Similar articles for PMID: 12941329

Year	Number of Results
1956	1
1974	1
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1999	5
2000	6
2001	12
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1

Adenosine kinase inhibitors: polar 7-substitutent of pyridopyrimidine derivatives improving their locomotor selectivity.

Zheng GZ, Mao Y, Lee CH, Pratt JK, Koenig JR, Perner RJ, Cowart MD, Gfesser GA, McGaraughty S, Chu KL, Zhu C, Yu H, Kohlhaas K, Alexander KM, Wismer CT, Mikusa J, Jarvis MF, Kowaluk EA, Stewart AO. Zheng GZ, et al. Bioorg Med Chem Lett. 2003 Sep 15;13(18):3041-4. doi: 10.1016/s0960-894x(03)00642-5. Bioorg Med Chem Lett. 2003. PMID: 12941329

2

Structure-activity studies of 5-substituted pyridopyrimidines as adenosine kinase inhibitors.

Cowart M, Lee CH, Gfesser GA, Bayburt EK, Bhagwat SS, Stewart AO, Yu H, Kohlhaas KL, McGaraughty S, Wismer CT, Mikusa J, Zhu C, Alexander KM, Jarvis MF, Kowaluk EA. Cowart M, et al. Bioorg Med Chem Lett. 2001 Jan 8;11(1):83-6. doi: 10.1016/s0960-894x(00)00602-8. Bioorg Med Chem Lett. 2001. PMID: 11140740

3

Synthesis and biological evaluation of 6,7-disubstituted 4-aminopyrido[2,3-d]pyrimidines as adenosine kinase inhibitors.

Perner RJ, Lee CH, Jiang M, Gu YG, Didomenico S, Bayburt EK, Alexander KM, Kohlhaas KL, Jarvis MF, Kowaluk EL, Bhagwat SS. Perner RJ, et al. Bioorg Med Chem Lett. 2005 Jun 2;15(11):2803-7. doi: 10.1016/j.bmcl.2005.03.098. Epub 2005 Apr 25. Bioorg Med Chem Lett. 2005. PMID: 15911258

4

5,6,7-trisubstituted 4-aminopyrido[2,3-d]pyrimidines as novel inhibitors of adenosine kinase.

Perner RJ, Gu YG, Lee CH, Bayburt EK, McKie J, Alexander KM, Kohlhaas KL, Wismer CT, Mikusa J, Jarvis MF, Kowaluk EA, Bhagwat SS. Perner RJ, et al. J Med Chem. 2003 Nov 20;46(24):5249-57. doi: 10.1021/jm030327l. J Med Chem. 2003. PMID: 14613327

5

Pyridopyrimidine analogues as novel adenosine kinase inhibitors.

Zheng GZ, Lee C, Pratt JK, Perner RJ, Jiang MQ, Gomtsyan A, Matulenko MA, Mao Y, Koenig JR, Kim KH, Muchmore S, Yu H, Kohlhaas K, Alexander KM, McGaraughty S, Chu KL, Wismer CT, Mikusa J, Jarvis MF, Marsh K, Kowaluk EA, Bhagwat SS, Stewart AO. Zheng GZ, et al. Bioorg Med Chem Lett. 2001 Aug 20;11(16):2071-4. doi: 10.1016/s0960-894x(01)00375-4. Bioorg Med Chem Lett. 2001. PMID: 11514141

6

Analgesic and anti-inflammatory effects of A-286501, a novel orally active adenosine kinase inhibitor.

Jarvis MF, Yu H, McGaraughty S, Wismer CT, Mikusa J, Zhu C, Chu K, Kohlhaas K, Cowart M, Lee CH, Stewart AO, Cox BF, Polakowski J, Kowaluk EA. Jarvis MF, et al. Pain. 2002 Mar;96(1-2):107-18. doi: 10.1016/s0304-3959(01)00435-3. Pain. 2002. PMID: 11932067

7

Design, synthesis, and structure-activity relationship of 6-alkynylpyrimidines as potent adenosine kinase inhibitors.

Gomtsyan A, Didomenico S, Lee CH, Matulenko MA, Kim K, Kowaluk EA, Wismer CT, Mikusa J, Yu H, Kohlhaas K, Jarvis MF, Bhagwat SS. Gomtsyan A, et al. J Med Chem. 2002 Aug 15;45(17):3639-48. doi: 10.1021/jm020049a. J Med Chem. 2002. PMID: 12166937

8

Recent developments in the discovery of novel adenosine kinase inhibitors: mechanism of action and therapeutic potential.

McGaraughty S, Cowart M, Jarvis MF. McGaraughty S, et al. CNS Drug Rev. 2001 Winter;7(4):415-32. doi: 10.1111/j.1527-3458.2001.tb00208.x. CNS Drug Rev. 2001. PMID: 11830758 Free PMC article. Review.

9

Synthesis and structure-activity relationships of 5-heteroatom-substituted pyridopyrimidines as adenosine kinase inhibitors.

Gfesser GA, Bayburt EK, Cowart M, DiDomenico S, Gomtsyan A, Lee CH, Stewart AO, Jarvis MF, Kowaluk EA, Bhagwat SS. Gfesser GA, et al. Eur J Med Chem. 2003 Mar;38(3):245-52. doi: 10.1016/s0223-5234(03)00019-9. Eur J Med Chem. 2003. PMID: 12667691

10

ABT-702 (4-amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin- 3-yl)pyrido[2,3-d]pyrimidine), a novel orally effective adenosine kinase inhibitor with analgesic and anti-inflammatory properties. II. In vivo characterization in the rat.

Kowaluk EA, Mikusa J, Wismer CT, Zhu CZ, Schweitzer E, Lynch JJ, Lee CH, Jiang M, Bhagwat SS, Gomtsyan A, McKie J, Cox BF, Polakowski J, Reinhart G, Williams M, Jarvis MF. Kowaluk EA, et al. J Pharmacol Exp Ther. 2000 Dec;295(3):1165-74. J Pharmacol Exp Ther. 2000. PMID: 11082454

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