Similar articles for PMID: 18068982

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1

Design and synthesis of novel potent and selective integrin alphanubeta3 antagonists--novel synthetic routes to isoquinolinone, benzoxazinone, and quinazolinone acetates.

Seitz W, Geneste H, Backfisch G, Delzer J, Graef C, Hornberger W, Kling A, Subkowski T, Zimmermann N. Seitz W, et al. Bioorg Med Chem Lett. 2008 Jan 15;18(2):527-31. doi: 10.1016/j.bmcl.2007.11.089. Epub 2007 Nov 28. Bioorg Med Chem Lett. 2008. PMID: 18068982

2

Identification of novel short chain 4-substituted indoles as potent alphavbeta3 antagonist using structure-based drug design.

Raboisson P, Desjarlais RL, Reed R, Lattanze J, Chaikin M, Manthey CL, Tomczuk BE, Marugán JJ. Raboisson P, et al. Eur J Med Chem. 2007 Mar;42(3):334-43. doi: 10.1016/j.ejmech.2006.10.015. Epub 2006 Dec 20. Eur J Med Chem. 2007. PMID: 17184884

3

Synthesis and initial evaluation of novel, non-peptidic antagonists of the alpha(v)-integrins alpha(v)beta(3) and alpha(v)beta(5).

Letourneau JJ, Liu J, Ohlmeyer MH, Riviello C, Rong Y, Li H, Appell KC, Bansal S, Jacob B, Wong A, Webb ML. Letourneau JJ, et al. Bioorg Med Chem Lett. 2009 Jan 15;19(2):352-5. doi: 10.1016/j.bmcl.2008.11.074. Epub 2008 Nov 24. Bioorg Med Chem Lett. 2009. PMID: 19081719

4

Novel potent and selective alphavbeta3/alphavbeta5 integrin dual antagonists with reduced binding affinity for human serum albumin.

Raboisson P, Manthey CL, Chaikin M, Lattanze J, Crysler C, Leonard K, Pan W, Tomczuk BE, Marugán JJ. Raboisson P, et al. Eur J Med Chem. 2006 Jul;41(7):847-61. doi: 10.1016/j.ejmech.2006.03.008. Epub 2006 May 11. Eur J Med Chem. 2006. PMID: 16697080

5

A novel class of sodium/calcium exchanger inhibitors: design, synthesis, and structure-activity relationships of 4-phenyl-3-(piperidin-4-yl)-3,4-dihydro-2(1H)-quinazolinone derivatives.

Hasegawa H, Muraoka M, Matsui K, Kojima A. Hasegawa H, et al. Bioorg Med Chem Lett. 2006 Feb;16(3):727-30. doi: 10.1016/j.bmcl.2005.10.012. Epub 2005 Oct 24. Bioorg Med Chem Lett. 2006. PMID: 16249082

6

A novel class of sodium/calcium exchanger inhibitor: design, synthesis, and structure-activity relationships of 3,4-dihydro-2(1H)-quinazolinone derivatives.

Hasegawa H, Muraoka M, Ohmori M, Matsui K, Kojima A. Hasegawa H, et al. Bioorg Med Chem. 2005 Jun 1;13(11):3721-35. doi: 10.1016/j.bmc.2005.03.019. Bioorg Med Chem. 2005. PMID: 15863001

7

Tricyclic pharmacophore-based molecules as novel integrin alpha(v)beta3 antagonists. Part 1: design and synthesis of a lead compound exhibiting alpha(v)beta3/alpha(IIb)beta3 dual antagonistic activity.

Kubota D, Ishikawa M, Yamamoto M, Murakami S, Hachisu M, Katano K, Ajito K. Kubota D, et al. Bioorg Med Chem. 2006 Apr 1;14(7):2089-108. doi: 10.1016/j.bmc.2005.10.060. Epub 2005 Nov 23. Bioorg Med Chem. 2006. PMID: 16309911

8

Design, synthesis, and biological evaluation of novel potent and selective alphavbeta3/alphavbeta5 integrin dual inhibitors with improved bioavailability. Selection of the molecular core.

Marugán JJ, Manthey C, Anaclerio B, Lafrance L, Lu T, Markotan T, Leonard KA, Crysler C, Eisennagel S, Dasgupta M, Tomczuk B. Marugán JJ, et al. J Med Chem. 2005 Feb 24;48(4):926-34. doi: 10.1021/jm049725u. J Med Chem. 2005. PMID: 15715463

9

Discovery of piperidine carboxamide TRPV1 antagonists.

Cheung WS, Calvo RR, Tounge BA, Zhang SP, Stone DR, Brandt MR, Hutchinson T, Flores CM, Player MR. Cheung WS, et al. Bioorg Med Chem Lett. 2008 Aug 15;18(16):4569-72. doi: 10.1016/j.bmcl.2008.07.035. Epub 2008 Jul 15. Bioorg Med Chem Lett. 2008. PMID: 18662879

10

Tricyclic pharmacophore-based molecules as novel integrin alphavbeta3 antagonists. Part IV: preliminary control of alphavbeta3 selectivity by meta-oriented substitution.

Kubota D, Ishikawa M, Ishikawa M, Yahata N, Murakami S, Fujishima K, Kitakaze M, Ajito K. Kubota D, et al. Bioorg Med Chem. 2006 Jun 15;14(12):4158-81. doi: 10.1016/j.bmc.2006.01.062. Epub 2006 Feb 28. Bioorg Med Chem. 2006. PMID: 16504518

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