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Items: 1 to 20 of 109

1.

Boron cluster-based development of potent nonsecosteroidal vitamin D receptor ligands: direct observation of hydrophobic interaction between protein surface and carborane.

Fujii S, Masuno H, Taoda Y, Kano A, Wongmayura A, Nakabayashi M, Ito N, Shimizu M, Kawachi E, Hirano T, Endo Y, Tanatani A, Kagechika H.

J Am Chem Soc. 2011 Dec 28;133(51):20933-41. doi: 10.1021/ja208797n. Epub 2011 Nov 30.

PMID:
22066785
2.

Novel vitamin D receptor ligands bearing a spherical hydrophobic core structure--comparison of bicyclic hydrocarbon derivatives with boron cluster derivatives.

Wongmayura A, Fujii S, Ito S, Kano A, Taoda Y, Kawachi E, Kagechika H, Tanatani A.

Bioorg Med Chem Lett. 2012 Feb 15;22(4):1756-60. doi: 10.1016/j.bmcl.2011.12.137. Epub 2012 Jan 10.

PMID:
22285943
3.

Structural development of p-carborane-based potent non-secosteroidal vitamin D analogs.

Fujii S, Sekine R, Kano A, Masuno H, Songkram C, Kawachi E, Hirano T, Tanatani A, Kagechika H.

Bioorg Med Chem. 2014 Nov 1;22(21):5891-901. doi: 10.1016/j.bmc.2014.09.020. Epub 2014 Sep 16.

PMID:
25284253
4.

Design and synthesis of tetraol derivatives of 1,12-dicarba-closo-dodecaborane as non-secosteroidal vitamin D analogs.

Fujii S, Kano A, Masuno H, Songkram C, Kawachi E, Hirano T, Tanatani A, Kagechika H.

Bioorg Med Chem Lett. 2014 Sep 15;24(18):4515-9. doi: 10.1016/j.bmcl.2014.07.075. Epub 2014 Aug 6.

PMID:
25149512
5.

Potent estrogen agonists based on carborane as a hydrophobic skeletal structure. A new medicinal application of boron clusters.

Endo Y, Iijima T, Yamakoshi Y, Fukasawa H, Miyaura C, Inada M, Kubo A, Itai A.

Chem Biol. 2001 Apr;8(4):341-55.

6.

Design, synthesis and X-ray crystallographic study of new nonsecosteroidal vitamin D receptor ligands.

Demizu Y, Takahashi T, Kaneko F, Sato Y, Okuda H, Ochiai E, Horie K, Takagi K, Kakuda S, Takimoto-Kamimura M, Kurihara M.

Bioorg Med Chem Lett. 2011 Oct 15;21(20):6104-7. doi: 10.1016/j.bmcl.2011.08.047. Epub 2011 Aug 17.

PMID:
21889334
7.

Synthesis and structure-activity relationship of p-carborane-based non-secosteroidal vitamin D analogs.

Fujii S, Kano A, Songkram C, Masuno H, Taoda Y, Kawachi E, Hirano T, Tanatani A, Kagechika H.

Bioorg Med Chem. 2014 Feb 15;22(4):1227-35. doi: 10.1016/j.bmc.2014.01.015. Epub 2014 Jan 21.

PMID:
24486205
8.

Dicarba-closo-dodecaboranes as a pharmacophore. Novel potent retinoidal agonists.

Endo Y, Iijima T, Kagechika H, Ohta K, Kawachi E, Shudo K.

Chem Pharm Bull (Tokyo). 1999 Apr;47(4):585-7.

PMID:
10319433
9.

Novel retinoid X receptor (RXR) antagonists having a dicarba-closo-dodecaborane as a hydrophobic moiety.

Ohta K, Iijima T, Kawachi E, Kagechika H, Endo Y.

Bioorg Med Chem Lett. 2004 Dec 6;14(23):5913-8.

PMID:
15501068
10.

Potent androgen antagonists based on carborane as a hydrophobic core structure.

Fujii S, Goto T, Ohta K, Hashimoto Y, Suzuki T, Ohta S, Endo Y.

J Med Chem. 2005 Jul 14;48(14):4654-62.

PMID:
16000001
11.

Crystal structure, docking study and structure-activity relationship of carborane-containing androgen receptor antagonist 3-(12-hydroxymethyl-1,12-dicarba-closo-dodecaboran-1-yl)benzonitrile.

Ohta K, Goto T, Fujii S, Kawahata M, Oda A, Ohta S, Yamaguchi K, Hirono S, Endo Y.

Bioorg Med Chem. 2011 Jun 1;19(11):3540-8. doi: 10.1016/j.bmc.2011.04.017. Epub 2011 Apr 20.

PMID:
21536446
12.
13.

Ligand binding domain of vitamin D receptors.

Rochel N, Moras D.

Curr Top Med Chem. 2006;6(12):1229-41. Review.

PMID:
16848737
14.

Protein kinase C modulators bearing dicarba-CLOSO-dodecaborane as a hydrophobic pharmacophore.

Endo Y, Yoshimi T, Kimura K, Itai A.

Bioorg Med Chem Lett. 1999 Sep 6;9(17):2561-4.

PMID:
10498208
15.
16.

Crystal structures of the vitamin D receptor complexed to superagonist 20-epi ligands.

Tocchini-Valentini G, Rochel N, Wurtz JM, Mitschler A, Moras D.

Proc Natl Acad Sci U S A. 2001 May 8;98(10):5491-6.

17.
18.

(2,2':6',2' '-Terpyridine)platinum(II) complexes containing (thioalkyl)dicarba-closo-dodecaborane(12) ligands.

Todd JA, Turner P, Ziolkowski EJ, Rendina LM.

Inorg Chem. 2005 Sep 5;44(18):6401-8.

PMID:
16124820
19.

Ligand recognition by the vitamin D receptor.

Choi M, Yamamoto K, Masuno H, Nakashima K, Taga T, Yamada S.

Bioorg Med Chem. 2001 Jul;9(7):1721-30.

PMID:
11425573
20.

New estrogenic antagonists bearing dicarba-closo-dodecaborane as a hydrophobic pharmacophore.

Endo Y, Yoshimi T, Yamakoshi Y.

Chem Pharm Bull (Tokyo). 2000 Feb;48(2):312-4.

PMID:
10705532

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