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Items: 1 to 20 of 106

2.

Design, synthesis, and evaluation of cyclofenil derivatives for potential SPECT imaging agents.

Zhu H, Huang L, Zhang Y, Xu X, Sun Y, Shen YM.

J Biol Inorg Chem. 2010 May;15(4):591-9. doi: 10.1007/s00775-010-0627-0. Epub 2010 Mar 1.

PMID:
20195693
3.

Synthesis and biodistribution of fluorine-18-labeled fluorocyclofenils for imaging the estrogen receptor.

Seo JW, Chi DY, Dence CS, Welch MJ, Katzenellenbogen JA.

Nucl Med Biol. 2007 May;34(4):383-90. Epub 2007 Mar 30.

4.

Synthesis of new carbon-11 labeled cyclofenil derivatives for PET imaging of breast cancer estrogen receptors.

Gao M, Wang M, Mock BH, Miller KD, Sledge GW, Hutchins GD, Zheng QH.

Appl Radiat Isot. 2008 Apr;66(4):523-9. Epub 2007 Nov 19.

PMID:
18155914
5.

Synthesis and evaluation of aryl-substituted diarylpropionitriles, selective ligands for estrogen receptor beta, as positron-emission tomographic imaging agents.

Moon BS, Carlson KE, Katzenellenbogen JA, Choi TH, Chi DY, Kim JY, Cheon GJ, Koh HY, Lee KC, An G.

Bioorg Med Chem. 2009 May 1;17(9):3479-88. doi: 10.1016/j.bmc.2009.02.064. Epub 2009 Mar 9.

PMID:
19359182
6.

PET imaging of breast cancer with fluorine-18 radiolabeled estrogens and progestins.

Jonson SD, Welch MJ.

Q J Nucl Med. 1998 Mar;42(1):8-17. Review.

PMID:
9646640
7.

Characterization of the pharmacophore properties of novel selective estrogen receptor downregulators (SERDs).

Kieser KJ, Kim DW, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA.

J Med Chem. 2010 Apr 22;53(8):3320-9. doi: 10.1021/jm100047k.

8.

Imaging progesterone receptor in breast tumors: synthesis and receptor binding affinity of fluoroalkyl-substituted analogues of tanaproget.

Zhou HB, Lee JH, Mayne CG, Carlson KE, Katzenellenbogen JA.

J Med Chem. 2010 Apr 22;53(8):3349-60. doi: 10.1021/jm100052k.

9.

Estrogenic diazenes: heterocyclic non-steroidal estrogens of unusual structure with selectivity for estrogen receptor subtypes.

Ghosh U, Ganessunker D, Sattigeri VJ, Carlson KE, Mortensen DJ, Katzenellenbogen BS, Katzenellenbogen JA.

Bioorg Med Chem. 2003 Feb 20;11(4):629-57.

PMID:
12538029
10.

Studies on the ligand specificity and potential identity of microsomal antiestrogen-binding sites.

Watts CK, Sutherland RL.

Mol Pharmacol. 1987 May;31(5):541-51.

PMID:
3553893
11.

Aryl cyclopentadienyl tricarbonyl rhenium complexes: novel ligands for the estrogen receptor with potential use as estrogen radiopharmaceuticals.

Mull ES, Sattigeri VJ, Rodriguez AL, Katzenellenbogen JA.

Bioorg Med Chem. 2002 May;10(5):1381-98.

PMID:
11886802
12.
13.

Novel 7α-alkoxy-17α-(4'-halophenylethynyl)estradiols as potential SPECT/PET imaging agents for estrogen receptor expressing tumours: synthesis and binding affinity evaluation.

Neto C, Oliveira MC, Gano L, Marques F, Yasuda T, Thiemann T, Kniess T, Santos I.

Steroids. 2012 Sep;77(11):1123-32. doi: 10.1016/j.steroids.2012.05.004. Epub 2012 May 24.

PMID:
22633985
14.
15.

Design and synthesis of functionalized cyclopentadienyl tricarbonylmetal complexes for technetium-94m PET imaging of estrogen receptors.

Bigott HM, Parent E, Luyt LG, Katzenellenbogen JA, Welch MJ.

Bioconjug Chem. 2005 Mar-Apr;16(2):255-64.

PMID:
15769078
16.

Molecular mechanisms of estrogen action: selective ligands and receptor pharmacology.

Katzenellenbogen BS, Choi I, Delage-Mourroux R, Ediger TR, Martini PG, Montano M, Sun J, Weis K, Katzenellenbogen JA.

J Steroid Biochem Mol Biol. 2000 Nov 30;74(5):279-85. Review.

PMID:
11162936
17.

18F-labeled difluoroestradiols: preparation and preclinical evaluation as estrogen receptor-binding radiopharmaceuticals.

Seimbille Y, Rousseau J, Bénard F, Morin C, Ali H, Avvakumov G, Hammond GL, van Lier JE.

Steroids. 2002 Aug;67(9):765-75.

PMID:
12123788
18.

Novel Selective Estrogen Receptor Ligand Conjugates Incorporating Endoxifen-Combretastatin and Cyclofenil-Combretastatin Hybrid Scaffolds: Synthesis and Biochemical Evaluation.

Kelly PM, Keely NO, Bright SA, Yassin B, Ana G, Fayne D, Zisterer DM, Meegan MJ.

Molecules. 2017 Aug 31;22(9). pii: E1440. doi: 10.3390/molecules22091440.

19.

Synthesis and biological evaluation of two agents for imaging estrogen receptor β by positron emission tomography: challenges in PET imaging of a low abundance target.

Lee JH, Peters O, Lehmann L, Dence CS, Sharp TL, Carlson KE, Zhou D, Jeyakumar M, Welch MJ, Katzenellenbogen JA.

Nucl Med Biol. 2012 Nov;39(8):1105-16. doi: 10.1016/j.nucmedbio.2012.05.011. Epub 2012 Jun 30.

20.

Estrogen receptor-beta potency-selective ligands: structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues.

Meyers MJ, Sun J, Carlson KE, Marriner GA, Katzenellenbogen BS, Katzenellenbogen JA.

J Med Chem. 2001 Nov 22;44(24):4230-51.

PMID:
11708925

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