Similar articles for PMID: 14516196

Year	Number of Results
1994	5
1995	2
1996	2
1997	4
1998	9
1999	7
2000	16
2001	11
2002	26
2003	33
2004	21
2005	22
2006	30
2007	16
2008	6
2009	11
2010	20
2011	24
2012	20
2013	16
2014	19
2015	16
2016	8
2017	11
2018	9
2019	8
2020	3
2021	6
2022	6
2023	1
2024	0

1

The structural basis for the selectivity of benzotriazole inhibitors of PTP1B.

Scapin G, Patel SB, Becker JW, Wang Q, Desponts C, Waddleton D, Skorey K, Cromlish W, Bayly C, Therien M, Gauthier JY, Li CS, Lau CK, Ramachandran C, Kennedy BP, Asante-Appiah E. Scapin G, et al. Biochemistry. 2003 Oct 7;42(39):11451-9. doi: 10.1021/bi035098j. Biochemistry. 2003. PMID: 14516196

2

Small molecule interactions with protein-tyrosine phosphatase PTP1B and their use in inhibitor design.

Burke TR Jr, Ye B, Yan X, Wang S, Jia Z, Chen L, Zhang ZY, Barford D. Burke TR Jr, et al. Biochemistry. 1996 Dec 17;35(50):15989-96. doi: 10.1021/bi961256d. Biochemistry. 1996. PMID: 8973169

3

Selective protein tyrosine phosphatase 1B inhibitors: targeting the second phosphotyrosine binding site with non-carboxylic acid-containing ligands.

Liu G, Xin Z, Liang H, Abad-Zapatero C, Hajduk PJ, Janowick DA, Szczepankiewicz BG, Pei Z, Hutchins CW, Ballaron SJ, Stashko MA, Lubben TH, Berg CE, Rondinone CM, Trevillyan JM, Jirousek MR. Liu G, et al. J Med Chem. 2003 Jul 31;46(16):3437-40. doi: 10.1021/jm034088d. J Med Chem. 2003. PMID: 12877578

4

Discovery of a potent, selective protein tyrosine phosphatase 1B inhibitor using a linked-fragment strategy.

Szczepankiewicz BG, Liu G, Hajduk PJ, Abad-Zapatero C, Pei Z, Xin Z, Lubben TH, Trevillyan JM, Stashko MA, Ballaron SJ, Liang H, Huang F, Hutchins CW, Fesik SW, Jirousek MR. Szczepankiewicz BG, et al. J Am Chem Soc. 2003 Apr 9;125(14):4087-96. doi: 10.1021/ja0296733. J Am Chem Soc. 2003. PMID: 12670229

5

PTP1B as a drug target: recent developments in PTP1B inhibitor discovery.

Zhang S, Zhang ZY. Zhang S, et al. Drug Discov Today. 2007 May;12(9-10):373-81. doi: 10.1016/j.drudis.2007.03.011. Epub 2007 Apr 6. Drug Discov Today. 2007. PMID: 17467573 Review.

6

Allele-specific inhibitors of protein tyrosine phosphatases.

Hoffman HE, Blair ER, Johndrow JE, Bishop AC. Hoffman HE, et al. J Am Chem Soc. 2005 Mar 9;127(9):2824-5. doi: 10.1021/ja043378w. J Am Chem Soc. 2005. PMID: 15740097

7

Monocyclic thiophenes as protein tyrosine phosphatase 1B inhibitors: capturing interactions with Asp48.

Wan ZK, Lee J, Xu W, Erbe DV, Joseph-McCarthy D, Follows BC, Zhang YL. Wan ZK, et al. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4941-5. doi: 10.1016/j.bmcl.2006.06.051. Epub 2006 Jun 27. Bioorg Med Chem Lett. 2006. PMID: 16806920

8

Development of a robust scintillation proximity assay for protein tyrosine phosphatase 1B using the catalytically inactive (C215S) mutant.

Skorey KI, Kennedy BP, Friesen RW, Ramachandran C. Skorey KI, et al. Anal Biochem. 2001 Apr 15;291(2):269-78. doi: 10.1006/abio.2001.5029. Anal Biochem. 2001. PMID: 11401301

9

Structure-based optimization of protein tyrosine phosphatase 1B inhibitors: from the active site to the second phosphotyrosine binding site.

Wilson DP, Wan ZK, Xu WX, Kirincich SJ, Follows BC, Joseph-McCarthy D, Foreman K, Moretto A, Wu J, Zhu M, Binnun E, Zhang YL, Tam M, Erbe DV, Tobin J, Xu X, Leung L, Shilling A, Tam SY, Mansour TS, Lee J. Wilson DP, et al. J Med Chem. 2007 Sep 20;50(19):4681-98. doi: 10.1021/jm0702478. Epub 2007 Aug 17. J Med Chem. 2007. PMID: 17705360

10

Structure-based optimization of benzoic acids as inhibitors of protein tyrosine phosphatase 1B and low molecular weight protein tyrosine phosphatase.

Maccari R, Ottanà R, Ciurleo R, Paoli P, Manao G, Camici G, Laggner C, Langer T. Maccari R, et al. ChemMedChem. 2009 Jun;4(6):957-62. doi: 10.1002/cmdc.200800427. ChemMedChem. 2009. PMID: 19288492

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