Similar articles for PMID: 17960925

Year	Number of Results
1954	2
1972	1
1975	1
1976	2
1977	2
1979	1
1980	1
1982	1
1983	2
1984	1
1985	1
1987	2
1988	1
1989	2
1991	3
1992	1
1993	2
1994	1
1995	2
1998	4
1999	2
2000	1
2001	3
2002	2
2003	8
2004	15
2005	35
2006	46
2007	46
2008	37
2009	25
2010	14
2011	9
2012	8
2013	13
2014	13
2015	6
2016	4
2017	5
2018	2
2019	2
2020	1
2021	3
2022	3
2023	2
2024	0

1

Identification of phosphinate dipeptide analog inhibitors directed against the Plasmodium falciparum M17 leucine aminopeptidase as lead antimalarial compounds.

Skinner-Adams TS, Lowther J, Teuscher F, Stack CM, Grembecka J, Mucha A, Kafarski P, Trenholme KR, Dalton JP, Gardiner DL. Skinner-Adams TS, et al. J Med Chem. 2007 Nov 29;50(24):6024-31. doi: 10.1021/jm070733v. Epub 2007 Oct 26. J Med Chem. 2007. PMID: 17960925

2

The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity.

Grembecka J, Mucha A, Cierpicki T, Kafarski P. Grembecka J, et al. J Med Chem. 2003 Jun 19;46(13):2641-55. doi: 10.1021/jm030795v. J Med Chem. 2003. PMID: 12801228

3

The M17 leucine aminopeptidase of the malaria parasite Plasmodium falciparum: importance of active site metal ions in the binding of substrates and inhibitors.

Maric S, Donnelly SM, Robinson MW, Skinner-Adams T, Trenholme KR, Gardiner DL, Dalton JP, Stack CM, Lowther J. Maric S, et al. Biochemistry. 2009 Jun 16;48(23):5435-9. doi: 10.1021/bi9003638. Biochemistry. 2009. PMID: 19408962

4

KBE009: An antimalarial bestatin-like inhibitor of the Plasmodium falciparum M1 aminopeptidase discovered in an Ugi multicomponent reaction-derived peptidomimetic library.

González-Bacerio J, Maluf SEC, Méndez Y, Pascual I, Florent I, Melo PMS, Budu A, Ferreira JC, Moreno E, Carmona AK, Rivera DG, Alonso Del Rivero M, Gazarini ML. González-Bacerio J, et al. Bioorg Med Chem. 2017 Sep 1;25(17):4628-4636. doi: 10.1016/j.bmc.2017.06.047. Epub 2017 Jul 4. Bioorg Med Chem. 2017. PMID: 28728898

5

Plasmodium chabaudi chabaudi and P. falciparum: inhibition of aminopeptidase and parasite growth by bestatin and nitrobestatin.

Nankya-Kitaka MF, Curley GP, Gavigan CS, Bell A, Dalton JP. Nankya-Kitaka MF, et al. Parasitol Res. 1998 Jul;84(7):552-8. doi: 10.1007/s004360050447. Parasitol Res. 1998. PMID: 9694371

6

Characterization of the Plasmodium falciparum M17 leucyl aminopeptidase. A protease involved in amino acid regulation with potential for antimalarial drug development.

Stack CM, Lowther J, Cunningham E, Donnelly S, Gardiner DL, Trenholme KR, Skinner-Adams TS, Teuscher F, Grembecka J, Mucha A, Kafarski P, Lua L, Bell A, Dalton JP. Stack CM, et al. J Biol Chem. 2007 Jan 19;282(3):2069-80. doi: 10.1074/jbc.M609251200. Epub 2006 Nov 15. J Biol Chem. 2007. PMID: 17107951 Free article.

7

M17 leucine aminopeptidase of the human malaria parasite Plasmodium vivax.

Lee JY, Song SM, Seok JW, Jha BK, Han ET, Song HO, Yu HS, Hong Y, Kong HH, Chung DI. Lee JY, et al. Mol Biochem Parasitol. 2010 Mar;170(1):45-8. doi: 10.1016/j.molbiopara.2009.11.003. Epub 2009 Nov 18. Mol Biochem Parasitol. 2010. PMID: 19931315

8

A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases.

Vassiliou S, Xeilari M, Yiotakis A, Grembecka J, Pawełczak M, Kafarski P, Mucha A. Vassiliou S, et al. Bioorg Med Chem. 2007 May 1;15(9):3187-200. doi: 10.1016/j.bmc.2007.02.042. Epub 2007 Feb 22. Bioorg Med Chem. 2007. PMID: 17337192

9

Inhibitors of Plasmodium falciparum methionine aminopeptidase 1b possess antimalarial activity.

Chen X, Chong CR, Shi L, Yoshimoto T, Sullivan DJ Jr, Liu JO. Chen X, et al. Proc Natl Acad Sci U S A. 2006 Sep 26;103(39):14548-53. doi: 10.1073/pnas.0604101103. Epub 2006 Sep 18. Proc Natl Acad Sci U S A. 2006. PMID: 16983082 Free PMC article.

10

High antiplasmodial activity of novel plasmepsins I and II inhibitors.

Dell'Agli M, Parapini S, Galli G, Vaiana N, Taramelli D, Sparatore A, Liu P, Dunn BM, Bosisio E, Romeo S. Dell'Agli M, et al. J Med Chem. 2006 Dec 14;49(25):7440-9. doi: 10.1021/jm061033d. J Med Chem. 2006. PMID: 17149873 Free article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

304 results

Results by year