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Computational reverse-engineering of a spider-venom derived peptide active against Plasmodium falciparum SUB1.

Bastianelli G, Bouillon A, Nguyen C, Crublet E, Pêtres S, Gorgette O, Le-Nguyen D, Barale JC, Nilges M.

PLoS One. 2011;6(7):e21812. doi: 10.1371/journal.pone.0021812. Epub 2011 Jul 27.


Isolation and characterization of Psalmopeotoxin I and II: two novel antimalarial peptides from the venom of the tarantula Psalmopoeus cambridgei.

Choi SJ, Parent R, Guillaume C, Deregnaucourt C, Delarbre C, Ojcius DM, Montagne JJ, Célérier ML, Phelipot A, Amiche M, Molgo J, Camadro JM, Guette C.

FEBS Lett. 2004 Aug 13;572(1-3):109-17.


In Silico screening on the three-dimensional model of the Plasmodium vivax SUB1 protease leads to the validation of a novel anti-parasite compound.

Bouillon A, Giganti D, Benedet C, Gorgette O, Pêtres S, Crublet E, Girard-Blanc C, Witkowski B, Ménard D, Nilges M, Mercereau-Puijalon O, Stoven V, Barale JC.

J Biol Chem. 2013 Jun 21;288(25):18561-73. doi: 10.1074/jbc.M113.456764. Epub 2013 May 7.


Solution structure of PcFK1, a spider peptide active against Plasmodium falciparum.

Pimentel C, Choi SJ, Chagot B, Guette C, Camadro JM, Darbon H.

Protein Sci. 2006 Mar;15(3):628-34. Epub 2006 Feb 1.


Proteolytic activity of Plasmodium falciparum subtilisin-like protease 3 on parasite profilin, a multifunctional protein.

Alam A, Bhatnagar RK, Relan U, Mukherjee P, Chauhan VS.

Mol Biochem Parasitol. 2013 Oct;191(2):58-62. doi: 10.1016/j.molbiopara.2013.09.006. Epub 2013 Sep 27.


Determination with matrix-assisted laser desorption/ionization tandem time-of-flight mass spectrometry of the extensive disulfide bonding in tarantula venom peptide Psalmopeotoxin I.

Combes A, Choi SJ, Pimentel C, Darbon H, Waidelich D, Mestivier D, Camadro JM.

Eur J Mass Spectrom (Chichester). 2009;15(4):517-29. doi: 10.1255/ejms.1000.


A multifunctional serine protease primes the malaria parasite for red blood cell invasion.

Koussis K, Withers-Martinez C, Yeoh S, Child M, Hackett F, Knuepfer E, Juliano L, Woehlbier U, Bujard H, Blackman MJ.

EMBO J. 2009 Mar 18;28(6):725-35. doi: 10.1038/emboj.2009.22. Epub 2009 Feb 12.


Characterization of Plasmodium falciparum integral membrane protein Pf25-IMP and identification of its red blood cell binding sequences inhibiting merozoite invasion in vitro.

Curtidor H, Arévalo G, Vanegas M, Vizcaíno C, Patarroyo MA, Forero M, Patarroyo ME.

Protein Sci. 2008 Sep;17(9):1494-504. doi: 10.1110/ps.036251.108. Epub 2008 Jun 12.


Molecular determinants of binding to the Plasmodium subtilisin-like protease 1.

Fulle S, Withers-Martinez C, Blackman MJ, Morris GM, Finn PW.

J Chem Inf Model. 2013 Mar 25;53(3):573-83. doi: 10.1021/ci300581z. Epub 2013 Mar 4.


Plasmodium subtilisin-like protease 1 (SUB1): insights into the active-site structure, specificity and function of a pan-malaria drug target.

Withers-Martinez C, Suarez C, Fulle S, Kher S, Penzo M, Ebejer JP, Koussis K, Hackett F, Jirgensons A, Finn P, Blackman MJ.

Int J Parasitol. 2012 May 15;42(6):597-612. doi: 10.1016/j.ijpara.2012.04.005. Epub 2012 Apr 27.


Quinolylhydrazones as novel inhibitors of Plasmodium falciparum serine protease PfSUB1.

