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Items: 1 to 20 of 159

1.

Site-selective conjugation of thiols with aziridine-2-carboxylic acid-containing peptides.

Galonić DP, van der Donk WA, Gin DY.

J Am Chem Soc. 2004 Oct 13;126(40):12712-3.

PMID:
15469231
2.

Aziridine-2-carboxylic acid-containing peptides: application to solution- and solid-phase convergent site-selective peptide modification.

Galonić DP, Ide ND, van der Donk WA, Gin DY.

J Am Chem Soc. 2005 May 25;127(20):7359-69.

PMID:
15898784
3.

Selective ring-opening of nonactivated amino aziridines by thiols and unusual nucleophilic substitution of a dibenzylamino group.

Concellón JM, Bernad PL, Suárez JR, García-Granda S, Díaz MR.

J Org Chem. 2005 Nov 11;70(23):9411-6.

PMID:
16268615
4.

Aziridine-mediated ligation and site-specific modification of unprotected peptides.

Dyer FB, Park CM, Joseph R, Garner P.

J Am Chem Soc. 2011 Dec 21;133(50):20033-5. doi: 10.1021/ja207133t. Epub 2011 Nov 23.

PMID:
22112239
5.

Chemoselective peptidomimetic ligation using thioacid peptides and aziridine templates.

Assem N, Natarajan A, Yudin AK.

J Am Chem Soc. 2010 Aug 18;132(32):10986-7. doi: 10.1021/ja104488d.

PMID:
20666404
6.

Ring opening of a resin-bound chiral aziridine with phenol nucleophiles.

Ottesen LK, Jaroszewski JW, Franzyk H.

J Org Chem. 2010 Aug 6;75(15):4983-91. doi: 10.1021/jo100505c.

PMID:
20617832
7.

Facile, fmoc-compatible solid-phase synthesis of peptide C-terminal thioesters.

Swinnen D, Hilvert D.

Org Lett. 2000 Aug 10;2(16):2439-42.

PMID:
10956516
8.

Ring opening of pymisyl-protected aziridines with organocuprates.

Bornholdt J, Felding J, Clausen RP, Kristensen JL.

Chemistry. 2010 Nov 2;16(41):12474-80. doi: 10.1002/chem.201001026.

PMID:
20839183
9.

Solid-phase synthesis, cyclization, and site-specific functionalization of aziridine-containing tetrapeptides.

Chung BKW, White CJ, Yudin AK.

Nat Protoc. 2017 Jun;12(6):1277-1287. doi: 10.1038/nprot.2017.035. Epub 2017 May 24.

PMID:
28538738
10.

Synthesis of trifluoromethyl γ-aminophosphonates by nucleophilic aziridine ring opening.

Cytlak T, Saweliew M, Kubicki M, Koroniak H.

Org Biomol Chem. 2015 Oct 21;13(39):10050-9. doi: 10.1039/c5ob01411e.

PMID:
26299334
11.

The stereoselective synthesis of aziridine analogues of diaminopimelic acid (DAP) and their interaction with dap epimerase.

Diaper CM, Sutherland A, Pillai B, James MN, Semchuk P, Blanchard JS, Vederas JC.

Org Biomol Chem. 2005 Dec 21;3(24):4402-11. Epub 2005 Nov 15.

PMID:
16327902
12.

Chemistry of tetrathiomolybdate: aziridine ring opening reactions and facile synthesis of interesting sulfur heterocycles.

Sureshkumar D, Koutha SM, Chandrasekaran S.

J Am Chem Soc. 2005 Sep 21;127(37):12760-1.

PMID:
16159244
13.

Diastereoselective formation of aziridines from diazocarbonyl compounds and N-(O-pivaloylated D-galactosyl)benzylideneamines and ring-opening reactions with p-toluenethiol.

Zhao Y, Wang G, Zhou S, Li Z, Meng X.

Org Biomol Chem. 2014 Jun 7;12(21):3362-5. doi: 10.1039/c4ob00443d. Epub 2014 Apr 22.

PMID:
24752733
14.

Chiral phosphoric acid-catalyzed desymmetrization of meso-aziridines with functionalized mercaptans.

Larson SE, Baso JC, Li G, Antilla JC.

Org Lett. 2009 Nov 19;11(22):5186-9. doi: 10.1021/ol902123h.

15.

Efficient synthesis of taurine and structurally diverse substituted taurines from aziridines.

Hu L, Zhu H, Du DM, Xu J.

J Org Chem. 2007 Jun 8;72(12):4543-6. Epub 2007 May 12.

PMID:
17497929
16.

Toward tubulysin: gram-scale synthesis of tubuvaline-tubuphenylalanine fragment.

Chandrasekhar S, Mahipal B, Kavitha M.

J Org Chem. 2009 Dec 18;74(24):9531-4. doi: 10.1021/jo9015503.

PMID:
19928810
17.

An efficient copper-catalyzed synthesis of hexahydro-1H- phenothiazines.

Prasad DJ, Sekar G.

Org Biomol Chem. 2009 Dec 21;7(24):5091-7. doi: 10.1039/b916664e. Epub 2009 Oct 23.

PMID:
20024103
18.

Amine-promoted synthesis of vinyl aziridines.

Armstrong A, Pullin RD, Jenner CR, Scutt JN.

J Org Chem. 2010 May 21;75(10):3499-502. doi: 10.1021/jo100407s.

PMID:
20465292
19.

Solid-phase synthesis of peptide and glycopeptide thioesters through side-chain-anchoring strategies.

Ficht S, Payne RJ, Guy RT, Wong CH.

Chemistry. 2008;14(12):3620-9. doi: 10.1002/chem.200701978.

PMID:
18278777
20.

Conformational modulation of in vitro activity of cyclic RGD peptides via aziridine aldehyde-driven macrocyclization chemistry.

Roxin Á, Chen J, Scully CC, Rotstein BH, Yudin AK, Zheng G.

Bioconjug Chem. 2012 Jul 18;23(7):1387-95. doi: 10.1021/bc300239a. Epub 2012 Jun 25.

PMID:
22709546

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