.

Tahar R, Vivas L, Basco L, Thompson E, Ibrahim H, Boyer J, Nepveu F.

J Antimicrob Chemother. 2011 Nov;66(11):2566-72. doi: 10.1093/jac/dkr320.

PMID:
21862474
12.

Synthesis and antimalarial evaluation of new 1,4-bis(3-aminopropyl)piperazine derivatives.

Ryckebusch A, Deprez-Poulain R, Debreu-Fontaine MA, Vandaele R, Mouray E, Grellier P, Sergheraert C.

Bioorg Med Chem Lett. 2003 Nov 3;13(21):3783-7.

PMID:
14552779
13.

Synthesis and evaluation of 1-amino-6-halo-β-carbolines as antimalarial and antiprion agents.

Thompson MJ, Louth JC, Little SM, Jackson MP, Boursereau Y, Chen B, Coldham I.

ChemMedChem. 2012 Apr;7(4):578-86. doi: 10.1002/cmdc.201200002.

PMID:
22275299
14.

Synthesis and evaluation of sulfonylurea derivatives as novel antimalarials.

León C, Rodrigues J, Gamboa de Domínguez N, Charris J, Gut J, Rosenthal PJ, Domínguez JN.

Eur J Med Chem. 2007 Jun;42(6):735-42.

PMID:
17321641
15.

A prodrug form of a Plasmodium falciparum glutathione reductase inhibitor conjugated with a 4-anilinoquinoline.

Davioud-Charvet E, Delarue S, Biot C, Schwöbel B, Boehme CC, Müssigbrodt A, Maes L, Sergheraert C, Grellier P, Schirmer RH, Becker K.

J Med Chem. 2001 Nov 22;44(24):4268-76.

PMID:
11708927
17.

Antimalarial t-butylperoxyamines.

Sundar N, Jacob VT, Bhat SV, Valecha N, Biswas S.

Bioorg Med Chem Lett. 2001 Sep 3;11(17):2269-72.

PMID:
11527712
18.

Synthesis and evaluation of the antiplasmodial activity of novel indeno[2,1-c]quinoline derivatives.

Barteselli A, Parapini S, Basilico N, Mommo D, Sparatore A.

Bioorg Med Chem. 2014 Nov 1;22(21):5757-65. doi: 10.1016/j.bmc.2014.09.040.

PMID:
25311562
19.

New quinoline-5,8-dione and hydroxynaphthoquinone derivatives inhibit a chloroquine resistant Plasmodium falciparum strain.

Hussain H, Specht S, Sarite SR, Hoerauf A, Krohn K.

Eur J Med Chem. 2012 Aug;54:936-42. doi: 10.1016/j.ejmech.2012.06.046.

PMID:
22781704
20.

Antimalarial activity of new acridinone derivatives.

Fernández-Calienes A, Pellón R, Docampo M, Fascio M, D'Accorso N, Maes L, Mendiola J, Monzote L, Gille L, Rojas L.

Biomed Pharmacother. 2011 Jun;65(3):210-4. doi: 10.1016/j.biopha.2011.04.001.

PMID:
21641752

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