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Items: 1 to 20 of 107

1.

Derivatives of 3-sec-butyl-1-oxo-2,3-dihydroisoquinoline as inhibitors of mu-calpain.

Chicharro R, Alonso M, Mazo MT, Arán VJ, Herradón B.

ChemMedChem. 2006 Jul;1(7):710-4. No abstract available.

PMID:
16902923
2.

Design and synthesis of 4-aryl-4-oxobutanoic acid amides as calpain inhibitors.

Zhang Y, Jung SY, Jin C, Kim ND, Gong P, Lee YS.

Bioorg Med Chem Lett. 2009 Jan 15;19(2):502-7. doi: 10.1016/j.bmcl.2008.11.030. Epub 2008 Nov 14.

PMID:
19041242
3.

Exploration of peptidyl hydrazones as water-soluble calpain inhibitors.

Nakamura M, Inoue J.

Bioorg Med Chem Lett. 2002 Jun 17;12(12):1603-6.

PMID:
12039572
4.

A novel series of urea-based peptidomimetic calpain inhibitors.

Sanders ML, Donkor IO.

Bioorg Med Chem Lett. 2006 Apr 1;16(7):1965-8. Epub 2006 Jan 18.

PMID:
16412635
5.

Syntheses and SH-enzyme inhibitory activities of new epoxysuccinic acid piperazine derivatives against mu-calpain and cathepsin B.

Inoue J, Yoshida Y, Nakamura M, Cui YS, Nagao Y.

Drug Des Discov. 1999 Aug;16(2):165-9.

PMID:
10533812
6.

Exploration of the importance of the P2-P3-NHCO-moiety in a potent di- or tripeptide inhibitor of calpain I: insights into the development of nonpeptidic inhibitors of calpain I.

Chatterjee S, Iqbal M, Mallya S, Senadhi SE, O'Kane TM, McKenna BA, Bozyczko-Coyne D, Kauer JC, Siman R, Mallamo JP.

Bioorg Med Chem. 1998 May;6(5):509-22.

PMID:
9629465
7.

Synthesis and biological evaluation of chromone carboxamides as calpain inhibitors.

Lee KS, Seo SH, Lee YH, Kim HD, Son MH, Chung BY, Lee JY, Jin C, Lee YS.

Bioorg Med Chem Lett. 2005 Jun 2;15(11):2857-60. Epub 2005 Apr 25.

PMID:
15911268
8.

Molecular modeling, synthesis, and biological evaluation of macrocyclic calpain inhibitors.

Abell AD, Jones MA, Coxon JM, Morton JD, Aitken SG, McNabb SB, Lee HY, Mehrtens JM, Alexander NA, Stuart BG, Neffe AT, Bickerstaffe R.

Angew Chem Int Ed Engl. 2009;48(8):1455-8. doi: 10.1002/anie.200805014.

PMID:
19145612
10.

P2-proline-derived inhibitors of calpain I.

Tripathy R, Gu ZQ, Dunn D, Senadhi SE, Ator MA, Chatterjee S.

Bioorg Med Chem Lett. 1998 Oct 6;8(19):2647-52.

PMID:
9873596
11.

Design and synthesis of calpain inhibitory 6-pyridone 2-carboxamide derivatives.

Lee KY, Lee KS, Jin C, Lee YS.

Eur J Med Chem. 2009 Mar;44(3):1331-4. doi: 10.1016/j.ejmech.2008.02.023. Epub 2008 Mar 7.

PMID:
18396356
12.

Synthesis of a reported calpain inhibitor isolated from Streptomyces griseus.

Donkor IO, Sanders ML.

Bioorg Med Chem Lett. 2001 Oct 8;11(19):2647-9.

PMID:
11551769
13.

A survey of calpain inhibitors.

Donkor IO.

Curr Med Chem. 2000 Dec;7(12):1171-88. Review.

PMID:
11032966
14.

Synthesis of a small library of diketopiperazines as potential inhibitors of calpain.

Zeng Y, Li Q, Hanzlik RP, Aubé J.

Bioorg Med Chem Lett. 2005 Jun 15;15(12):3034-8.

PMID:
15896956
15.

A facile synthesis of emodin derivatives, emodin carbaldehyde, citreorosein, and their 10-deoxygenated derivatives and their inhibitory activities on μ-calpain.

Liang JL, Cha HC, Lee SH, Son JK, Chang HW, Eom JE, Kwon Y, Jahng Y.

Arch Pharm Res. 2012 Mar;35(3):447-54. doi: 10.1007/s12272-012-0307-4. Epub 2012 Apr 5.

PMID:
22477191
16.

Cell-penetrating inhibitors of calpain.

Mehdi S.

Trends Biochem Sci. 1991 Apr;16(4):150-3. Review.

PMID:
1877091
17.

Developments in the design and synthesis of calpain inhibitors.

Neffe AT, Abell AD.

Curr Opin Drug Discov Devel. 2005 Nov;8(6):684-700. Review.

PMID:
16312145
18.

Peptidyl aldehyde inhibitors of calpain incorporating P2-proline mimetics.

Donkor IO, Korukonda R, Huang TL, LeCour L Jr.

Bioorg Med Chem Lett. 2003 Mar 10;13(5):783-4.

PMID:
12617890
19.

Inhibition of human mu-calpain by conformationally constrained calpastatin peptides.

Pfizer J, Assfalg-Machleidt I, Machleidt W, Schaschke N.

Biol Chem. 2008 Jan;389(1):83-90.

PMID:
18095873
20.

Discovery of phenyl alanine derived ketoamides carrying benzoyl residues as novel calpain inhibitors.

Lubisch W, Möller A.

Bioorg Med Chem Lett. 2002 May 20;12(10):1335-8.

PMID:
11992771

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