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Items: 1 to 20 of 257

1.

Solid-phase combinatorial synthesis of peptide-biphenyl hybrids as calpain inhibitors.

Montero A, Albericio F, Royo M, Herradón B.

Org Lett. 2004 Oct 28;6(22):4089-92. Erratum in: Org Lett. 2006 Aug 3;8(16):3621.

PMID:
15496106
2.

Studies on aromatic compounds: inhibition of calpain I by biphenyl derivatives and peptide-biphenyl hybrids.

Montero A, Alonso M, Benito E, Chana A, Mann E, Navas JM, Herradón B.

Bioorg Med Chem Lett. 2004 Jun 7;14(11):2753-7.

PMID:
15125927
3.

Peptide-biphenyl hybrids as calpain inhibitors.

Montero A, Mann E, Chana A, Herradón B.

Chem Biodivers. 2004 Mar;1(3):442-57.

PMID:
17191858
4.

Design and synthesis of novel fluoropeptidomimetics as potential mimics of the transition state during peptide hydrolysis.

Annedi SC, Li W, Samson S, Kotra LP.

J Org Chem. 2003 Feb 7;68(3):1043-9. Erratum in: J Org Chem. 2004 Oct 29;69(22):7790.

PMID:
12558433
5.

New renin inhibitors containing novel analogues of statine.

Jones DM, Sueiras-Diaz J, Szelke M, Leckie BJ, Beattie SR, Morton J, Neidle S, Kuroda R.

J Pept Res. 1997 Aug;50(2):109-21.

PMID:
9273895
7.

General inverse solid-phase synthesis method for C-terminally modified peptide mimetics.

Sasubilli R, Gutheil WG.

J Comb Chem. 2004 Nov-Dec;6(6):911-5.

PMID:
15530118
8.

A practical enantioselective synthesis of odanacatib, a potent Cathepsin K inhibitor, via triflate displacement of an alpha-trifluoromethylbenzyl triflate.

O'Shea PD, Chen CY, Gauvreau D, Gosselin F, Hughes G, Nadeau C, Volante RP.

J Org Chem. 2009 Feb 20;74(4):1605-10. doi: 10.1021/jo8020314.

PMID:
19140725
9.
10.

Solid-phase synthesis of a library based on biphenyl-containing trypsin-like serine protease inhibitors.

Shi S, Zhu S, Gerritz SW, Rachwal B, Ruan Z, Hutchins R, Kakarla R, Sofia MJ, Sutton J, Cheney D.

Bioorg Med Chem Lett. 2009 Nov 15;19(22):6477-80. doi: 10.1016/j.bmcl.2009.08.100. Epub 2009 Sep 17.

PMID:
19804972
11.
12.

A nonacid degradable linker for solid-phase synthesis.

Colombo A, De la Figuera N, Fernàndez JC, Fernández-Forner D, Albericio F, Forns P.

Org Lett. 2007 Oct 11;9(21):4319-22. Epub 2007 Sep 15.

PMID:
17867699
13.

Alpha-diketone and alpha-keto ester derivatives of N-protected amino acids and peptides as novel inhibitors of cysteine and serine proteinases.

Angelastro MR, Mehdi S, Burkhart JP, Peet NP, Bey P.

J Med Chem. 1990 Jan;33(1):11-3. No abstract available.

PMID:
2296008
14.

Fmoc solid-phase synthesis of peptide thioesters using an intramolecularn,S-acyl shift.

Ollivier N, Behr JB, El-Mahdi O, Blanpain A, Melnyk O.

Org Lett. 2005 Jun 23;7(13):2647-50.

PMID:
15957912
15.

Ellagitannins and hexahydroxydiphenoyl esters as inhibitors of vertebrate squalene epoxidase.

Abe I, Kashiwagi Y, Noguchi H, Tanaka T, Ikeshiro Y, Kashiwada Y.

J Nat Prod. 2001 Aug;64(8):1010-4.

PMID:
11520216
16.

alpha-Biphenylsulfonylamino 2-methylpropyl phosphonates: enantioselective synthesis and selective inhibition of MMPs.

Biasone A, Tortorella P, Campestre C, Agamennone M, Preziuso S, Chiappini M, Nuti E, Carelli P, Rossello A, Mazza F, Gallina C.

Bioorg Med Chem. 2007 Jan 15;15(2):791-9. Epub 2006 Oct 25.

PMID:
17088065
17.

Developments in the design and synthesis of calpain inhibitors.

Neffe AT, Abell AD.

Curr Opin Drug Discov Devel. 2005 Nov;8(6):684-700. Review.

PMID:
16312145
18.

Novel fluoropeptidomimetics: synthesis, stability studies and protease inhibition.

Annedi SC, Majumder K, Wei L, Oyiliagu CE, Samson S, Kotra LP.

Bioorg Med Chem. 2005 Apr 15;13(8):2943-58. Erratum in: Bioorg Med Chem. 2006 May 1;14(9):3245.

PMID:
15781404
19.

Design and synthesis of 4-quinolinone 2-carboxamides as calpain inhibitors.

Nam DH, Lee KS, Kim SH, Kim SM, Jung SY, Chung SH, Kim HJ, Kim ND, Jin C, Lee YS.

Bioorg Med Chem Lett. 2008 Jan 1;18(1):205-9. Epub 2007 Oct 30.

PMID:
18024028
20.

1,2-Benzothiazine 1,1-dioxide P(2)-P(3) peptide mimetic aldehyde calpain I inhibitors.

Wells GJ, Tao M, Josef KA, Bihovsky R.

J Med Chem. 2001 Oct 11;44(21):3488-503.

PMID:
11585453

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