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Items: 1 to 20 of 57

1.

Fully automated synthesis and initial PET evaluation of [11C]PBR28.

Wang M, Yoder KK, Gao M, Mock BH, Xu XM, Saykin AJ, Hutchins GD, Zheng QH.

Bioorg Med Chem Lett. 2009 Oct 1;19(19):5636-9. doi: 10.1016/j.bmcl.2009.08.051. Epub 2009 Aug 15.

2.

Synthesis and evaluation in monkey of two sensitive 11C-labeled aryloxyanilide ligands for imaging brain peripheral benzodiazepine receptors in vivo.

Briard E, Zoghbi SS, Imaizumi M, Gourley JP, Shetty HU, Hong J, Cropley V, Fujita M, Innis RB, Pike VW.

J Med Chem. 2008 Jan 10;51(1):17-30. Epub 2007 Dec 8.

PMID:
18067245
3.

Novel Pyrazolo[1,5-a]pyrimidines as Translocator Protein 18 kDa (TSPO) Ligands: Synthesis, in Vitro Biological Evaluation, [(18)F]-Labeling, and in Vivo Neuroinflammation PET Images.

Damont A, Médran-Navarrete V, Cacheux F, Kuhnast B, Pottier G, Bernards N, Marguet F, Puech F, Boisgard R, Dollé F.

J Med Chem. 2015 Sep 24;58(18):7449-64. doi: 10.1021/acs.jmedchem.5b00932. Epub 2015 Sep 3.

PMID:
26280386
4.

Positron Emission Tomography studies with [11C]PBR28 in the Healthy Rodent Brain: Validating SUV as an Outcome Measure of Neuroinflammation.

Tóth M, Doorduin J, Häggkvist J, Varrone A, Amini N, Halldin C, Gulyás B.

PLoS One. 2015 May 21;10(5):e0125917. doi: 10.1371/journal.pone.0125917. eCollection 2015.

5.

Evaluation of N-benzyl-N-[11C]methyl-2- (7-methyl-8-oxo-2-phenyl-7,8-dihydro-9H-purin-9-yl)acetamide ([11C]DAC) as a novel translocator protein (18 kDa) radioligand in kainic acid-lesioned rat.

Yanamoto K, Yamasaki T, Kumata K, Yui J, Odawara C, Kawamura K, Hatori A, Inoue O, Yamaguchi M, Suzuki K, Zhang MR.

Synapse. 2009 Nov;63(11):961-71. doi: 10.1002/syn.20678.

PMID:
19593823
6.

Synthesis of 6-[¹⁸F]fluoro-PBR28, a novel radiotracer for imaging the TSPO 18 kDa with PET.

Damont A, Boisgard R, Kuhnast B, Lemée F, Raggiri G, Scarf AM, Da Pozzo E, Selleri S, Martini C, Tavitian B, Kassiou M, Dollé F.

Bioorg Med Chem Lett. 2011 Aug 15;21(16):4819-22. doi: 10.1016/j.bmcl.2011.06.048. Epub 2011 Jun 17.

PMID:
21741237
7.

Evaluation of the PBR/TSPO radioligand [(18)F]DPA-714 in a rat model of focal cerebral ischemia.

Martín A, Boisgard R, Thézé B, Van Camp N, Kuhnast B, Damont A, Kassiou M, Dollé F, Tavitian B.

J Cereb Blood Flow Metab. 2010 Jan;30(1):230-41. doi: 10.1038/jcbfm.2009.205. Epub 2009 Sep 30.

8.

Improved synthesis of the peripheral benzodiazepine receptor ligand [11C]DPA-713 using [11C]methyl triflate.

Thominiaux C, Dollé F, James ML, Bramoullé Y, Boutin H, Besret L, Grégoire MC, Valette H, Bottlaender M, Tavitian B, Hantraye P, Selleri S, Kassiou M.

Appl Radiat Isot. 2006 May;64(5):570-3. Epub 2006 Jan 20.

PMID:
16427784
9.

Development of N-[4-[6-(isopropylamino)pyrimidin-4-yl]-1,3-thiazol-2-yl]-N-methyl-4-[11C]methylbenzamide for positron emission tomography imaging of metabotropic glutamate 1 receptor in monkey brain.

Fujinaga M, Yamasaki T, Maeda J, Yui J, Xie L, Nagai Y, Nengaki N, Hatori A, Kumata K, Kawamura K, Zhang MR.

J Med Chem. 2012 Dec 27;55(24):11042-51. doi: 10.1021/jm301597s. Epub 2012 Dec 10.

