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Items: 1 to 20 of 199

1.

Synthesis and biological evaluation of (±)-3-(2-(2-fluorobenzyloxy) naphthalen-6-yl)-2-aminopropanoic acid derivatives as novel PTP1B inhibitors.

Sun LP, Shen Q, Piao HH, Ma WP, Gao LX, Zhang W, Nan FJ, Li J, Piao HR.

Eur J Med Chem. 2011 Sep;46(9):3630-8. doi: 10.1016/j.ejmech.2011.05.027. Epub 2011 May 20.

PMID:
21680062
2.

Synthesis and biological evaluation of 2,4,6-trihydroxychalcone derivatives as novel protein tyrosine phosphatase 1B inhibitors.

Sun LP, Gao LX, Ma WP, Nan FJ, Li J, Piao HR.

Chem Biol Drug Des. 2012 Oct;80(4):584-90. doi: 10.1111/j.1747-0285.2012.01431.x. Epub 2012 Jul 13.

PMID:
22805439
3.

Synthesis and biological evaluation of heterocyclic ring-substituted maslinic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B.

Qiu WW, Shen Q, Yang F, Wang B, Zou H, Li JY, Li J, Tang J.

Bioorg Med Chem Lett. 2009 Dec 1;19(23):6618-22. doi: 10.1016/j.bmcl.2009.10.017. Epub 2009 Oct 8.

PMID:
19846303
4.

Synthesis and biological evaluation of novel bis-aromatic amides as novel PTP1B inhibitors.

Wang WL, Huang C, Gao LX, Tang CL, Wang JQ, Wu MC, Sheng L, Chen HJ, Nan FJ, Li JY, Li J, Feng B.

Bioorg Med Chem Lett. 2014 Apr 15;24(8):1889-94. doi: 10.1016/j.bmcl.2014.03.015. Epub 2014 Mar 15.

PMID:
24684845
5.

[Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].

Du X, Zhang SE, Liu JZ, Nie FL, Ye F, Tian JY, Xiao ZY.

Yao Xue Xue Bao. 2012 Mar;47(3):367-73. Chinese.

PMID:
22645761
6.

Novel thiophene derivatives as PTP1B inhibitors with selectivity and cellular activity.

Ye D, Zhang Y, Wang F, Zheng M, Zhang X, Luo X, Shen X, Jiang H, Liu H.

Bioorg Med Chem. 2010 Mar 1;18(5):1773-82. doi: 10.1016/j.bmc.2010.01.055. Epub 2010 Jan 28.

PMID:
20153651
7.

Design, synthesis, and biological evaluation of bromophenol derivatives as protein tyrosine phosphatase 1B inhibitors.

Jiang B, Shi D, Cui Y, Guo S.

Arch Pharm (Weinheim). 2012 Jun;345(6):444-53. doi: 10.1002/ardp.201100373. Epub 2012 Feb 3.

PMID:
22307562
8.

PTP1B inhibitors: synthesis and evaluation of difluoro-methylenephosphonate bioisosteres on a sulfonamide scaffold.

Holmes CP, Li X, Pan Y, Xu C, Bhandari A, Moody CM, Miguel JA, Ferla SW, De Francisco MN, Frederick BT, Zhou S, Macher N, Jang L, Irvine JD, Grove JR.

Bioorg Med Chem Lett. 2008 Apr 15;18(8):2719-24. doi: 10.1016/j.bmcl.2008.03.007. Epub 2008 Mar 6.

PMID:
18372175
9.

Synthesis of (glycopyranosyl-triazolyl)-purines and their inhibitory activities against protein tyrosine phosphatase 1B (PTP1B).

Luo L, He XP, Shen Q, Li JY, Shi XX, Xie J, Li J, Chen GR.

Chem Biodivers. 2011 Nov;8(11):2035-44. doi: 10.1002/cbdv.201000242.

PMID:
22083916
10.

Discovery of potent, selective and orally bioavailable triaryl-sulfonamide based PTP1B inhibitors.

