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Items: 1 to 20 of 102

1.

Globoidnan A: a lignan from Eucalyptus globoidea inhibits HIV integrase.

Ovenden SP, Yu J, Wan SS, Sberna G, Tait RM, Rhodes D, Cox S, Coates J, Walsh NG, Meurer-Grimes BM.

Phytochemistry. 2004 Dec;65(24):3255-9.

PMID:
15561191
2.

The complestatins as HIV-1 integrase inhibitors. Efficient isolation, structure elucidation, and inhibitory activities of isocomplestatin, chloropeptin I, new complestatins, A and B, and acid-hydrolysis products of chloropeptin I.

Singh SB, Jayasuriya H, Salituro GM, Zink DL, Shafiee A, Heimbuch B, Silverman KC, Lingham RB, Genilloud O, Teran A, Vilella D, Felock P, Hazuda D.

J Nat Prod. 2001 Jul;64(7):874-82.

PMID:
11473415
3.

Isolation, structure and HIV-1 integrase inhibitory activity of exophillic acid, a novel fungal metabolite from Exophiala pisciphila.

Ondeyka JG, Zink DL, Dombrowski AW, Polishook JD, Felock PJ, Hazuda DJ, Singh SB.

J Antibiot (Tokyo). 2003 Dec;56(12):1018-23.

4.

Isolation, structure, and HIV-1 integrase inhibitory activity of Cytosporic acid, a fungal metabolite produced by a Cytospora sp.

Jayasuriya H, Guan Z, Polishook JD, Dombrowski AW, Felock PJ, Hazuda DJ, Singh SB.

J Nat Prod. 2003 Apr;66(4):551-3.

PMID:
12713414
6.

Four novel bis-(naphtho-gamma-pyrones) isolated from Fusarium species as inhibitors of HIV-1 integrase.

Singh SB, Zink DL, Bills GF, Teran A, Silverman KC, Lingham RB, Felock P, Hazuda DJ.

Bioorg Med Chem Lett. 2003 Feb 24;13(4):713-7.

PMID:
12639565
7.

Design and synthesis of substituted 4-oxo-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazine-2-carboxamides, novel HIV-1 integrase inhibitors.

Langford HM, Williams PD, Homnick CF, Vacca JP, Felock PJ, Stillmock KA, Witmer MV, Hazuda DJ, Gabryelski LJ, Schleif WA.

Bioorg Med Chem Lett. 2008 Jan 15;18(2):721-5. Epub 2007 Nov 19.

PMID:
18078751
8.

HIV-1 protease and HIV-1 integrase inhibitory substances from Eclipta prostrata.

Tewtrakul S, Subhadhirasakul S, Cheenpracha S, Karalai C.

Phytother Res. 2007 Nov;21(11):1092-5.

PMID:
17696192
9.

Dissecting Tn5 transposition using HIV-1 integrase diketoacid inhibitors.

Czyz A, Stillmock KA, Hazuda DJ, Reznikoff WS.

Biochemistry. 2007 Sep 25;46(38):10776-89. Epub 2007 Aug 29.

PMID:
17725323
10.

Triketoacid inhibitors of HIV-integrase: a new chemotype useful for probing the integrase pharmacophore.

Walker MA, Johnson T, Ma Z, Banville J, Remillard R, Kim O, Zhang Y, Staab A, Wong H, Torri A, Samanta H, Lin Z, Deminie C, Terry B, Krystal M, Meanwell N.

Bioorg Med Chem Lett. 2006 Jun 1;16(11):2920-4. Epub 2006 Mar 20.

PMID:
16546383
11.

HIV integrase inhibitory activity of Agastache rugosa.

Kim HK, Lee HK, Shin CG, Huh H.

Arch Pharm Res. 1999 Oct;22(5):520-3.

PMID:
10549582
12.

Integracides: tetracyclic triterpenoid inhibitors of HIV-1 integrase produced by Fusarium sp.

Singh SB, Zink DL, Dombrowski AW, Polishook JD, Ondeyka JG, Hirshfield J, Felock P, Hazuda DJ.

Bioorg Med Chem. 2003 Apr 3;11(7):1577-82.

PMID:
12628681
13.

Chromone and chromanone derivatives as strand transfer inhibitors of HIV-1 integrase.

Park JH, Lee SU, Kim SH, Shin SY, Lee JY, Shin CG, Yoo KH, Lee YS.

Arch Pharm Res. 2008 Jan;31(1):1-5.

PMID:
18277599
14.

Discovery of structurally diverse HIV-1 integrase inhibitors based on a chalcone pharmacophore.

Deng J, Sanchez T, Al-Mawsawi LQ, Dayam R, Yunes RA, Garofalo A, Bolger MB, Neamati N.

Bioorg Med Chem. 2007 Jul 15;15(14):4985-5002. Epub 2007 Apr 25.

PMID:
17502148
16.

Peptides derived from the reverse transcriptase of human immunodeficiency virus type 1 as novel inhibitors of the viral integrase.

Oz Gleenberg I, Avidan O, Goldgur Y, Herschhorn A, Hizi A.

J Biol Chem. 2005 Jun 10;280(23):21987-96. Epub 2005 Mar 23.

17.

Discovery of 3-acetyl-4-hydroxy-2-pyranone derivatives and their difluoridoborate complexes as a novel class of HIV-1 integrase inhibitors.

Ramkumar K, Tambov KV, Gundla R, Manaev AV, Yarovenko V, Traven VF, Neamati N.

Bioorg Med Chem. 2008 Oct 1;16(19):8988-98. doi: 10.1016/j.bmc.2008.08.067. Epub 2008 Aug 30. Erratum in: Bioorg Med Chem. 2009 Jan 15;17(2):929. Manaev, Alexandr V [corrected to Manaev, Alexander V].

PMID:
18805696
18.

Novel HIV-1 integrase inhibitors derived from quinolone antibiotics.

Sato M, Motomura T, Aramaki H, Matsuda T, Yamashita M, Ito Y, Kawakami H, Matsuzaki Y, Watanabe W, Yamataka K, Ikeda S, Kodama E, Matsuoka M, Shinkai H.

J Med Chem. 2006 Mar 9;49(5):1506-8.

PMID:
16509568
19.

Dihydroxypyridopyrazine-1,6-dione HIV-1 integrase inhibitors.

Wai JS, Kim B, Fisher TE, Zhuang L, Embrey MW, Williams PD, Staas DD, Culberson C, Lyle TA, Vacca JP, Hazuda DJ, Felock PJ, Schleif WA, Gabryelski LJ, Jin L, Chen IW, Ellis JD, Mallai R, Young SD.

Bioorg Med Chem Lett. 2007 Oct 15;17(20):5595-9. Epub 2007 Aug 22.

PMID:
17822898
20.

Structure, stereochemistry, and biological activity of integramycin, a novel hexacyclic natural product produced by Actinoplanes sp. that inhibits HIV-1 integrase.

Singh SB, Zink DL, Heimbach B, Genilloud O, Teran A, Silverman KC, Lingham RB, Felock P, Hazuda DJ.

Org Lett. 2002 Apr 4;4(7):1123-6.

PMID:
11922798

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