Similar articles for PMID: 12517430

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1

2-Phenylimidazo[2,1-i]purin-5-ones: structure-activity relationships and characterization of potent and selective inverse agonists at Human A3 adenosine receptors.

Ozola V, Thorand M, Diekmann M, Qurishi R, Schumacher B, Jacobson KA, Müller CE. Ozola V, et al. Bioorg Med Chem. 2003 Feb 6;11(3):347-56. doi: 10.1016/s0968-0896(02)00456-x. Bioorg Med Chem. 2003. PMID: 12517430 Free PMC article.

2

Imidazo[2,1-i]purin-5-ones and related tricyclic water-soluble purine derivatives: potent A(2A)- and A(3)-adenosine receptor antagonists.

Müller CE, Thorand M, Qurishi R, Diekmann M, Jacobson KA, Padgett WL, Daly JW. Müller CE, et al. J Med Chem. 2002 Aug 1;45(16):3440-50. doi: 10.1021/jm011093d. J Med Chem. 2002. PMID: 12139454 Free PMC article.

3

1,8-disubstituted xanthine derivatives: synthesis of potent A2B-selective adenosine receptor antagonists.

Hayallah AM, Sandoval-Ramírez J, Reith U, Schobert U, Preiss B, Schumacher B, Daly JW, Müller CE. Hayallah AM, et al. J Med Chem. 2002 Mar 28;45(7):1500-10. doi: 10.1021/jm011049y. J Med Chem. 2002. PMID: 11906291

4

Selective allosteric enhancement of agonist binding and function at human A3 adenosine receptors by a series of imidazoquinoline derivatives.

Gao ZG, Kim SG, Soltysiak KA, Melman N, IJzerman AP, Jacobson KA. Gao ZG, et al. Mol Pharmacol. 2002 Jul;62(1):81-9. doi: 10.1124/mol.62.1.81. Mol Pharmacol. 2002. PMID: 12065758 Free PMC article.

5

New 2-heterocyclyl-imidazo[2,1-i]purin-5-one derivatives as potent and selective human A3 adenosine receptor antagonists.

Baraldi PG, Preti D, Zaid AN, Saponaro G, Tabrizi MA, Baraldi S, Romagnoli R, Moorman AR, Varani K, Cosconati S, Di Maro S, Marinelli L, Novellino E, Borea PA. Baraldi PG, et al. J Med Chem. 2011 Jul 28;54(14):5205-20. doi: 10.1021/jm2004738. Epub 2011 Jun 28. J Med Chem. 2011. PMID: 21675777

6

[(3)H]8-Ethyl-4-methyl-2-phenyl-(8R)-4,5,7,8-tetrahydro-1H-imidazo[2,1-i]-purin-5-one ([(3)H]PSB-11), a novel high-affinity antagonist radioligand for human A(3) adenosine receptors.

Müller CE, Diekmann M, Thorand M, Ozola V. Müller CE, et al. Bioorg Med Chem Lett. 2002 Feb 11;12(3):501-3. doi: 10.1016/s0960-894x(01)00785-5. Bioorg Med Chem Lett. 2002. PMID: 11814828

7

Synthesis and biological activity of a new series of N6-arylcarbamoyl, 2-(Ar)alkynyl-N6-arylcarbamoyl, and N6-carboxamido derivatives of adenosine-5'-N-ethyluronamide as A1 and A3 adenosine receptor agonists.

Baraldi PG, Cacciari B, Pineda de Las Infantas MJ, Romagnoli R, Spalluto G, Volpini R, Costanzi S, Vittori S, Cristalli G, Melman N, Park KS, Ji XD, Jacobson KA. Baraldi PG, et al. J Med Chem. 1998 Aug 13;41(17):3174-85. doi: 10.1021/jm980147p. J Med Chem. 1998. PMID: 9703463 Free PMC article.

8

N6-Substituted adenosine derivatives: selectivity, efficacy, and species differences at A3 adenosine receptors.

Gao ZG, Blaustein JB, Gross AS, Melman N, Jacobson KA. Gao ZG, et al. Biochem Pharmacol. 2003 May 15;65(10):1675-84. doi: 10.1016/s0006-2952(03)00153-9. Biochem Pharmacol. 2003. PMID: 12754103 Free PMC article.

9

Design, synthesis, and biological evaluation of new 8-heterocyclic xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists.

Baraldi PG, Tabrizi MA, Preti D, Bovero A, Romagnoli R, Fruttarolo F, Zaid NA, Moorman AR, Varani K, Gessi S, Merighi S, Borea PA. Baraldi PG, et al. J Med Chem. 2004 Mar 11;47(6):1434-47. doi: 10.1021/jm0309654. J Med Chem. 2004. PMID: 14998332

10

2-Substituted adenosine derivatives: affinity and efficacy at four subtypes of human adenosine receptors.

Gao ZG, Mamedova LK, Chen P, Jacobson KA. Gao ZG, et al. Biochem Pharmacol. 2004 Nov 15;68(10):1985-93. doi: 10.1016/j.bcp.2004.06.011. Biochem Pharmacol. 2004. PMID: 15476669 Free PMC article.

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