Patel D, Jain M, Shah SR, Bahekar R, Jadav P, Joharapurkar A, Dhanesha N, Shaikh M, Sairam KV, Kapadnis P.

Bioorg Med Chem Lett. 2012 Jan 15;22(2):1111-7. doi: 10.1016/j.bmcl.2011.11.122. Epub 2011 Dec 6.

PMID:
22189136
11.

Preparation of triazole-linked glycosylated α-ketocarboxylic acid derivatives as new PTP1B inhibitors.

Song Z, He XP, Li C, Gao LX, Wang ZX, Tang Y, Xie J, Li J, Chen GR.

Carbohydr Res. 2011 Jan 3;346(1):140-5. doi: 10.1016/j.carres.2010.10.023. Epub 2010 Oct 30.

PMID:
21111404
12.

Synthesis and biological evaluation of 4,4-dimethyl lithocholic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B.

He HB, Gao LX, Deng QF, Ma WP, Tang CL, Qiu WW, Tang J, Li JY, Li J, Yang F.

Bioorg Med Chem Lett. 2012 Dec 1;22(23):7237-42. doi: 10.1016/j.bmcl.2012.09.040. Epub 2012 Sep 21.

PMID:
23067554
13.

Bromophenols as inhibitors of protein tyrosine phosphatase 1B with antidiabetic properties.

Shi D, Li J, Jiang B, Guo S, Su H, Wang T.

Bioorg Med Chem Lett. 2012 Apr 15;22(8):2827-32. doi: 10.1016/j.bmcl.2012.02.074. Epub 2012 Mar 2.

PMID:
22444684
14.

Peptidomimetics as potent and selective PTP1B inhibitors.

Patel D, Jain M, Shah SR, Bahekar R, Jadav P, Shah K, Joharapurkar A, Shaikh M, Sairam KV.

Med Chem. 2013 Aug;9(5):660-71.

PMID:
23030658
15.

Design, Synthesis and Biological Evaluation of Stilbene Derivatives as Novel Inhibitors of Protein Tyrosine Phosphatase 1B.

He H, Ge Y, Dai H, Cui S, Ye F, Jin J, Shi Y.

Molecules. 2016 Dec 16;21(12). pii: E1722. doi: 10.3390/molecules21121722.

16.

Design, synthesis and insulin-sensitising effects of novel PTP1B inhibitors.

Tang YB, Lu D, Chen Z, Hu C, Yang Y, Tian JY, Ye F, Wu L, Zhang ZY, Xiao Z.

Bioorg Med Chem Lett. 2013 Apr 15;23(8):2313-8. doi: 10.1016/j.bmcl.2013.02.073. Epub 2013 Feb 26.

PMID:
23499238
17.

Design, synthesis, and biological evaluation of 2-substituted ethenesulfonic acid ester derivatives as selective PTP1B inhibitors.

Liu J, Deng X, Jin Y, Xu B, Liu W, Jiang F, Fu L.

Pharmazie. 2015 Jul;70(7):446-51.

PMID:
26373204
18.

Dinuclear copper complexes of organic claw: potent inhibition of protein tyrosine phosphatases.

Ma L, Lu L, Zhu M, Wang Q, Gao F, Yuan C, Wu Y, Xing S, Fu X, Mei Y, Gao X.

J Inorg Biochem. 2011 Sep;105(9):1138-47. doi: 10.1016/j.jinorgbio.2011.05.015. Epub 2011 May 27.

PMID:
21708098
19.

Chemical constituents from Sambucus adnata and their protein-tyrosine phosphatase 1B inhibitory activities.

Sasaki T, Li W, Morimura H, Li S, Li Q, Asada Y, Koike K.

Chem Pharm Bull (Tokyo). 2011;59(11):1396-9.

20.

Potent inhibition of protein tyrosine phosphatases by copper complexes with multi-benzimidazole derivatives.

Li Y, Lu L, Zhu M, Wang Q, Yuan C, Xing S, Fu X, Mei Y.

Biometals. 2011 Dec;24(6):993-1004. doi: 10.1007/s10534-011-9460-3. Epub 2011 May 27.

PMID:
21618062

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