Similar articles for PMID: 12057635

Year	Number of Results
1993	4
1994	2
1995	4
1996	6
1997	5
1998	14
1999	7
2000	11
2001	12
2002	8
2003	5
2004	4
2005	1
2008	3
2009	1
2010	2
2011	1
2017	1
2024	0

1

6-Carboxy-5,7-diarylcyclopenteno[1,2-b]pyridine derivatives: a novel class of endothelin receptor antagonists.

Niiyama K, Mase T, Takahashi H, Naya A, Katsuki K, Nagase T, Ito S, Hayama T, Hisaka A, Ozaki S, Ihara M, Yano M, Fukuroda T, Noguchi K, Nishikibe M, Ishikawa K. Niiyama K, et al. Bioorg Med Chem. 2002 Aug;10(8):2461-70. doi: 10.1016/s0968-0896(02)00122-0. Bioorg Med Chem. 2002. PMID: 12057635

2

Structure-Activity relationships of 2-substituted 5,7-Diarylcyclopenteno[1,2-b]pyridine-6-carboxylic acids as a novel class of endothelin receptor antagonists.

Niiyama K, Takahashi H, Nagase T, Kojima H, Amano Y, Katsuki K, Yamakawa T, Ozaki S, Ihara M, Yano M, Fukuroda T, Nishikibe M, Ishikawa K. Niiyama K, et al. Bioorg Med Chem Lett. 2002 Nov 4;12(21):3041-5. doi: 10.1016/s0960-894x(02)00663-7. Bioorg Med Chem Lett. 2002. PMID: 12372497

3

Structure-activity relationships of a novel class of endothelin receptor selective antagonists; 6-carboxy-2-isopropylamino-5,7-diarylcyclopenteno[1,2-b]pyridines.

Takahashi H, Ohtake N, Sakamoto T, Iino T, Kawanishi N, Nakamura M, Yoshizumi T, Niiyama K, Ozaki S, Okada H, Kano A, Takahashi H, Ishii Y, Okada M, Saito M, Sawazaki Y, Hayama T, Nishikibe M. Takahashi H, et al. Bioorg Med Chem Lett. 2004 Mar 22;14(6):1503-7. doi: 10.1016/j.bmcl.2004.01.008. Bioorg Med Chem Lett. 2004. PMID: 15006391

4

Benzofuro[3,2-b]pyridines as mixed ET(A)/ET(B) and selective ET(B) endothelin receptor antagonists.

Mederski WW, Osswald M, Dorsch D, Christadler M, Schmitges CJ, Wilm C. Mederski WW, et al. Bioorg Med Chem Lett. 1999 Feb 22;9(4):619-22. doi: 10.1016/s0960-894x(99)00040-2. Bioorg Med Chem Lett. 1999. PMID: 10098676

5

Structure-activity relationships of a novel class of endothelin-A receptor antagonists and discovery of potent and selective receptor antagonist, 2-(benzo[1,3]dioxol-5-yl)-6-isopropyloxy-4-(4-methoxyphenyl)-2H-chromene-3-carboxylic acid (S-1255). 1. Study on structure-activity relationships and basic structure crucial for ET(A) antagonism.

Ishizuka N, Matsumura K, Sakai K, Fujimoto M, Mihara S, Yamamori T. Ishizuka N, et al. J Med Chem. 2002 May 9;45(10):2041-55. doi: 10.1021/jm010382z. J Med Chem. 2002. PMID: 11985472

6

Pharmacological properties of J-104132 (L-753,037), a potent, orally active, mixed ETA/ETB endothelin receptor antagonist.

Nishikibe M, Ohta H, Okada M, Ishikawa K, Hayama T, Fukuroda T, Noguchi K, Saito M, Kanoh T, Ozaki S, Kamei T, Hara K, William D, Kivlighn S, Krause S, Gabel R, Zingaro G, Nolan N, O'Brien J, Clayton F, Lynch J, Pettibone D, Siegl P. Nishikibe M, et al. J Pharmacol Exp Ther. 1999 Jun;289(3):1262-70. J Pharmacol Exp Ther. 1999. PMID: 10336515

7

Potent and orally active ET(A) selective antagonists with 5,7-diarylcyclopenteno[1,2-b]pyridine-6-carboxylic acid structures.

Yoshizumi T, Takahashi H, Ohtake N, Jona H, Sato Y, Kishino H, Sakamoto T, Ozaki S, Takahashi H, Shibata Y, Ishii Y, Saito M, Okada M, Hayama T, Nishikibe M. Yoshizumi T, et al. Bioorg Med Chem. 2004 May 1;12(9):2139-50. doi: 10.1016/j.bmc.2004.02.033. Bioorg Med Chem. 2004. PMID: 15080914

8

Pharmacology of L-744,453, a novel nonpeptidyl endothelin antagonist.

Williams DL Jr, Murphy KL, Nolan NA, O'Brien JA, Lis EV Jr, Pettibone DJ, Clineschmidt BV, Krause SM, Veber DF, Naylor EM, Chakravarty PK, Walsh TF, Dhanoa DM, Chen A, Bagley SW, Fitch KJ, Greenlee WJ. Williams DL Jr, et al. Life Sci. 1996;58(14):1149-57. doi: 10.1016/0024-3205(96)00073-2. Life Sci. 1996. PMID: 8614266

9

In vivo labeling of endothelin receptors with [(11)C]L-753,037: studies in mice and a dog.

Aleksic S, Szabo Z, Scheffel U, Ravert HT, Mathews WB, Kerenyi L, Rauseo PA, Gibson RE, Burns HD, Dannals RF. Aleksic S, et al. J Nucl Med. 2001 Aug;42(8):1274-80. J Nucl Med. 2001. PMID: 11483691 Free article.

10

Selective endothelin A receptor antagonists. 3. Discovery and structure-activity relationships of a series of 4-phenoxybutanoic acid derivatives.

Astles PC, Brealey C, Brown TJ, Facchini V, Handscombe C, Harris NV, McCarthy C, McLay IM, Porter B, Roach AG, Sargent C, Smith C, Walsh RJ. Astles PC, et al. J Med Chem. 1998 Jul 16;41(15):2732-44. doi: 10.1021/jm9707131. J Med Chem. 1998. PMID: 9667964

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

90 results

Results by year