Gemma S, Giovani S, Brindisi M, Tripaldi P, Brogi S, Savini L, Fiorini I, Novellino E, Butini S, Campiani G, Penzo M, Blackman MJ.

Bioorg Med Chem Lett. 2012 Aug 15;22(16):5317-21. doi: 10.1016/j.bmcl.2012.06.023. Epub 2012 Jun 23.


In silico study of subtilisin-like protease 1 (SUB1) from different Plasmodium species in complex with peptidyl-difluorostatones and characterization of potent pan-SUB1 inhibitors.

Brogi S, Giovani S, Brindisi M, Gemma S, Novellino E, Campiani G, Blackman MJ, Butini S.

J Mol Graph Model. 2016 Mar;64:121-130. doi: 10.1016/j.jmgm.2016.01.005. Epub 2016 Jan 19.


Conserved regions from Plasmodium falciparum MSP11 specifically interact with host cells and have a potential role during merozoite invasion of red blood cells.

Obando-Martinez AZ, Curtidor H, Vanegas M, Arévalo-Pinzón G, Patarroyo MA, Patarroyo ME.

J Cell Biochem. 2010 Jul 1;110(4):882-92. doi: 10.1002/jcb.22600.


Characterization of Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1) and its role in microneme secretion during erythrocyte invasion.

Bansal A, Singh S, More KR, Hans D, Nangalia K, Yogavel M, Sharma A, Chitnis CE.

J Biol Chem. 2013 Jan 18;288(3):1590-602. doi: 10.1074/jbc.M112.411934. Epub 2012 Nov 30. Erratum in: J Biol Chem. 2013 Jul 5;288(27):19643.


The malaria parasite egress protease SUB1 is a calcium-dependent redox switch subtilisin.

Withers-Martinez C, Strath M, Hackett F, Haire LF, Howell SA, Walker PA, Christodoulou E, Dodson GG, Blackman MJ.

Nat Commun. 2014 May 2;5:3726. doi: 10.1038/ncomms4726. Erratum in: Nat Commun. 2014;5:4031. Evangelos, Christodoulou [corrected to Christodoulou, Evangelos].


Rational design of the first difluorostatone-based PfSUB1 inhibitors.

Giovani S, Penzo M, Brogi S, Brindisi M, Gemma S, Novellino E, Savini L, Blackman MJ, Campiani G, Butini S.

Bioorg Med Chem Lett. 2014 Aug 1;24(15):3582-6. doi: 10.1016/j.bmcl.2014.05.044. Epub 2014 May 23.


Identification of peptides with high red blood cell and hepatocyte binding activity in the Plasmodium falciparum multi-stage invasion proteins: PfSPATR and MCP-1.

Curtidor H, García J, Vanegas M, Puentes F, Forero M, Patarroyo ME.

Biochimie. 2008 Nov-Dec;90(11-12):1750-9. doi: 10.1016/j.biochi.2008.08.003. Epub 2008 Sep 13.


Merozoite surface protein 8 of Plasmodium falciparum contains two epidermal growth factor-like domains.

Black CG, Wu T, Wang L, Hibbs AR, Coppel RL.

Mol Biochem Parasitol. 2001 May;114(2):217-26.


Plasmodium falciparum encodes a conserved active inhibitor-2 for Protein Phosphatase type 1: perspectives for novel anti-plasmodial therapy.

Fréville A, Cailliau-Maggio K, Pierrot C, Tellier G, Kalamou H, Lafitte S, Martoriati A, Pierce RJ, Bodart JF, Khalife J.

BMC Biol. 2013 Jul 9;11:80. doi: 10.1186/1741-7007-11-80.


Synthesis, biophysical, and biological studies of wild-type and mutant psalmopeotoxins--anti-malarial cysteine knot peptides from Psalmopoeus cambridgei.

Kamolkijkarn P, Prasertdee T, Netirojjanakul C, Sarnpitak P, Ruchirawat S, Deechongkit S.

Peptides. 2010 Apr;31(4):533-40. doi: 10.1016/j.peptides.2010.01.001. Epub 2010 Jan 11.


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