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Items: 1 to 20 of 151

1.
2.

Novel cyclopentanone derivatives pentenocins A and B with interleukin-1beta converting enzyme inhibitory activity, produced by Trichoderma hamatum FO-6903.

Matsumoto T, Ishiyama A, Yamaguchi Y, Masuma R, Ui H, Shiomi K, Yamada H, Omura S.

J Antibiot (Tokyo). 1999 Aug;52(8):754-7. No abstract available. Erratum in: J Antibiot (Tokyo). 2003 May;56(5):C-2.

3.

First synthesis and structural elucidation of (-)-presphaerene.

Lee J, Hong J.

J Org Chem. 2004 Sep 17;69(19):6433-40.

PMID:
15357605
4.

Peptidomimetic aminomethylene ketone inhibitors of interleukin-1 beta-converting enzyme (ICE).

Semple G, Ashworth DM, Batt AR, Baxter AJ, Benzies DW, Elliot LH, Evans DM, Franklin RJ, Hudson P, Jenkins PD, Pitt GR, Rooker DP, Yamamoto S, Isomura Y.

Bioorg Med Chem Lett. 1998 Apr 21;8(8):959-64.

PMID:
9871520
5.

Conformationally constrained inhibitors of caspase-1 (interleukin-1 beta converting enzyme) and of the human CED-3 homologue caspase-3 (CPP32, apopain).

Karanewsky DS, Bai X, Linton SD, Krebs JF, Wu J, Pham B, Tomaselli KJ.

Bioorg Med Chem Lett. 1998 Oct 6;8(19):2757-62.

PMID:
9873617
7.

Solid-phase synthesis of azidomethylene inhibitors targeting cysteine proteases.

Yang PY, Wu H, Lee MY, Xu A, Srinivasan R, Yao SQ.

Org Lett. 2008 May 15;10(10):1881-4. doi: 10.1021/ol800575z. Epub 2008 Apr 12.

PMID:
18407644
8.

Succinic acid amides as P2-P3 replacements for inhibitors of interleukin-1beta converting enzyme (ICE or caspase 1).

Galatsis P, Caprathe B, Gilmore J, Thomas A, Linn K, Sheehan S, Harter W, Kostlan C, Lunney E, Stankovic C, Rubin J, Brady K, Allen H, Talanian R.

Bioorg Med Chem Lett. 2010 Sep 1;20(17):5184-90. doi: 10.1016/j.bmcl.2010.07.004. Epub 2010 Jul 8.

PMID:
20656488
9.

First examples of peptidomimetic inhibitors of interleukin-1 beta converting enzyme.

Dolle RE, Prouty CP, Prasad CV, Cook E, Saha A, Ross TM, Salvino JM, Helaszek CT, Ator MA.

J Med Chem. 1996 Jun 21;39(13):2438-40. No abstract available.

PMID:
8691439
10.

EI-1507-1 and -2, novel interleukin-1 beta converting enzyme inhibitors produced by Streptomyces sp. E-1507.

Tsukuda E, Tanaka T, Ochiai K, Kondo H, Yoshida M, Agatsuma T, Saitoh Y, Teshiba S, Matsuda Y.

J Antibiot (Tokyo). 1996 Apr;49(4):333-9.

11.

Structure-based design of nonpeptide inhibitors of interleukin-1beta converting enzyme (ICE, caspase-1).

Shahripour AB, Plummer MS, Lunney EA, Albrecht HP, Hays SJ, Kostlan CR, Sawyer TK, Walker NP, Brady KD, Allen HJ, Talanian RV, Wong WW, Humblet C.

Bioorg Med Chem. 2002 Jan;10(1):31-40.

PMID:
11738604
12.

Rapid optimization of an ICE inhibitor synthesis using multiple reaction conditions in a parallel array.

Warmus JS, Ryder TR, Hodges JC, Kennedy RM, Brady KD.

Bioorg Med Chem Lett. 1998 Sep 8;8(17):2309-14.

PMID:
9873533
13.

Serine and threonine beta-lactones: a new class of hepatitis A virus 3C cysteine proteinase inhibitors.

Lall MS, Ramtohul YK, James MN, Vederas JC.

J Org Chem. 2002 Mar 8;67(5):1536-47.

PMID:
11871884
15.

Total synthesis of plakortone B.

Xie XG, Wu XW, Lee HK, Peng XS, Wong HN.

Chemistry. 2010 Jun 18;16(23):6933-41. doi: 10.1002/chem.201000189.

PMID:
20432418
16.

Noncovalent tripeptidyl benzyl- and cyclohexyl-amine inhibitors of the cysteine protease caspase-1.

Löser R, Abbenante G, Madala PK, Halili M, Le GT, Fairlie DP.

J Med Chem. 2010 Mar 25;53(6):2651-5. doi: 10.1021/jm901790w.

PMID:
20170165
17.

Enzyme-assisted enantioselective synthesis of natural (-)-beta-necrodol and its enantiomer.

Galano JM, Audran G, Mikolajèzyk L, Monti H.

J Org Chem. 2001 Jan 12;66(1):323-6. No abstract available.

PMID:
11429920
18.

Organic azide inhibitors of cysteine proteases.

Le GT, Abbenante G, Madala PK, Hoang HN, Fairlie DP.

J Am Chem Soc. 2006 Sep 27;128(38):12396-7. Erratum in: J Am Chem Soc. 2007 Aug 1;129(30):9532.

PMID:
16984172
19.
20.

Functionalised 2,3-dimethyl-3-aminotetrahydrofuran-4-one and N-(3-oxo-hexahydrocyclopenta[b]furan-3a-yl)acylamide based scaffolds: synthesis and cysteinyl proteinase inhibition.

Watts J, Benn A, Flinn N, Monk T, Ramjee M, Ray P, Wang Y, Quibell M.

Bioorg Med Chem. 2004 Jun 1;12(11):2903-25. Erratum in: Bioorg Med Chem. 2005 Sep 15;13(18):5502.

PMID:
15142551

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