PMID:
23194448
10.

Acute neuroinflammation in a clinically relevant focal cortical ischemic stroke model in rat: longitudinal positron emission tomography and immunofluorescent tracking.

Tóth M, Little P, Arnberg F, Häggkvist J, Mulder J, Halldin C, Gulyás B, Holmin S.

Brain Struct Funct. 2016 Apr;221(3):1279-90. doi: 10.1007/s00429-014-0970-y. Epub 2015 Jan 20.

PMID:
25601153
11.

Brain and whole-body imaging in nonhuman primates of [11C]PBR28, a promising PET radioligand for peripheral benzodiazepine receptors.

Imaizumi M, Briard E, Zoghbi SS, Gourley JP, Hong J, Fujimura Y, Pike VW, Innis RB, Fujita M.

Neuroimage. 2008 Feb 1;39(3):1289-98. Epub 2007 Oct 12.

12.

Mixed-affinity binding in humans with 18-kDa translocator protein ligands.

Owen DR, Gunn RN, Rabiner EA, Bennacef I, Fujita M, Kreisl WC, Innis RB, Pike VW, Reynolds R, Matthews PM, Parker CA.

J Nucl Med. 2011 Jan;52(1):24-32. doi: 10.2967/jnumed.110.079459. Epub 2010 Dec 13.

13.

In vivo imaging and quantitative analysis of TSPO in rat peripheral tissues using small-animal PET with [18F]FEDAC.

Yanamoto K, Kumata K, Fujinaga M, Nengaki N, Takei M, Wakizaka H, Hosoi R, Momosaki S, Yamasaki T, Yui J, Kawamura K, Hatori A, Inoue O, Zhang MR.

Nucl Med Biol. 2010 Oct;37(7):853-60. doi: 10.1016/j.nucmedbio.2010.04.183.

PMID:
20870161
14.

PET imaging of lung inflammation with [18F]FEDAC, a radioligand for translocator protein (18 kDa).

Hatori A, Yui J, Yamasaki T, Xie L, Kumata K, Fujinaga M, Yoshida Y, Ogawa M, Nengaki N, Kawamura K, Fukumura T, Zhang MR.

PLoS One. 2012;7(9):e45065. doi: 10.1371/journal.pone.0045065. Epub 2012 Sep 12.

16.

Synthesis of fluorine substituted pyrazolopyrimidines as potential leads for the development of PET-imaging agents for the GABAA receptors.

Hoepping A, Diekers M, Deuther-Conrad W, Scheunemann M, Fischer S, Hiller A, Wegner F, Steinbach J, Brust P.

Bioorg Med Chem. 2008 Feb 1;16(3):1184-94. Epub 2007 Nov 26.

PMID:
18023192
17.

Fully automated radiosynthesis of [¹¹C]PBR28, a radiopharmaceutical for the translocator protein (TSPO) 18 kDa, using a GE TRACERlab FXC-Pro.

Hoareau R, Shao X, Henderson BD, Scott PJ.

Appl Radiat Isot. 2012 Aug;70(8):1779-83. doi: 10.1016/j.apradiso.2012.03.006. Epub 2012 Mar 29.

PMID:
22503515
18.

Synthesis and evaluation of novel carbon-11 labeled oxopurine analogues for positron emission tomography imaging of translocator protein (18 kDa) in peripheral organs.

Kumata K, Yui J, Hatori A, Fujinaga M, Yanamoto K, Yamasaki T, Kawamura K, Wakizaka H, Nengaki N, Yoshida Y, Ogawa M, Fukumura T, Zhang MR.

J Med Chem. 2011 Sep 8;54(17):6040-9. doi: 10.1021/jm200516a. Epub 2011 Aug 4.

PMID:
21790126
19.

PET radioligands targeting the brain GABAA /benzodiazepine receptor complex.

Andersson JD, Halldin C.

J Labelled Comp Radiopharm. 2013 Mar-Apr;56(3-4):196-206. doi: 10.1002/jlcr.3008. Review.

PMID:
24285326
20.

Development of Fluorinated Non-Peptidic Ghrelin Receptor Ligands for Potential Use in Molecular Imaging.

Moldovan RP, Els-Heindl S, Worm DJ, Kniess T, Kluge M, Beck-Sickinger AG, Deuther-Conrad W, Krügel U, Brust P.

Int J Mol Sci. 2017 Apr 5;18(4). pii: E768. doi: 10.3390/ijms18040768.

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